NMDA Receptor
NMDA Receptor(NMDA受体)
NMDA (N-methyl-D-aspartate) receptor is a glutamate-gated cation channels that plays a vital role in regulating synaptic transmission, neuroplasticity and central nervous system development. It is involved in a range of physiological processes such as learning, memory and pain etc.
NMDA Receptor 相关产品(76)
- GC14357PMPA (NMDA antagonist)CAS: 113919-36-1
PMPA（NMDA 拮抗剂）是一种 NMDA 受体拮抗剂，对 NR2A、NR2B、NR2C 和 NR2D 的 Ki 值分别为 0.84、2.74、3.53 和 4.16 μM。
- GC15752CGP 78608 hydrochlorideCAS: 206648-13-7
CGP 78608 hydrochloride 是一种高效的选择性拮抗剂，作用于 NMDA 受体的甘氨酸结合位点，IC50 为 6 nM。
- GC16131Remacemide hydrochlorideCAS: 111686-79-4
Remacemide hydrochloride (FPL 12924AA) 是 Na+ 通道的中度抑制剂，是一种弱的非竞争性 NMDA 受体拮抗剂，对 MK-801 结合和 NMDA 电流的 IC50 分别为 68 μM 和 76 μM。
- GC16240MNI-caged-NMDACAS: 1227675-52-6
NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC14357 | PMPA (NMDA antagonist) | 113919-36-1 | - | |
PMPA（NMDA 拮抗剂）是一种 NMDA 受体拮抗剂，对 NR2A、NR2B、NR2C 和 NR2D 的 Ki 值分别为 0.84、2.74、3.53 和 4.16 μM。 | ||||
| GC14381 | Ro 8-4304 hydrochloride | 1312991-77-7 | - | |
NMDA receptor antagonist | ||||
| GC14414 | CIQ | 486427-17-2 | >98.00% | |
A subunit-selective NMDA receptor potentiator | ||||
| GC14442 | TCS 46b | 302799-86-6 | - | |
NR1A/NR2B NMDA receptor antagonist,orally active | ||||
| GC14470 | Arcaine sulfate | 14923-17-2 | >95.00% | |
An NMDA receptor antagonist | ||||
| GC14547 | Quinolinic acid | 89-00-9 | >99.00% | |
An excitotoxic agonist at NMDA receptors | ||||
| GC14598 | 5,7-Dichlorokynurenic acid sodium salt | 1184986-70-6 | - | |
An NMDA receptor antagonist | ||||
| GC14770 | TCN 213 | 556803-08-8 | - | |
TCN 213 是一种选择性的、可克服的、依赖甘氨酸的 GluN1/GluN2A NMDAR 拮抗剂，在 75、750、7500 nM 甘氨酸存在下，IC50 分别为 0.55、3.5、40 μM。 | ||||
| GC14782 | Ro 04-5595 hydrochloride | 64047-73-0 | - | |
NR2B-containing NMDA receptors antagonist | ||||
| GC14810 | L-701,324 | 142326-59-8 | >99.50% | |
An NMDA receptor antagonist | ||||
| GC14897 | DL-AP5 Sodium salt | 1303993-72-7 | - | |
A competitive NMDA antagonist | ||||
| GC15065 | TCN 201 | 852918-02-6 | >98.50% | |
An NR2A-selective NMDA receptor antagonist | ||||
| GC15112 | D-AP7 | 81338-23-0 | - | |
NMDA receptor antagonist | ||||
| GC15156 | Conantokin-T | 127476-26-0 | - | |
Non-competitive NMDA receptor antagonist | ||||
| GC15343 | Eliprodil | 119431-25-3 | >98.50% | |
An NMDA receptor antagonist | ||||
| GC15732 | Synthalin sulfate | 182285-12-7 | - | |
NMDA receptor antagonist | ||||
| GC15752 | CGP 78608 hydrochloride | 206648-13-7 | - | |
CGP 78608 hydrochloride 是一种高效的选择性拮抗剂，作用于 NMDA 受体的甘氨酸结合位点，IC50 为 6 nM。 | ||||
| GC16131 | Remacemide hydrochloride | 111686-79-4 | - | |
Remacemide hydrochloride (FPL 12924AA) 是 Na+ 通道的中度抑制剂，是一种弱的非竞争性 NMDA 受体拮抗剂，对 MK-801 结合和 NMDA 电流的 IC50 分别为 68 μM 和 76 μM。 | ||||
| GC16240 | MNI-caged-NMDA | 1227675-52-6 | - | |
NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group | ||||
| GC16272 | CGS 19755 | 110347-85-8 | >98.00% | |
NMDA receptor antagonist | ||||
| GC16315 | D-AP5 | 79055-68-8 | >98.00% | |
D-AP5是一种选择性N-甲基-D-天门冬胺酸（NMDA）受体拮抗剂，K d 值为1.4μM。 | ||||
| GC16776 | QNZ 46 | 1237744-13-6 | >98.00% | |
An antagonist of NR2C- and NR2D-subunit containing NMDA receptors | ||||
| GC16799 | 5,7-Dichlorokynurenic acid | 131123-76-7 | - | |
An NMDA receptor antagonist | ||||
| GC16915 | (2R,3S)-Chlorpheg | 140924-23-8 | - | |
NMDA receptor antagonist | ||||