Others
Others 相关产品(2412)
- GA22830H-Pro-4MβNA . HClCAS: 100930-07-2
H-Pro-4Mβ;不适用。 HCl (H-Pro-4MβNA hydrochloride) 可用于 Fap 激活的抗肿瘤化合物的制备。
- GA23122L-2-Oxothiazolidine-4-carboxylic acidCAS: 19771-63-2纯度: >98.00%
A prodrug form of cysteine with antioxidant activity
- GA23477Relaxin H2 (human)CAS: 99489-94-8
Relaxin H2 is the major stored and circulating isoform of the peptide hormone relaxin in humans. This pregnancy hormone has also shown cardioprotective activity. The observed long-term effects of relaxin H2 on connective tissues may be due to alterations in the turnover of collagen and proteoglycans.
- GA23674Z-Ala-Ala-Asn-AMCCAS: 149697-16-5纯度: >98.50%
Z-Ala-Ala-Asn-AMC(Cbz-Ala-Ala-Asn-AMC)是一种在被蛋白酶切割后可释放高荧光强度AMC的合成荧光肽底物(Ex/Em: 380nm/430nm),被广泛用于天冬酰胺内肽酶(Legumain)活性的测定。
- GA23790Z-Glu-Tyr-OHCAS: 988-75-0纯度: >99.00%
Z-Glu-Tyr-OH可作为构建更复杂肽链的关键中间体,保护基团可在特定条件下选择性脱除,从而允许肽链的定向延伸。
- GA24007β-Endorphin (30-31) (bovine, camel, mouse, ovine)CAS: 13115-71-4纯度: >98.00%
β-内啡肽 (30-31) (牛、骆驼、小鼠、绵羊) (甘氨酰-L-谷氨酰胺),作为 β-内啡肽的酶裂解产物,显然是 β-内啡肽 (1-31) 的内源性拮抗剂) 在几个系统中。
- GC10104GlimepirideCAS: 93479-97-1纯度: >99.50% / >98.00%
Glimepiride为第二代磺酰脲类药物,可刺激胰岛β细胞释放胰岛素,作为单药或与二甲双胍、胰岛素联合用于治疗2型糖尿病。
- GC10274Atomoxetine HClCAS: 82248-59-7纯度: >99.50% / >98.00%
Atomoxetine HCl是一种强效、选择性的去甲肾上腺素摄取抑制剂,对去甲肾上腺素、血清素(5-HT)和多巴胺(DA)的K i 值分别为5、77和1451nM。
- GC10348Alendronate sodium hydrateCAS: 121268-17-5纯度: >98.00%
Alendronate sodium hydrate是含氮双膦酸盐,强力抑制骨吸收,常用于预防和治疗骨质疏松症的研究。
- GC10430Migalastat (GR181413A) hydrochlorideCAS: 75172-81-5纯度: >98.00% / >99.50%
Migalastat (GR181413A) hydrochloride是一种口服的α-半乳糖苷酶A竞争性抑制剂,IC 50 值为0.04μM。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GA22430 | H-Gly-D-Tyr-OH | 133706-65-7 | - | |
H-Gly-D-Tyr-OH 用于固相肽合成。 | ||||
| GA22476 | H-Gly-Leu-OH | 869-19-2 | >98.00% | |
甘氨酰-l-亮氨酸是一种二肽,可以是甘氨酰-亮氨酸二肽酶的常见底物。 | ||||
| GA22830 | H-Pro-4MβNA . HCl | 100930-07-2 | - | |
H-Pro-4Mβ;不适用。 HCl (H-Pro-4MβNA hydrochloride) 可用于 Fap 激活的抗肿瘤化合物的制备。 | ||||
| GA22964 | H-Tyr-Ala-OH | 730-08-5 | >99.50% | |
H-Tyr-Ala-OH (Tyrosylanine) 是一种含有 L-酪氨酸和 L-丙氨酸的二肽。 | ||||
| GA23032 | H-Val-βNA | 729-24-8 | - | |
H-Val-β;NA(L-缬氨酸 β;-萘酰胺)可用作氨肽酶和缬氨酸芳基酰胺酶底物。 | ||||
| GA23122 | L-2-Oxothiazolidine-4-carboxylic acid | 19771-63-2 | >98.00% | |
A prodrug form of cysteine with antioxidant activity | ||||
