关于 "Oxidative Phosphorylation" 的结果48+ 个结果
筛选:Metabolism×
- Roflumilast-d4 N-OxideCAS: 1794760-31-8
Roflumilast-d4 N-Oxide 是 Roflumilast 的氘代物。Roflumilast 是一种选择性的 PDE4 抑制剂,作用于 PDE4A1,PDEA4,PDEB1 和 PDEB2,IC50 分别为 0.7,0.9,0.7 和 0.2 nM。
- Dibutyryl-cAMP, sodium saltCAS: 16980-89-5
Dibutyryl-cAMP, sodium salt,又称为Bucladesine,是一种细胞膜可透性环核苷酸类似物,能模拟内源性cAMP的作用,并作为磷酸二酯酶抑制剂。
- D-Mannose-6-Phosphate (sodium salt hydrate)
A phosphorylated aldohexose with diverse roles
- Elesclomol (STA-4783)CAS: 488832-69-5
Elesclomol(也称为 STA-4783)最初是在基于细胞的表型筛选中发现的促凋亡活性,是一种新型小分子,可通过快速产生活性氧 (ROS) 有效诱导癌细胞凋亡以及难以控制的氧化应激水平的诱导。
- α-D-Glucose-1,6-bisphosphate (potassium salt hydrate)CAS: 91183-87-8
A bis-phosphorylated derivative of α-D-glucose
- 5α-hydroxy-6-keto CholesterolCAS: 13027-33-3
A cytotoxic metabolite of ozone-oxidized cholesterol
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC68325 | Roflumilast-d4 N-Oxide | 1794760-31-8 | PDE | ||
Roflumilast-d4 N-Oxide 是 Roflumilast 的氘代物。Roflumilast 是一种选择性的 PDE4 抑制剂,作用于 PDE4A1,PDEA4,PDEB1 和 PDEB2,IC50 分别为 0.7,0.9,0.7 和 0.2 nM。 | |||||
| GC40879 | 4-hydroxy Solifenacin N-oxide | 2747991-39-3 | Neuroscience | ||
An N-oxide form of 4-hydroxy solifenacin | |||||
| GC49686 | N-desmethyl Regorafenib N-oxide | 835621-12-0 | Tie-2 | ||
An active metabolite of regorafenib | |||||
| GC44904 | S-Methyl-L-Cysteine-S-oxide | 6853-87-8 | Metabolism | ||
An alliin analog | |||||
| GC16612 | GGsTop | 926281-37-0 | Others | ||
GGsTop是γ-谷氨酰转肽酶(GGT)的不可逆抑制剂(Ki = 170μM)。 | |||||
| GC12824 | Dibutyryl-cAMP, sodium salt | 16980-89-5 | PDE | ||
Dibutyryl-cAMP, sodium salt,又称为Bucladesine,是一种细胞膜可透性环核苷酸类似物,能模拟内源性cAMP的作用,并作为磷酸二酯酶抑制剂。 | |||||
| GC16944 | SR 1664 | 1338259-05-4 | PPAR | ||
An inhibitor of Cdk5-mediated PPARγ phosphorylation | |||||
| GC18632 | 6-hydroxy Bexarotene | 368451-07-4 | ROR/RAR/RXR | ||
An oxidative metabolite of bexarotene | |||||
| GC49868 | D-α-Tocopheryl Quinone | 7559-04-8 | Ferroptosis | ||
An oxidative metabolite of vitamin E | |||||
| GC52278 | Creatine Phosphate (sodium salt hydrate) | 19333-65-4 | Metabolism | ||
A phosphorylated form of creatine | |||||
| GC43501 | D-Mannose-6-Phosphate (sodium salt hydrate) | - | Carbohydrate Metabolism | ||
A phosphorylated aldohexose with diverse roles | |||||
| GC44636 | Phospho-L-Arginine (lithium salt hydrate) | - | Metabolism | ||
A phosphorylated form of L-arginine | |||||
| GC13885 | Elesclomol (STA-4783) | 488832-69-5 | Other Apoptosis | ||
Elesclomol(也称为 STA-4783)最初是在基于细胞的表型筛选中发现的促凋亡活性,是一种新型小分子,可通过快速产生活性氧 (ROS) 有效诱导癌细胞凋亡以及难以控制的氧化应激水平的诱导。 | |||||
| GC48278 | α-D-Glucose-1,6-bisphosphate (potassium salt hydrate) | 91183-87-8 | Carbohydrate Metabolism | ||
A bis-phosphorylated derivative of α-D-glucose | |||||
| GC42039 | 1-Stearoyl-2-15(S)-HETE-sn-glycero-3-PC | 154436-51-8 | Lipoxygenase | ||
An oxidized phospholipid | |||||
| GC42040 | 1-Stearoyl-2-15(S)-HETE-sn-glycero-3-PE | 947381-58-0 | Lipoxygenase | ||
An oxidized phospholipid | |||||
| GC42041 | 1-Stearoyl-2-15(S)-HpETE-sn-glycero-3-PC | 154436-48-3 | Lipoxygenase | ||
An oxidized phospholipid | |||||
| GC42042 | 1-Stearoyl-2-15(S)-HpETE-sn-glycero-3-PE | 154436-49-4 | Lipoxygenase | ||
An oxidized phospholipid | |||||
| GC46761 | 9-Oxononanoic Acid | 2553-17-5 | Cyclooxygenase | ||
An oxidized fatty acid | |||||
| GC49879 | Metformin hydroxy analog 2 | 98026-16-5 | Cancer Biology | ||
An oxidation product of metformin | |||||
| GC44308 | NADP+ (sodium salt hydrate) | 698999-85-8 | Mitochondrial Metabolism | ||
The oxidized form of NADPH | |||||
| GC44062 | L-hydroxy Arginine (acetate) | 1140844-61-6 | Vasodilation | ||
A substrate for nitric oxide synthase | |||||
| GC40534 | 20-hydroxy Prostaglandin F2α | 57930-92-4 | Cyclooxygenase | ||
A CYP450 ω-oxidation metabolite of PGF2α | |||||
| GC40693 | 5α-hydroxy-6-keto Cholesterol | 13027-33-3 | Sterol Lipids | ||
A cytotoxic metabolite of ozone-oxidized cholesterol | |||||
