关于 "CYP3A/CYP450" 的结果35+ 个结果
筛选:Metabolism×
- VoriconazoleCAS: 137234-62-9
Voriconazole是一种强效竞争性抑制剂，可抑制CYP2B6（IC 50 =1.71μM）、CYP2C9（IC 50 =3.62μM）、CYP2C19（IC 50 =5.25μM）和CYP3A（IC 50 =2.90μM）。
- (±)4(5)-EpDPA methyl esterCAS: 121818-29-9
Stable precursor of (±)4(5)-EpDPA, a CYP450 metabolite of DHA
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC40440 | (±)8(9)-EET | - | PPAR | ||
A racemic version of a CYP450 metabolite of arachidonic acid | |||||
| GC42888 | Azamulin | 76530-44-4 | P450 | ||
A selective CYP3A inhibitor | |||||
| GC14269 | Cobicistat (GS-9350) | 1004316-88-4 | HIV | ||
An inhibitor of CYP3A | |||||
| GC40528 | 11α-hydroxy Testosterone | 3066-12-4 | Androgen Receptor | ||
A CYP3A metabolite of testosterone | |||||
| GC13836 | 2,3-dihydrothieno-Thiadiazole Carboxylate | 152467-47-5 | P450 | ||
Selective CYP450 inhibitor | |||||
| GC16575 | Alizarin | 72-48-0 | P450 | ||
A CYP450 inhibitor | |||||
| GC49030 | 7-Ethoxycoumarin | 31005-02-4 | Enzyme Substrates | ||
A CYP450 substrate | |||||
| GC52062 | 7-Benzyloxy-4-(trifluoromethyl)coumarin | 220001-53-6 | P450 | ||
A fluorogenic substrate for CYP1A2 and CYP3A | |||||
| GC16259 | SKF 525A (hydrochloride) | 62-68-0 | P450 | ||
A nonspecific CYP450 inhibitor | |||||
| GC10554 | 3-Cyano-7-ethoxycoumarin | 117620-77-6 | CYP3A/CYP450 | ||
A fluorogenic CYP450 substrate | |||||
| GC41945 | 16-hydroxy Hexadecanoic Acid | 506-13-8 | P450 | ||
CYP450 metabolite of palmitic acid | |||||
| GC40272 | (±)8(9)-DiHET | 192461-96-4 | Cyclooxygenase | ||
A CYP450 metabolite of arachidonic acid | |||||
| GC42083 | 20-HETE Ethanolamide | 942069-11-6 | Endocannabinoid/Endocannabinoid-like | ||
A putative CYP450 metabolite of AEA | |||||
| GC44299 | N-Acetyl-4-benzoquinone imine | 50700-49-7 | Drug Metabolite | ||
A reactive CYP450 metabolite of acetaminophen | |||||
| GC40534 | 20-hydroxy Prostaglandin F2α | 57930-92-4 | Cyclooxygenase | ||
A CYP450 ω-oxidation metabolite of PGF2α | |||||
| GC44819 | Resorufin benzyl ether | 87687-02-3 | P450 | ||
A fluorometric substrate for CYP450-linked enzymes | |||||
| GC42085 | 20-hydroxy N-Arachidonoyl Taurine | - | P450 | ||
A potential CYP450 metabolite of N-arachidonoyl-taurine | |||||
| GC19483 | MS-PPOH | 206052-02-0 | P450 | ||
A potent, selective inhibitor of microsomal CYP450 epoxidase activity | |||||
| GC40438 | (±)5(6)-EET | 87173-80-6 | Vasodilation | ||
A racemic version of a CYP450 metabolite of arachidonic acid | |||||
| GC40466 | (±)11(12)-EET | 87173-81-7 | Innate Immunity | ||
A racemic version of a CYP450 metabolite of arachidonic acid | |||||
| GC13079 | Voriconazole | 137234-62-9 | Fungal | ||
Voriconazole是一种强效竞争性抑制剂，可抑制CYP2B6（IC50=1.71μM）、CYP2C9（IC50=3.62μM）、CYP2C19（IC50=5.25μM）和CYP3A（IC50=2.90μM）。 | |||||
| GC41660 | (±)4(5)-EpDPA methyl ester | 121818-29-9 | P450 | ||
Stable precursor of (±)4(5)-EpDPA, a CYP450 metabolite of DHA | |||||
| GC31464 | CDD3505 | 173865-33-3 | P450 | ||
CDD3505 is used for elevating high density lipoprotein cholesterol (HDL) by inducing hepatic cytochrome P450IIIA (CYP3A) activity. | |||||
| GC31460 | CDD3506 | 197913-15-8 | P450 | ||
CDD3506可以通过诱导肝CYP3A的活动，来提高高密度脂蛋白胆固醇(HDL)的水平。 | |||||