| GA23477 | Relaxin H2 (human) | 99489-94-8 | - | |
Relaxin H2 is the major stored and circulating isoform of the peptide hormone relaxin in humans. This pregnancy hormone has also shown cardioprotective activity. The observed long-term effects of relaxin H2 on connective tissues may be due to alterations in the turnover of collagen and proteoglycans. | ||||
| GA23674 | Z-Ala-Ala-Asn-AMC | 149697-16-5 | >98.50% | |
Z-Ala-Ala-Asn-AMC(Cbz-Ala-Ala-Asn-AMC)是一种在被蛋白酶切割后可释放高荧光强度AMC的合成荧光肽底物(Ex/Em: 380nm/430nm),被广泛用于天冬酰胺内肽酶(Legumain)活性的测定。 | ||||
| GA23790 | Z-Glu-Tyr-OH | 988-75-0 | >99.00% | |
Z-Glu-Tyr-OH可作为构建更复杂肽链的关键中间体,保护基团可在特定条件下选择性脱除,从而允许肽链的定向延伸。 | ||||
| GA24007 | β-Endorphin (30-31) (bovine, camel, mouse, ovine) | 13115-71-4 | >98.00% | |
β-内啡肽 (30-31) (牛、骆驼、小鼠、绵羊) (甘氨酰-L-谷氨酰胺),作为 β-内啡肽的酶裂解产物,显然是 β-内啡肽 (1-31) 的内源性拮抗剂) 在几个系统中。 | ||||
| GC10005 | SEP-0372814 | 1516895-53-6 | - | |
A PDE10A inhibitor | ||||
| GC10021 | CPI-360 | 1802175-06-9 | >99.00% | |
A selective EZH2 inhibitor | ||||
| GC10042 | Vitamin E | 59-02-9 | >99.00% / >98.00% | |
脂溶性维生素 | ||||
| GC10104 | Glimepiride | 93479-97-1 | >99.50% / >98.00% | |
Glimepiride为第二代磺酰脲类药物,可刺激胰岛β细胞释放胰岛素,作为单药或与二甲双胍、胰岛素联合用于治疗2型糖尿病。 | ||||
| GC10173 | ETP 45835 dihydrochloride | - | - | |
Mnk1/2 inhibitor | ||||
| GC10233 | BRD 7552 | 1137359-47-7 | >98.00% | |
An inducer of PDX1 expression | ||||
| GC10239 | Phenindione | 83-12-5 | >98.00% | |
An anticoagulant and vitamin K antagonist | ||||
| GC10259 | BRD4770 | 1374601-40-7 | >99.50% | |
An inhibitor of EHMT2/G9a | ||||
| GC10274 | Atomoxetine HCl | 82248-59-7 | >99.50% / >98.00% | |
Atomoxetine HCl是一种强效、选择性的去甲肾上腺素摄取抑制剂,对去甲肾上腺素、血清素(5-HT)和多巴胺(DA)的K i 值分别为5、77和1451nM。 | ||||
| GC10290 | Medrysone | 2668-66-8 | >98.50% | |
An anti-inflammatory steroid | ||||
| GC10318 | Hexa-D-arginine | 673202-67-0 | >99.50% | |
A furin inhibitor | ||||
| GC10348 | Alendronate sodium hydrate | 121268-17-5 | >98.00% | |
Alendronate sodium hydrate是含氮双膦酸盐,强力抑制骨吸收,常用于预防和治疗骨质疏松症的研究。 | ||||
| GC10427 | Tolperisone HCl | 3644-61-9 | >99.50% | |
An inhibitor of voltage-gated sodium channels | ||||
| GC10430 | Migalastat (GR181413A) hydrochloride | 75172-81-5 | >98.00% / >99.50% | |
Migalastat (GR181413A) hydrochloride是一种口服的α-半乳糖苷酶A竞争性抑制剂,IC 50 值为0.04μM。 | ||||
