关于 "Dopamine Receptor" 的结果40+ 个结果
- Propionylpromazine hydrochlorideCAS: 7681-67-6
A promazine neuroleptic and dopamine receptor antagonist
Dopamine Receptor - L-741,742 hydrochlorideCAS: 874882-93-6
highly potent and selective D4 dopamine receptor antagonist
Dopamine Receptor - (-)-StepholidineCAS: 16562-13-3
A dopamine receptor antagonist and 5-HT 1A partial agonist
Dopamine Receptor - Tiapride hydrochlorideCAS: 51012-33-0
Tiapride is a drug that selectively blocks D2 and D3 dopamine receptors in the brain and is used to treat a variety of neurological and psychiatric disorders.
Dopamine Receptor - NaxagolideCAS: 88058-88-2
Naxagolide ((+)-PHNO; Dopazinol) 是一种有效的多巴胺 D2 (dopamine D2) (Dopamine Receptor) 激动剂。Naxagolide 具有用于帕金森病 (PD) 研究的潜力。
Dopamine Receptor - Promazine hydrochlorideCAS: 53-60-1
Promazine (Romtiazin, Sinophenin) is an antagonist at types 1, 2, and 4 dopamine receptors, 5-HT receptor types 2A and 2C, muscarinic receptors 1 through 5, alpha(1)-receptors, and histamine H1-receptors with antipsychotic effects.
Dopamine Receptor - Quetiapine D4 hemifumarateCAS: 1217310-65-0
Quetiapine D4 hemifumarate 是 Quetiapine hemifumarate 的氘代物。Quetiapine 是一种 5-HT 受体激动剂,也是一种多巴胺受体 (dopamine receptor) 拮抗剂。具有抗抑郁和抗焦虑作用。
Dopamine Receptor - (+)-AJ 76 hydrochlorideCAS: 85379-09-5
(+)-AJ 76 hydrochloride是一种对突触前受体具有优先作用的多巴胺受体(dopamine receptors, DRs)拮抗剂(hD3、hD4、hD2S、hD2L和rD2受体的pKi值分别为6.95、6.67、6.37、6.21和6.07)。
Dopamine Receptor - Pimozide-d4-1
Pimozide-d4-1 氘代标记的 Pimozide。Pimozide 是 dopamine receptor 的拮抗剂,对 dopamine D2,D3 和 D1 受体的 Ki 值分别为 1.4 nM,2.5 nM 和 588 nM,同时对 α1-adrenoceptor 也有较高亲和性,Ki 值为 39 nM;Pimozide 也是 STAT3 和 STAT5 的抑制剂。
Dopamine Receptor - Dopamine-d5 hydrochlorideCAS: 2193106-55-5
Dopamine-d5 (hydrochloride) 是一种氘代标记的 Dopamine (hydrochloride)。Dopamine hydrochloride (ASL279) 是在脑黑质,脑腹侧被盖区和下丘脑中产生的一种儿茶酚胺类神经递质,在大脑和身体中起着重要作用。Dopamine hydrochloride (ASL279) 通过 D2 多巴胺受体 (D2 dopamine receptor) 来诱导 VEGFR2 的内吞作用,这对于促进血管生成是至关重要的。
Dopamine Receptor - Dopamine D2 receptor agonist-2CAS: 1610591-93-9
Dopamine D2 receptor agonist-2(化合物36)是一种有效的多巴胺D2受体偏向性激动配体,Ki值为11.2 nM。
Dopamine Receptor - Dopamine serotonin antagonist-1CAS: 1977-07-7
Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs (muscarinic Designer Receptors Exclusively Activated by Designer Drugs) agonist, and binds to DREADD receptor subtypes hM3Dq and hM4Di with Ki of 6.3 and 4.2 nM, respectively.
