GlpBio

关于 "Antibiotic" 的结果30 个结果

货号产品名称CAS 号靶点化学结构
GC31586Monacolin J (Antibiotic MB 530A)79952-42-4HMG-CoA ReductaseAutophagyGC31586 structure
Monacolin J (Antibiotic MB 530A) 是一种胆固醇生物合成抑制剂,可抑制 HMG-CoA 还原酶的活性。
GC92249MRSA Antibiotic 2667410-02-8GC92249 structure
MRSA antibiotic 2 is an antibiotic.
GC45383Antibiotic PF 1052147317-15-5Natural ProductsImmunology/InflammationFood-Borne IllnessesGC45383 structure
A fungal metabolite
GC32220Antibiotic-5d251349-54-9BacterialGC32220 structure
Antibiotic-5d是一种合成的抗微生物化合物。
GF16717antibiotics-antimycoticGF16717 structure
GC26403G418 Selective Antibiotic, SterileGC26403 structure

G418 Selective Antibiotic, Sterile G418、G 418或者G-418,是一种结构类似于庆大霉素B1 (Gentamycin B1)的氨基糖苷类抗生素,常用于筛选表达neo基因的真核或原核多克隆或单克隆细胞。

GC91670MRSA Antibiotic 1667410-81-3AntibioticMRSAImmunology/InflammationGC91670 structure
MRSA antibiotic 1 is an antibiotic.
GC48226Urdamycin A98474-21-6Natural ProductsImmunology/InflammationBacterial DiseasesCancer BiologyGC48226 structure
A bacterial metabolite
GC47924Parvodicin C2110882-85-4Natural ProductsImmunology/InflammationMRSAGC47924 structure
A glycopeptide antibiotic
GC48533Vanoxonin86933-99-5Natural ProductsApoptosisDNA/RNA SynthesisGC48533 structure
A bacterial metabolite
GC60668Calcimycin hemimagnesium72124-77-7ApoptosisBacterialAutophagyFungalGC60668 structure
Calcimycin(A-23187)hemimagnesium是一种抗生素和独特的二价阳离子离子载体(divalentcationionophore),如钙离子和镁离子。Calcimycinhemimagnesium通过增加细胞内钙浓度诱导Ca2+依赖性细胞死亡。Calcimycinhemimagnesium抑制革兰氏阳性细菌和一些真菌的生长,还抑制ATP酶的活性并解耦哺乳动物细胞的氧化磷酸化(OXPHOS),诱导细胞凋亡(apoptosis)。
GC18936A-83016F142435-72-1Natural ProductsImmunology/InflammationPneumoniaGC18936 structure
An aurodox antibiotic
GC63650Pentachloropseudilin69640-38-6MyosinGC63650 structure
Pentachloropseudilin (Antibiotic A 15104 Y; PClP) 是一种可逆的、变构有效的肌球蛋白 (Myo1s) 抑制剂,对 Myo1s 的 IC50 范围为 1 至 5 μM,对于 2 类和 5 类肌球蛋白,IC50 范围 > 90 μM。Pentachloropseudilin 是转化生长因子-β (TGF-β) 刺激的信号传导的有效抑制剂,对 TGF-β 的 IC50 值为 0.1-0.2 μM。
GC17519Concanamycin A80890-47-7AutophagyProton PumpGC17519 structure
Concanamycin A 是液泡型 ATP 酶 (V-ATPase) 的特异性抑制剂,IC50 值为 10 nM 。
GC43882Hygrolidin83329-73-1AntibioticADC CytotoxinFungalGC43882 structure
A macrocyclic lactone
GC43883Hymeglusin29066-42-0Natural ProductsInnate ImmunityCholesterol MetabolismBacterial DiseasesGC43883 structure
An HMG-CoA synthase inhibitor
GC42888Azamulin76530-44-4P450GC42888 structure
A selective CYP3A inhibitor
GC45514Micronomicin (sulfate)66803-19-8AntibioticBacterialGC45514 structure
An aminoglycoside antibiotic
GC15299Staurosporine(CGP 41251)62996-74-1PKCBroad Spectrum Protein Kinase InhibitorPKAGC15299 structure
Staurosporin 是一种小激酶抑制剂,是一种从细菌 Streptomyces staurosporeus 中提取的生物碱。
GC44050Leucinostatin A76600-38-9Natural ProductsImmunosuppressantsAdaptive ImmunityCandidiasisBacterial DiseasesCancer BiologyGC44050 structure
A fungal metabolite with diverse biological activities
GC11947Ansamitocin P-366547-09-9OthersMicrotubule/TubulinADC CytotoxinGC11947 structure
A microtubule depolymerizing agent
GC15966Avermectin B1b65195-56-4AntibioticGC15966 structure
An insecticide and anthelmintic
GC17427Geneticin, G-418 Sulfate108321-42-2AntibioticBacterialGC17427 structure

Geneticin,G-418硫酸盐是一类氨基糖苷类抗生素,其结构与新霉素卡那霉素相似。

GC36427Lasalocid sodium25999-20-6BacterialAutophagyGC36427 structure
An ionophore antibiotic