关于 "Nucleoside Antimetabolite/Analogue" 的结果17+ 个结果
筛选:Reverse Transcriptase×
- Islatravir (MK-8591)CAS: 865363-93-5
A nucleoside reverse transcriptase inhibitor
Reverse Transcriptase - Dapivirine (TMC120)CAS: 244767-67-7
A non-nucleoside reverse transcriptase inhibitor
Reverse Transcriptase - Rilpivirine HydrochlorideCAS: 700361-47-3
Rilpivirine (TMC278), is a second-generation non-nucleoside reverse transcriptase inhibitor (NNRTI) with higher potency, longer half-life and reduced side-effect profile compared with older NNRTIs, such as efavirenz.
Reverse Transcriptase - CensavudineCAS: 634907-30-5
Censavudine (OBP-601; BMS-986001),一种核苷类似物,是一种核苷逆转录酶 (nucleoside reverse transcriptase) 抑制剂。Censavudine 是一种有效的 HIV 抑制剂,对 HIV-2 和 HIV-1 的 EC50 范围分别为 30-81 nM 和 450-890 nM。
- DexelvucitabineCAS: 134379-77-4
Dexelbucitabine (Reverset; d-d4FC) 是一种胞苷 类似物,一种具有口服活性的核苷逆转录酶 (nucleoside reverse transcriptase) 抑制剂。Dexelbucitabine 是一种有效的抗 HIV-1 病毒剂,这些病毒聚合酶中含有胸苷类似物和/或 M184V 突变。Dexelvucitabine 是一种 2'-脱氧胞苷抗逆转录病毒剂。
Reverse Transcriptase - 3'-Azido-3'-deoxythymidine β-D-glucuronide (sodium salt)CAS: 133525-01-6
A zidovudine metabolite
Reverse Transcriptase
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC16092 | Entecavir Hydrate | 209216-23-9 | HBV | ||
An antiviral nucleoside analog | |||||
| GC11274 | Abacavir sulfate | 188062-50-2 | Reverse Transcriptase | ||
An antiviral nucleoside analog | |||||
| GC32306 | Islatravir (MK-8591) | 865363-93-5 | Reverse Transcriptase | ||
A nucleoside reverse transcriptase inhibitor | |||||
| GC13653 | Emtricitabine | 143491-57-0 | HIV | ||
A nucleoside reverse transcriptase inhibitor | |||||
| GC14720 | Zalcitabine | 7481-89-2 | HIV | ||
A nucleoside reverse transcriptase inhibitor | |||||
| GC19126 | Doravirine | 1338225-97-0 | Reverse Transcriptase | ||
A non-nucleoside reverse transcriptase inhibitor | |||||
| GC14452 | Dapivirine (TMC120) | 244767-67-7 | Reverse Transcriptase | ||
A non-nucleoside reverse transcriptase inhibitor | |||||
| GC15452 | Delavirdine mesylate | 147221-93-0 | HIV | ||
A non-nucleoside reverse transcriptase inhibitor | |||||
| GC35835 | Delavirdine | 136817-59-9 | Reverse Transcriptase | ||
A non-nucleoside reverse transcriptase inhibitor | |||||
| GC15330 | Didanosine | 69655-05-6 | HIV | ||
An antiviral nucleoside analog and inhibitor of reverse transcriptase | |||||
| GC11059 | Rilpivirine | 500287-72-9 | Reverse Transcriptase | ||
A non-nucleoside reverse transcriptase inhibitor | |||||
| GC25867 | Rilpivirine Hydrochloride | 700361-47-3 | Reverse Transcriptase | ||
Rilpivirine (TMC278), is a second-generation non-nucleoside reverse transcriptase inhibitor (NNRTI) with higher potency, longer half-life and reduced side-effect profile compared with older NNRTIs, such as efavirenz. | |||||
| GC64261 | Censavudine | 634907-30-5 | HIV | ||
Censavudine (OBP-601; BMS-986001),一种核苷类似物,是一种核苷逆转录酶 (nucleoside reverse transcriptase) 抑制剂。Censavudine 是一种有效的 HIV 抑制剂,对 HIV-2 和 HIV-1 的 EC50 范围分别为 30-81 nM 和 450-890 nM。 | |||||
| GC10317 | Lamivudine | 134678-17-4 | SARS-CoV | ||
Lamivudine是一种口服核苷类似物,作为核苷类逆转录酶抑制剂,抗乙肝病毒(HBV)活性的EC50值为0.07±0.02μg/ml。 | |||||
| GC16387 | Nevirapine | 129618-40-2 | HIV | ||
An NNRTI | |||||
| GC64590 | Dexelvucitabine | 134379-77-4 | Reverse Transcriptase | ||
Dexelbucitabine (Reverset; d-d4FC) 是一种胞苷 类似物,一种具有口服活性的核苷逆转录酶 (nucleoside reverse transcriptase) 抑制剂。Dexelbucitabine 是一种有效的抗 HIV-1 病毒剂,这些病毒聚合酶中含有胸苷类似物和/或 M184V 突变。Dexelvucitabine 是一种 2'-脱氧胞苷抗逆转录病毒剂。 | |||||
| GC10387 | 3'-Azido-3'-deoxythymidine β-D-glucuronide (sodium salt) | 133525-01-6 | Reverse Transcriptase | ||
A zidovudine metabolite | |||||