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC17075 | NPEC-caged-dopamine | 1257326-23-0 | Dopamine Receptor | ||
Dopamine receptor agonist | |||||
| GC14865 | RuBi-Dopa | - | Dopamine Receptor | ||
dopamine receptor activator | |||||
| GC30904 | Molindone hydrochloride (EN-1733A) | 15622-65-8 | Dopamine Receptor | ||
A dopamine receptor antagonist | |||||
| GC13931 | Bromocriptine mesylate | 22260-51-1 | Autophagy | ||
A dopamine receptor agonist | |||||
| GC11602 | Piribedil dihydrochloride | 1451048-94-4 | Dopamine Receptor | ||
A dopamine receptor agonist | |||||
| GC45188 | Zuclopenthixol | 53772-83-1 | Dopamine Receptor | ||
A dopamine receptor antagonist | |||||
| GC36929 | Piribedil | 3605-01-4 | Dopamine Receptor | ||
A dopamine receptor agonist | |||||
| GC16017 | Rotigotine hydrochloride | 125572-93-2 | Adrenergic Receptor | ||
A non-selective dopamine receptor agonist | |||||
| GC39736 | Propionylpromazine hydrochloride | 7681-67-6 | Dopamine Receptor | ||
A promazine neuroleptic and dopamine receptor antagonist | |||||
| GC13036 | L-741,742 hydrochloride | 874882-93-6 | Dopamine Receptor | ||
highly potent and selective D4 dopamine receptor antagonist | |||||
| GC14252 | (-)-Stepholidine | 16562-13-3 | Dopamine Receptor | ||
A dopamine receptor antagonist and 5-HT1A partial agonist | |||||
| GC10614 | Rotigotine | 99755-59-6 | Adrenergic Receptor | ||
A non-selective dopamine receptor agonist | |||||
| GC30975 | Tiapride hydrochloride | 51012-33-0 | Dopamine Receptor | ||
Tiapride is a drug that selectively blocks D2 and D3 dopamine receptors in the brain and is used to treat a variety of neurological and psychiatric disorders. | |||||
| GC67705 | Naxagolide | 88058-88-2 | Dopamine Receptor | ||
Naxagolide ((+)-PHNO; Dopazinol) 是一种有效的多巴胺 D2 (dopamine D2) (Dopamine Receptor) 激动剂。Naxagolide 具有用于帕金森病 (PD) 研究的潜力。 | |||||
| GC30974 | Promazine hydrochloride | 53-60-1 | Dopamine Receptor | ||
Promazine (Romtiazin, Sinophenin) is an antagonist at types 1, 2, and 4 dopamine receptors, 5-HT receptor types 2A and 2C, muscarinic receptors 1 through 5, alpha(1)-receptors, and histamine H1-receptors with antipsychotic effects. | |||||
| GC39724 | Quetiapine D4 hemifumarate | 1217310-65-0 | Dopamine Receptor | ||
Quetiapine D4 hemifumarate 是 Quetiapine hemifumarate 的氘代物。Quetiapine 是一种 5-HT 受体激动剂,也是一种多巴胺受体 (dopamine receptor) 拮抗剂。具有抗抑郁和抗焦虑作用。 | |||||
| GC13156 | (+)-AJ 76 hydrochloride | 85379-09-5 | Dopamine Receptor | ||
(+)-AJ 76 hydrochloride是一种对突触前受体具有优先作用的多巴胺受体(dopamine receptors, DRs)拮抗剂(hD3、hD4、hD2S、hD2L和rD2受体的pKi值分别为6.95、6.67、6.37、6.21和6.07)。 | |||||
| GC67752 | Pimozide-d4-1 | - | Dopamine Receptor | ||
Pimozide-d4-1 氘代标记的 Pimozide。Pimozide 是 dopamine receptor 的拮抗剂,对 dopamine D2,D3 和 D1 受体的 Ki 值分别为 1.4 nM,2.5 nM 和 588 nM,同时对 α1-adrenoceptor 也有较高亲和性,Ki 值为 39 nM;Pimozide 也是 STAT3 和 STAT5 的抑制剂。 | |||||
| GC68997 | Dopamine-d5 hydrochloride | 2193106-55-5 | Dopamine Receptor | ||
Dopamine-d5 (hydrochloride) 是一种氘代标记的 Dopamine (hydrochloride)。Dopamine hydrochloride (ASL279) 是在脑黑质,脑腹侧被盖区和下丘脑中产生的一种儿茶酚胺类神经递质,在大脑和身体中起着重要作用。Dopamine hydrochloride (ASL279) 通过 D2 多巴胺受体 (D2 dopamine receptor) 来诱导 VEGFR2 的内吞作用,这对于促进血管生成是至关重要的。 | |||||
| GC71157 | Dopamine D2 receptor agonist-2 | 1610591-93-9 | Dopamine Receptor | ||
Dopamine D2 receptor agonist-2(化合物36)是一种有效的多巴胺D2受体偏向性激动配体,Ki值为11.2 nM。 | |||||
| GC62940 | Dopamine | 51-61-6 | Dopamine Receptor | ||
An endogenous catecholamine | |||||
| GC11028 | Dopamine HCl | 62-31-7 | Dopamine Receptor | ||
An endogenous catecholamine | |||||
| GC30772 | Dopamine serotonin antagonist-1 | 1977-07-7 | Serotonin Transporter | ||
Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs (muscarinic Designer Receptors Exclusively Activated by Designer Drugs) agonist, and binds to DREADD receptor subtypes hM3Dq and hM4Di with Ki of 6.3 and 4.2 nM, respectively. | |||||
| GC15016 | SKF 83566 hydrobromide | 108179-91-5 | Dopamine Receptor | ||
A dopamine D1 receptor antagonist | |||||
