关于 "Aurora Kinase" 的结果13+ 个结果
筛选:Neuroscience×
- Calmodulin-Dependent Protein Kinase II(290-309) acetate
Calmodulin-DependentProteinKinaseII(290-309)acetate是有效的CaMK拮抗剂,抑制抑制Ca2+/钙调蛋白依赖性蛋白激酶II的IC50值为52nM。
- TrkB Agonist Prodrug R13CAS: 1609067-49-3
TrkB Agonist Prodrug R13(R13)是原肌球蛋白相关激酶B(TrkB)激活剂7,8-二羟基黄酮的前药形式。
- PKG Inhibitor (trifluoroacetate salt)
PKG Inhibitor (trifluoroacetate salt)是一种特定的cGMP依赖性PKG抑制剂Ki=86μM。
- A-3 hydrochlorideCAS: 78957-85-4
A-3 hydrochloride, a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases, againsts cAMP-dependent protein kinase (PKA) (Ki=4.3 ?M), casein kinase II (CK2) (Ki=5.1 ?M) and myosin light chain kinase (MLCK) (Ki=7.4 ?M), also inhibits Protein Kinase C (PKC) and casein kinase I (CK1) with Ki values of 47 ?M and 80 ?M, respectively.
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GP10017 | [Ser25] Protein Kinase C (19-31) | 136795-05-6 | Neuroscience Peptides | ||
PKC substrate | |||||
| GC31170 | Calmodulin-Dependent Protein Kinase II 290-309 | 115044-69-4 | Peptides | ||
A CaMKII inhibitor | |||||
| GC61521 | Calmodulin-Dependent Protein Kinase II(290-309) acetate | - | Peptides | ||
Calmodulin-DependentProteinKinaseII(290-309)acetate是有效的CaMK拮抗剂,抑制抑制Ca2+/钙调蛋白依赖性蛋白激酶II的IC50值为52nM。 | |||||
| GC43128 | Calmodulin-Dependent Protein Kinase II (290-309) (trifluoroacetate salt) | - | Peptides | ||
A CaMKII inhibitor | |||||
| GC43220 | Cdk5 Substrate | 164669-07-2 | Neuroscience | ||
A peptide substrate of Cdk5 | |||||
| GC44978 | Syk Inhibitor II | 726695-51-8 | 5-HT Receptor | ||
A selective blocker of spleen tyrosine kinase activity | |||||
| GC91148 | JAK Inhibitor 31 | 2891469-99-9 | JAK | ||
一种JAK2抑制剂 | |||||
| GC14583 | R 59-022 | 93076-89-2 | 5-HT Receptor | ||
R 59-022是一种二酰甘油激酶抑制剂(IC50 = 2.8µM)。 | |||||
| GC91977 | TrkB Agonist Prodrug R13 | 1609067-49-3 | Behavioral Neuroscience | ||
TrkB Agonist Prodrug R13(R13)是原肌球蛋白相关激酶B(TrkB)激活剂7,8-二羟基黄酮的前药形式。 | |||||
| GC92078 | PKG Inhibitor (trifluoroacetate salt) | - | cGMP | ||
PKG Inhibitor (trifluoroacetate salt)是一种特定的cGMP依赖性PKG抑制剂Ki=86μM。 | |||||
| GC60037 | A-3 hydrochloride | 78957-85-4 | PKA | ||
A-3 hydrochloride, a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases, againsts cAMP-dependent protein kinase (PKA) (Ki=4.3 ?M), casein kinase II (CK2) (Ki=5.1 ?M) and myosin light chain kinase (MLCK) (Ki=7.4 ?M), also inhibits Protein Kinase C (PKC) and casein kinase I (CK1) with Ki values of 47 ?M and 80 ?M, respectively. | |||||
| GC33732 | Syntide 2 | 108334-68-5 | Peptides | ||
A protein kinase substrate | |||||
| GC37710 | Syntide 2 (TFA) | - | Peptides | ||
A protein kinase substrate | |||||
