关于 "Antibiotic" 的结果30 个结果
| 货号 | 产品名称 | CAS 号 | 靶点 | 化学结构 |
|---|---|---|---|---|
| GC31586 | Monacolin J (Antibiotic MB 530A) | 79952-42-4 | HMG-CoA ReductaseAutophagy | |
Monacolin J (Antibiotic MB 530A) 是一种胆固醇生物合成抑制剂,可抑制 HMG-CoA 还原酶的活性。 | ||||
| GC92249 | MRSA Antibiotic 2 | 667410-02-8 | — | |
MRSA antibiotic 2 is an antibiotic. | ||||
| GC45383 | Antibiotic PF 1052 | 147317-15-5 | Natural ProductsImmunology/InflammationFood-Borne Illnesses | |
A fungal metabolite | ||||
| GC32220 | Antibiotic-5d | 251349-54-9 | Bacterial | |
Antibiotic-5d是一种合成的抗微生物化合物。 | ||||
| GF16717 | antibiotics-antimycotic | — | — | |
| GC26403 | G418 Selective Antibiotic, Sterile | — | — | |
G418 Selective Antibiotic, Sterile G418、G 418或者G-418,是一种结构类似于庆大霉素B1 (Gentamycin B1)的氨基糖苷类抗生素,常用于筛选表达neo基因的真核或原核多克隆或单克隆细胞。 | ||||
| GC91670 | MRSA Antibiotic 1 | 667410-81-3 | AntibioticMRSAImmunology/Inflammation | |
MRSA antibiotic 1 is an antibiotic. | ||||
| GC48226 | Urdamycin A | 98474-21-6 | Natural ProductsImmunology/InflammationBacterial DiseasesCancer Biology | |
A bacterial metabolite | ||||
| GC47924 | Parvodicin C2 | 110882-85-4 | Natural ProductsImmunology/InflammationMRSA | |
A glycopeptide antibiotic | ||||
| GC48533 | Vanoxonin | 86933-99-5 | Natural ProductsApoptosisDNA/RNA Synthesis | |
A bacterial metabolite | ||||
| GC60668 | Calcimycin hemimagnesium | 72124-77-7 | ApoptosisBacterialAutophagyFungal | |
Calcimycin(A-23187)hemimagnesium是一种抗生素和独特的二价阳离子离子载体(divalentcationionophore),如钙离子和镁离子。Calcimycinhemimagnesium通过增加细胞内钙浓度诱导Ca2+依赖性细胞死亡。Calcimycinhemimagnesium抑制革兰氏阳性细菌和一些真菌的生长,还抑制ATP酶的活性并解耦哺乳动物细胞的氧化磷酸化(OXPHOS),诱导细胞凋亡(apoptosis)。 | ||||
| GC18936 | A-83016F | 142435-72-1 | Natural ProductsImmunology/InflammationPneumonia | |
An aurodox antibiotic | ||||
| GC63650 | Pentachloropseudilin | 69640-38-6 | Myosin | |
Pentachloropseudilin (Antibiotic A 15104 Y; PClP) 是一种可逆的、变构有效的肌球蛋白 (Myo1s) 抑制剂,对 Myo1s 的 IC50 范围为 1 至 5 μM,对于 2 类和 5 类肌球蛋白,IC50 范围 > 90 μM。Pentachloropseudilin 是转化生长因子-β (TGF-β) 刺激的信号传导的有效抑制剂,对 TGF-β 的 IC50 值为 0.1-0.2 μM。 | ||||
| GC17519 | Concanamycin A | 80890-47-7 | AutophagyProton Pump | |
Concanamycin A 是液泡型 ATP 酶 (V-ATPase) 的特异性抑制剂,IC50 值为 10 nM 。 | ||||
| GC43882 | Hygrolidin | 83329-73-1 | AntibioticADC CytotoxinFungal | |
A macrocyclic lactone | ||||
| GC43883 | Hymeglusin | 29066-42-0 | Natural ProductsInnate ImmunityCholesterol MetabolismBacterial Diseases | |
An HMG-CoA synthase inhibitor | ||||
| GC42888 | Azamulin | 76530-44-4 | P450 | |
A selective CYP3A inhibitor | ||||
| GC45514 | Micronomicin (sulfate) | 66803-19-8 | AntibioticBacterial | |
An aminoglycoside antibiotic | ||||
| GC15299 | Staurosporine(CGP 41251) | 62996-74-1 | PKCBroad Spectrum Protein Kinase InhibitorPKA | |
Staurosporin 是一种小激酶抑制剂,是一种从细菌 Streptomyces staurosporeus 中提取的生物碱。 | ||||
| GC44050 | Leucinostatin A | 76600-38-9 | Natural ProductsImmunosuppressantsAdaptive ImmunityCandidiasisBacterial DiseasesCancer Biology | |
A fungal metabolite with diverse biological activities | ||||
| GC11947 | Ansamitocin P-3 | 66547-09-9 | OthersMicrotubule/TubulinADC Cytotoxin | |
A microtubule depolymerizing agent | ||||
| GC15966 | Avermectin B1b | 65195-56-4 | Antibiotic | |
An insecticide and anthelmintic | ||||
| GC17427 | Geneticin, G-418 Sulfate | 108321-42-2 | AntibioticBacterial | |
Geneticin,G-418硫酸盐是一类氨基糖苷类抗生素,其结构与新霉素卡那霉素相似。 | ||||
| GC36427 | Lasalocid sodium | 25999-20-6 | BacterialAutophagy | |
An ionophore antibiotic | ||||
