关于 "Topoisomerase" 的结果6 个结果
筛选:Microbiology & Virology×
- Chloroquinoxaline sulfonamideCAS: 97919-22-7
Chloroquinoxaline sulfonamide (Chloroquinoxaline) 是 sulfaquinoxaline 的结构类似物,是拓扑异构酶 II alpha/beta (topoisomerase II alpha/beta) 毒物。Chloroquinoxaline sulfonamide 用于控制家禽,兔,绵羊和牛的球虫病。 具有抗肿瘤活性。
- Etoposide phosphateCAS: 117091-64-2
Etoposidephosphate(BMY-40481)是一种有效的抗癌(anti-cancer)化疗试剂和一种选择性拓扑异构酶II(topoisomeraseII)抑制剂,可以防止DNA链的重新连接。Etoposidephosphate是依托泊苷的磷酸酯前药,被认为与Etoposide活性相当。Etoposidephosphate诱导细胞周期阻滞、凋亡(apoptosis)和自噬(autophagy)。
- Levofloxacin hydrate (Levofloxacin hemihydrate)CAS: 138199-71-0
Levofloxacin (Levaquin, Tavanic, Quixin, Iquix, Cravit) is a broad-spectrum, third-generation fluoroquinolone antibiotic and optically active L-isomer of ofloxacin with antibacterial activity. It acts by inhibiting DNA gyrase (bacterial topoisomerase II).
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC14363 | Mitoxantrone HCl | 70476-82-3 | SARS-CoV | ||
An inhibitor of DNA topoisomerase IIα and HIV-1 integrase | |||||
| GC60107 | Chloroquinoxaline sulfonamide | 97919-22-7 | Parasite | ||
Chloroquinoxaline sulfonamide (Chloroquinoxaline) 是 sulfaquinoxaline 的结构类似物,是拓扑异构酶 II alpha/beta (topoisomerase II alpha/beta) 毒物。Chloroquinoxaline sulfonamide 用于控制家禽,兔,绵羊和牛的球虫病。 具有抗肿瘤活性。 | |||||
| GC60374 | Trovafloxacin | 147059-72-1 | Bacterial | ||
A topoisomerase IV and DNA gyrase inhibitor | |||||
| GC60826 | Etoposide phosphate | 117091-64-2 | Autophagy | ||
Etoposidephosphate(BMY-40481)是一种有效的抗癌(anti-cancer)化疗试剂和一种选择性拓扑异构酶II(topoisomeraseII)抑制剂,可以防止DNA链的重新连接。Etoposidephosphate是依托泊苷的磷酸酯前药,被认为与Etoposide活性相当。Etoposidephosphate诱导细胞周期阻滞、凋亡(apoptosis)和自噬(autophagy)。 | |||||
| GC10128 | Temafloxacin (hydrochloride) | 105784-61-0 | Antibiotic | ||
A DNA topoisomerase inhibitor | |||||
| GC33929 | Levofloxacin hydrate (Levofloxacin hemihydrate) | 138199-71-0 | Bacterial | ||
Levofloxacin (Levaquin, Tavanic, Quixin, Iquix, Cravit) is a broad-spectrum, third-generation fluoroquinolone antibiotic and optically active L-isomer of ofloxacin with antibacterial activity. It acts by inhibiting DNA gyrase (bacterial topoisomerase II). | |||||
