GlpBio

Roluperidone (CYR-101)

目录号: GC30206纯度: >99.50%同义词: CYR-101; MIN-101; MT-210
A dual antagonist of 5-HT2A and σ2 receptors
Roluperidone (CYR-101)
Cas No.: 359625-79-9
规格价格库存数量操作
1mg¥244.00现货
1
5mg¥635.00现货
1
10mg¥1,060.00现货
1
25mg¥1,924.00现货
1
50mg¥2,880.00现货
1
100mg¥4,028.00现货
1
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文献被引

本产品暂无引用记录;以下为 GlpBio 产品在 Nature / Cell / Science 等顶刊的客户引用样例
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    187(9):2288-2304 (2024)
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    183(7):1867-1883 (2020)
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    31, 1291–1307 (2021)

产品描述 Description

CYR-101 is a dual antagonist of the serotonin (5-HT) receptor subtype 5-HT2A and sigma-2 (σ2) receptors (Kis = 7.53 and 8.19 nM, respectively).1

1.Davidson, M., Saoud, J., Staner, C., et al.Efficacy and safety of MIN-101: A 12-week randomized, double-blind, placebo-controlled trial of a new drug in development for the treatment of negative symptoms in schizophreniaAm. J. Psychiatry174(12)1195-1202(2017)

产品文档 Product Documents

Purity:>99.50%

化学性质Chemical Properties

CAS 号
359625-79-9
同义词
CYR-101; MIN-101; MT-210
SMILES
O=C1N(CC2CCN(CC(C3=CC=C(F)C=C3)=O)CC2)CC4=C1C=CC=C4
分子式
C22H23FN2O2
分子量
366.43 g/mol
溶解性
DMSO : 33.33 mg/mL (90.96 mM);Water : < 0.1 mg/mL (insoluble)
保存条件
Store at -20°C
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
为了提高溶解度，请将管子加热至 37°C，然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案：配备蓝冰进行发货。所有其他可用尺寸：配备 RT，或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol