关于 "LPA Receptor" 的结果28+ 个结果

A potent LPA receptor agonist

An LPA mimetic and LPA receptor agonist

A stable pan-antagonist at LPA receptors

Galanin Receptor Ligand M35 是一种高亲和力的甘丙肽受体配体，在大鼠脊髓、大鼠海马和离体小鼠胰岛中起着甘丙肽受体拮抗剂的作用。Galanin Receptor Ligand M35 对人 GalR1 和 GalR2 的 Ki 值分别为 0.11 nM、2.0 nM。

C34是一种可口服的Toll样受体4(TLR4)选择性拮抗剂，C34通过抑制TLR4/MyD88/NF-κB信号通路，减少促炎细胞因子的产生，从而发挥抗炎作用。

C3a Receptor Agonist是一种选择性的补体3a受体（C3aR）特异性激动剂。

A TGR5 agonist

Leptin Binding Domain Human Recombinant

Leptin Receptor Chicken Recombinant

Soluble RANK Receptor Human Recombinant

干扰素受体激动剂（化合物 6）是一种干扰素 (IFN) 受体诱导剂。

A2Areceptorantagonist1是adenosineA2Areceptor和A1receptor的拮抗剂,Ki值分别为4和264nM。

GABAA receptor agent 1 is a high affinity ligand for Gamma-aminobutyric acid A (GABAA) receptor that exerts potent anticonvulsant activity.

The peptide T1, MSRPACPNDKYE, is based on the sequence of the thrombin receptor domain that functions as a tethered ligand for the receptor itself. T1 has been selected from a phage peptide library as an inhibitor of thrombin triggered platelet aggregation, serotonin release and tyrosine phosphorylation. Its anti-aggregatory activity was about ten-fold higher than that of the previously reported peptide antagonists of the thrombin receptor. MSRPACPNDKYE has served as model peptide in protein modification and MS studies.

A GCGR antagonist

cFMS Receptor Inhibitor IV (Compound 42) 是一种有效的 cFMS 抑制剂，IC50 为 0.017 μM。

An orexin 2 receptor agonist

An AT 2 receptor agonist

A2Breceptorantagonist1是一个有效的A2B腺苷受体(A2Badenosinereceptor)拮抗剂，来自专利WO2009157938A1实例9B。

H3receptor-MO-1是一种组胺H3受体(histamineH3receptor)调节剂。

H3receptorantagonist1是组胺H3(histamineH3)受体拮抗剂，可用于神经疾病的研究。

S1p receptor agonist 1 是一种有效且具有口服活性的 S1P 受体激动剂，具有诱导 S1P1 内化的活性 (EC50=9.83 nM)。

Androgenreceptorantagonist1是一种口服有效的完整雄激素受体(AR)拮抗剂，IC50为59nM。Androgenreceptorantagonist1可用于合成PROTACAR降解剂，1μM和10μMPROTACAR降解剂作用于LNCaP细胞，分别导致24%和47%AR蛋白降解。

糖皮质激素受体激动剂是一种有效的糖皮质激素受体激动剂。