ACE
ACE(血管紧张素转换酶)
ACE, also known as angiotensin-converting enzyme, indirectly increases blood pressure by converting angiotensin I to angiotensin II and subsequently constricting the vessels.
ACE 相关产品(73)
- GC15493Enalaprilat DihydrateCAS: 84680-54-6纯度: >98.00%
Enalaprilat Dihydrate是一种具有口服活性的血管紧张素转换酶(ACE)抑制剂,在体内可迅速水解为活性代谢物Enalaprilat,Enalaprilat通过抑制血管紧张素II的生成,有效舒张血管,降低血压,并减轻心脏负荷。
- GA20760Angiotensin A (1-7)CAS: 1176306-10-7纯度: >98.50%
血管紧张素 A (1-7) 是肾素-血管紧张素系统 (RAS) 的成员,是一种血管活性肽,是 G 蛋白偶联受体 MrgD 的内源性配体。
- GC25723Perindopril L-ArginineCAS: 612548-45-5
Perindopril L-Argininel is a prodrug that is metabolized in the liver to its active diacid metabolite perindoprilat, which is rapidly and extensively absorbed, and become one of the highest tissue angiotensin-converting enzyme (ACE) affinities among the ACE inhibitors.
- GC30421Enalapril D5 maleate (MK-421 (D5 maleate))CAS: 349554-02-5
An internal standard for the quantification of enalapril
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC15493 | Enalaprilat Dihydrate | 84680-54-6 | >98.00% | |
Enalaprilat Dihydrate是一种具有口服活性的血管紧张素转换酶(ACE)抑制剂,在体内可迅速水解为活性代谢物Enalaprilat,Enalaprilat通过抑制血管紧张素II的生成,有效舒张血管,降低血压,并减轻心脏负荷。 | ||||
| GC15760 | Ramipril | 87333-19-5 | >98.00% | |
A prodrug from of ramiprilat | ||||
| GA20760 | Angiotensin A (1-7) | 1176306-10-7 | >98.50% | |
血管紧张素 A (1-7) 是肾素-血管紧张素系统 (RAS) 的成员,是一种血管活性肽,是 G 蛋白偶联受体 MrgD 的内源性配体。 | ||||
| GC10142 | Enalapril Maleate | 76095-16-4 | >99.50% | |
An ACE inhibitor | ||||
| GC10694 | Ramiprilat | 87269-97-4 | - | |
An ACE inhibitor | ||||
| GC11228 | Benazepril | 86541-75-5 | >98.00% | |
贝那普利,一种血管紧张素转换酶抑制剂,是一种用于治疗高血压的药物。 | ||||
| GC11266 | Lisinopril dihydrate | 83915-83-7 | >99.50% | |
An ACE inhibitor | ||||
| GC11560 | Resorcinolnaphthalein | 41307-63-5 | >98.50% | |
Activator of ACE2 | ||||
| GC11655 | Moexipril HCl | 82586-52-5 | >98.00% | |
A prodrug form of moexiprilat | ||||
| GC12368 | Quinapril HCl | 82586-55-8 | >99.00% | |
A prodrug form of quinaprilat | ||||
| GC12859 | Cilazapril | 88768-40-5 | - | |
A prodrug form of cilazaprilat | ||||
| GC13078 | Imidapril HCl | 89396-94-1 | >99.50% | |
A prodrug form of imidaprilat | ||||
| GC15166 | Perindopril Erbumine | 107133-36-8 | >99.50% | |
An orally active ACE inhibitor | ||||
| GC16192 | Diminazene Aceturate | 908-54-3 | >99.00% | |
An anti-protozoal diamidine | ||||
| GC16223 | Captopril | 62571-86-2 | >99.00% | |
Captopril是一种具有口服活性的血管紧张素转化酶(ACE)抑制剂,IC 50 值为0.025μM。 | ||||
| GC16307 | Lisinopril | 76547-98-3 | - | |
An ACE inhibitor | ||||
| GC16768 | Phosphoramidon Disodium Salt | 164204-38-0 | - | |
An inhibitor of NEP and NEP2 | ||||
| GC16871 | Perindopril | 82834-16-0 | - | |
An orally active ACE inhibitor | ||||
| GC17034 | Temocapril HCl | 110221-44-8 | >99.50% | |
A prodrug form of temocaprilat | ||||
| GC17667 | Cilazapril Monohydrate | 92077-78-6 | >99.00% | |
A prodrug form of cilazaprilat | ||||
| GC17941 | Benazepril HCl | 86541-74-4 | >99.50% / >98.00% | |
A prodrug of benazeprilat | ||||
| GC25723 | Perindopril L-Arginine | 612548-45-5 | - | |
Perindopril L-Argininel is a prodrug that is metabolized in the liver to its active diacid metabolite perindoprilat, which is rapidly and extensively absorbed, and become one of the highest tissue angiotensin-converting enzyme (ACE) affinities among the ACE inhibitors. | ||||
| GC30421 | Enalapril D5 maleate (MK-421 (D5 maleate)) | 349554-02-5 | - | |
An internal standard for the quantification of enalapril | ||||
| GC31354 | MLN-4760 | 305335-31-3 | >99.00% | |
MLN-4760是一种选择性的人血管紧张素转换酶2(ACE2;IC 50 =0.44nM)抑制剂,MLN-4760可高亲和力地结合ACE2的活性位点锌离子,模拟肽水解过程中的过渡态,从而阻断血管紧张素II向血管紧张素(1-7)的转化。 | ||||
