关于 "Topoisomerase" 的结果6 个结果

筛选:Microbiology & Virology×
  • GC14363 structure
    Mitoxantrone HCl
    CAS: 70476-82-3

    An inhibitor of DNA topoisomerase IIα and HIV-1 integrase

  • GC60107 structure
    Chloroquinoxaline sulfonamide
    CAS: 97919-22-7

    Chloroquinoxaline sulfonamide (Chloroquinoxaline) 是 sulfaquinoxaline 的结构类似物,是拓扑异构酶 II alpha/beta (topoisomerase II alpha/beta) 毒物。Chloroquinoxaline sulfonamide 用于控制家禽,兔,绵羊和牛的球虫病。 具有抗肿瘤活性。

  • GC60374 structure
    Trovafloxacin
    CAS: 147059-72-1

    A topoisomerase IV and DNA gyrase inhibitor

  • GC60826 structure
    Etoposide phosphate
    CAS: 117091-64-2

    Etoposidephosphate(BMY-40481)是一种有效的抗癌(anti-cancer)化疗试剂和一种选择性拓扑异构酶II(topoisomeraseII)抑制剂,可以防止DNA链的重新连接。Etoposidephosphate是依托泊苷的磷酸酯前药,被认为与Etoposide活性相当。Etoposidephosphate诱导细胞周期阻滞、凋亡(apoptosis)和自噬(autophagy)。

  • GC10128 structure
    Temafloxacin (hydrochloride)
    CAS: 105784-61-0

    A DNA topoisomerase inhibitor

  • GC33929 structure
    Levofloxacin hydrate (Levofloxacin hemihydrate)
    CAS: 138199-71-0

    Levofloxacin (Levaquin, Tavanic, Quixin, Iquix, Cravit) is a broad-spectrum, third-generation fluoroquinolone antibiotic and optically active L-isomer of ofloxacin with antibacterial activity. It acts by inhibiting DNA gyrase (bacterial topoisomerase II).