关于 "Rho" 的结果28+ 个结果
筛选:Cell Cycle/Checkpoint×
- Rho-Kinase-IN-2CAS: 2573071-18-6
Rho-Kinase-IN-2 (Compound 23) 是一种具有口服活性的、选择性的和中枢神经系统 (CNS) 渗透性的 Rho激酶 (ROCK) 抑制剂 (ROCK2 IC50=3 nM)。Rho-Kinase-IN-2 可用于亨廷顿病的研究。
- GSK269962A HClCAS: 2095432-71-4
GSK269962A HCl (GSK269962B, GSK269962) is a selective ROCK(Rho-associated protein kinase) inhibitor with IC50 values of 1.6 and 4 nM for ROCK1 and ROCK2, respectively.
- CCG-222740CAS: 1922098-69-8
CCG-222740 is a Rho/MRTF pathway inhibitor. CCG-222740 decreases the activation of stellate cells in vitro and in vivo, by reducing the levels of alpha smooth muscle actin(α-SMA) expression.
- ROCK inhibitor-2CAS: 1127308-52-4
ROCK inhibitor-2是一种选择性Rho激酶(ROCK)抑制剂,抑制ROCK1和ROCK2的IC 50 值分别为17nM和2nM,具有抗肿瘤活性。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC66050 | Rho-Kinase-IN-2 | 2573071-18-6 | ROCK | ||
Rho-Kinase-IN-2 (Compound 23) 是一种具有口服活性的、选择性的和中枢神经系统 (CNS) 渗透性的 Rho激酶 (ROCK) 抑制剂 (ROCK2 IC50=3 nM)。Rho-Kinase-IN-2 可用于亨廷顿病的研究。 | |||||
| GC33310 | Rho-Kinase-IN-1 | 1035094-83-7 | ROCK | ||
Rho-Kinase-IN-1是一个rho激酶抑制剂,来自专利US20090325960A1,化合物1.008。 | |||||
| GC70451 | Rho-Kinase-IN-3 | 864082-23-5 | ROCK | ||
Rho-Kinase-IN-3(化合物12)是一种强效且选择性的Rho激酶(ROCK1)抑制剂,IC50值为8nM。 | |||||
| GC72976 | Rhodblock 6 | 886625-06-5 | ROCK | ||
Rhodblock 6是一种Rho激酶(ROCK)抑制剂,抑制磷酸MRLC(肌球蛋白调节轻链)定位。 | |||||
| GC41698 | (D)2-Rh 110 (trifluoroacetate salt) | - | Proteolysis | ||
A fluorogenic caspase substrate | |||||
| GC44829 | Rhod-5N (potassium salt) | 888229-31-0 | Calcium Channel | ||
A low affinity fluorescent calcium probe | |||||
| GC41737 | (S)-Glycyl-H-1152 (hydrochloride) | 913844-45-8 | ROCK | ||
A ROCK inhibitor | |||||
| GC40009 | Bostrycin | 21879-81-2 | MRSA | ||
An anthraquinone with diverse biological activities | |||||
| GC40121 | (Z-DEVD)2-Rh 110 (trifluoroacetate salt) | - | Proteolysis | ||
A fluorogenic substrate for caspase-3 | |||||
| GC12314 | 3-(4-Pyridyl)indole | 7272-84-6 | ROCK | ||
A ROCK1 and ROCK2 inhibitor | |||||
| GC41742 | (Z-IETD)2-Rh 110 (trifluoroacetate salt) | - | Proteolysis | ||
A fluorogenic substrate for caspase-8 | |||||
| GC10512 | Y-27632 dihydrochloride | 129830-38-2 | Other Apoptosis | ||
Y-27632 dihydrochloride 作为一种选择性 Rho 激酶抑制剂,是一种新型支气管扩张剂。 | |||||
| GC12795 | CCG-1423 | 285986-88-1 | Ras | ||
An inhibitor of Rho-mediated cell signalling | |||||
| GC14986 | CCG-100602 | 1207113-88-9 | Rho | ||
A Rho/MKL1 transcriptional pathway inhibitor | |||||
| GC10419 | (R)-CCG-1423 | 2309931-09-5 | Rho | ||
A stereoisomer of CCG-1423, a Rho inhibitor | |||||
| GC14497 | (S)-CCG-1423 | 2319939-24-5 | Rho | ||
A stereoisomer of CCG-1423, a Rho inhibitor | |||||
| GC71056 | Zelasudil | 2365193-22-0 | ROCK | ||
Zelasudil是Rho相关(ROCK)激酶抑制剂。 | |||||
| GC66338 | ROCK1-IN-1 | 692869-38-8 | ROCK | ||
WAY-624704 is a novel Rho kinases (ROCK) inhibitor with an Ki of 17 nM. | |||||
| GC11181 | Thiazovivin | 1226056-71-8 | ROCK | ||
Thiazovivin是一种选择性Rho相关激酶(ROCK)抑制剂。 | |||||
| GC12827 | SLx-2119 | 911417-87-3 | ROCK | ||
SLx-2119是一种高效的Rho kinase (ROCK) 2抑制剂,IC50值为105nM。 | |||||
| GC37947 | Y-33075 | 199433-58-4 | ROCK | ||
Y-33075是一种有效的ROCK(Rho相关蛋白激酶)抑制剂,IC50值为3.6nM。 | |||||
| GC25482 | GSK269962A HCl | 2095432-71-4 | ROCK | ||
GSK269962A HCl (GSK269962B, GSK269962) is a selective ROCK(Rho-associated protein kinase) inhibitor with IC50 values of 1.6 and 4 nM for ROCK1 and ROCK2, respectively. | |||||
| GC38898 | CCG-222740 | 1922098-69-8 | ROCK | ||
CCG-222740 is a Rho/MRTF pathway inhibitor. CCG-222740 decreases the activation of stellate cells in vitro and in vivo, by reducing the levels of alpha smooth muscle actin(α-SMA) expression. | |||||
| GC37551 | ROCK inhibitor-2 | 1127308-52-4 | ROCK | ||
ROCK inhibitor-2是一种选择性Rho激酶(ROCK)抑制剂,抑制ROCK1和ROCK2的IC50值分别为17nM和2nM,具有抗肿瘤活性。 | |||||
