Adrenergic Receptor
Adrenergic Receptor(肾上腺素能受体)
Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.
Adrenergic Receptor 相关产品(404)
- GC25140BisoprololCAS: 66722-44-9
Bisoprolol is a cardioselective β1-adrenergic blocking agent used for secondary prevention of myocardial infarction (MI), heart failure, angina pectoris and mild to moderate hypertension.
- GC25197Carvedilol EP IMpurity ECAS: 64464-07-9
Carvedilol is a nonselective beta blocker/alpha-1 blocker and used in management of congestive heart failure (CHF).
- GC25786PropafenoneCAS: 54063-53-5
Propafenone (SA-79) is an orally active sodium channel blocking agent and a beta-adrenoceptor (β-adrenergic receptor) antagonist. Propafenone offers a broad spectrum of activity in the treatment of cardiac arrhythmias.
- GC30092Salmeterol (GR33343X)CAS: 89365-50-4纯度: >99.50%
Salmeterol (Astmerole, GR-33343X, SN408D) is a long-acting beta2-adrenergic receptor agonist with Ki value of 1.5 nM for WT β2AR and shows very high selectivity for the WT β2AR(β1Ki/β2Ki ratio of approximately 1500).
- GC30273Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide)CAS: 960151-65-9纯度: >99.50%
Tedatioxetine (Lu AA24530) hydrobromide 可作为 5-HT2A、5-HT2C、5-HT3 和 α；1A-肾上腺素受体拮抗剂，可作为 5-羟色胺和去甲肾上腺素 (NE) 的首选三重再摄取抑制剂 (TRI)。
- GC30391Indoramin D5 (Indoramine D5)CAS: 57165-41-0
Indoramine D5 (Indoramine D5) 是氘标记的 Indoramin，它是一种哌啶类抗肾上腺素能药物。
- GC30396Piribedil D8 (ET-495 D8)CAS: 1398044-45-5
Piribedil D8 (ET-495 D8) (ET-495 D8) 是氘标记的 Piribedil，它是一种抗帕金森病药物。
- GC30405Tolazoline (Imidaline)CAS: 59-98-3
Tolazoline (Imidaline)(Imidaline) 是一种非选择性竞争性 α-adrenergic receptor 拮抗剂。
- GC30434Ivabradine D3 HydrochlorideCAS: 1217809-61-4
An internal standard for the quantification of ivabradine
- GC30474Benzquinamide (P2647)CAS: 63-12-7
Benzquinamide(P2647)是一种止吐剂,并可以与α2A,α2B,以及α2C肾上腺素能受体（α2-AR）结合，Ki值分别为1,365,691和545nM。
- GC30547ACTH 1-14 (Adrenocorticotropic Hormone Fragment 1-14)CAS: 25696-21-3
ACTH 1-14（促肾上腺皮质激素片段 1-14）是促肾上腺皮质激素的片段，可调节皮质醇和雄激素的产生。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC17884 | JP1302 | 80259-18-3 | >99.50% | |
JP1302 是一种选择性的、高亲和力的 α 2C 肾上腺受体 (α 2C -adrenoceptor) 的拮抗剂，其对人类 α 2C 受体的 K b 值为 16 nM，K i 为 28 nM。 | ||||
| GC17888 | Metipranolol | 22664-55-7 | >98.00% | |
A β-AR antagonist | ||||
| GC17974 | Latrepirdine dihydrochloride | 97657-92-6 | >99.50% / >98.00% | |
A neuroprotective agent | ||||
| GC17998 | Isoxsuprine (hydrochloride) | 579-56-6 | >99.50% | |
An adrenergic receptor modulator | ||||
| GC18327 | Todralazine (hydrochloride) | 3778-76-5 | >98.00% | |
A β 2 -adrenergic receptor antagonist | ||||
| GC25140 | Bisoprolol | 66722-44-9 | - | |
Bisoprolol is a cardioselective β1-adrenergic blocking agent used for secondary prevention of myocardial infarction (MI), heart failure, angina pectoris and mild to moderate hypertension. | ||||
| GC25197 | Carvedilol EP IMpurity E | 64464-07-9 | - | |
Carvedilol is a nonselective beta blocker/alpha-1 blocker and used in management of congestive heart failure (CHF). | ||||
| GC25385 | Esmolol | 81147-92-4 | - | |
Esmolol is a cardioselective beta1 receptor blocker with rapid onset, a very short duration of action, and no significant intrinsic sympathomimetic or membrane stabilising activity at therapeutic dosages. | ||||
| GC25412 | Fenoterol | 13392-18-2 | >98.00% / >99.50% | |
Fenoterol (Phenoterol) is a β2 adrenoreceptor agonist with bronchodilator activity. | ||||
| GC25484 | Guanabenz | 5051-62-7 | - | |
Guanabenz (GBZ, GA, Wytensin, Wy-8678,BR-750) is an orally active central alpha 2-adrenoceptor (α2 adrenergic receptor) agonist with antihypertensive action. | ||||
| GC25663 | Nebivolol | 118457-14-0 | - | |
Nebivolol (Bystolic,R 065824) is a β1 receptor blocker with nitric oxide-potentiating vasodilatory effect used in treatment of hypertension and also for left ventricular failure. | ||||
| GC25786 | Propafenone | 54063-53-5 | - | |
Propafenone (SA-79) is an orally active sodium channel blocking agent and a beta-adrenoceptor (β-adrenergic receptor) antagonist. Propafenone offers a broad spectrum of activity in the treatment of cardiac arrhythmias. | ||||
| GC30092 | Salmeterol (GR33343X) | 89365-50-4 | >99.50% | |
Salmeterol (Astmerole, GR-33343X, SN408D) is a long-acting beta2-adrenergic receptor agonist with Ki value of 1.5 nM for WT β2AR and shows very high selectivity for the WT β2AR(β1Ki/β2Ki ratio of approximately 1500). | ||||
| GC30188 | Dapiprazole hydrochloride | 72822-13-0 | >99.50% | |
An α-adrenergic receptor antagonist | ||||
| GC30273 | Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) | 960151-65-9 | >99.50% | |
Tedatioxetine (Lu AA24530) hydrobromide 可作为 5-HT2A、5-HT2C、5-HT3 和 α；1A-肾上腺素受体拮抗剂，可作为 5-羟色胺和去甲肾上腺素 (NE) 的首选三重再摄取抑制剂 (TRI)。 | ||||
| GC30391 | Indoramin D5 (Indoramine D5) | 57165-41-0 | - | |
Indoramine D5 (Indoramine D5) 是氘标记的 Indoramin，它是一种哌啶类抗肾上腺素能药物。 | ||||
| GC30396 | Piribedil D8 (ET-495 D8) | 1398044-45-5 | - | |
Piribedil D8 (ET-495 D8) (ET-495 D8) 是氘标记的 Piribedil，它是一种抗帕金森病药物。 | ||||
| GC30405 | Tolazoline (Imidaline) | 59-98-3 | - | |
Tolazoline (Imidaline)(Imidaline) 是一种非选择性竞争性 α-adrenergic receptor 拮抗剂。 | ||||
| GC30434 | Ivabradine D3 Hydrochloride | 1217809-61-4 | - | |
An internal standard for the quantification of ivabradine | ||||
| GC30458 | Teoprolol | 65184-10-3 | - | |
Teoprolol是一种β-adrenergic受体阻滞剂。 | ||||
| GC30474 | Benzquinamide (P2647) | 63-12-7 | - | |
Benzquinamide(P2647)是一种止吐剂,并可以与α2A,α2B,以及α2C肾上腺素能受体（α2-AR）结合，Ki值分别为1,365,691和545nM。 | ||||
| GC30547 | ACTH 1-14 (Adrenocorticotropic Hormone Fragment 1-14) | 25696-21-3 | - | |
ACTH 1-14（促肾上腺皮质激素片段 1-14）是促肾上腺皮质激素的片段，可调节皮质醇和雄激素的产生。 | ||||
| GC30665 | D2343 | 72734-63-5 | - | |
D2343是一种β2肾上腺素能受体激动剂，也是一种α1-肾上腺素能受体抑制剂。 | ||||
| GC30679 | Fiduxosin | 208993-54-8 | - | |
Fiduxosin是一种α1-adrenoceptor拮抗剂，对α1a-adrenoceptor，α1b-adrenoceptor和α1d-adrenoceptor的Ki值分别为0.160nM，24.9nM和0.920nM。 | ||||