Adrenergic Receptor
Adrenergic Receptor(肾上腺素能受体)
Adrenergic receptor is a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine and epinephrine.
Adrenergic Receptor 相关产品(404)
- GC12206HEAT hydrochlorideCAS: 30007-39-7
HEAT (BE2254) hydrochloride 是一种选择性 alpha 1 adrenergic receptor 拮抗剂。
- GC12227SR 59230A hydrochlorideCAS: 1135278-41-9纯度: >99.50% / >98.00%
SR 59230A hydrochloride是一种高效、选择性的β3-肾上腺素受体拮抗剂，对β3、β1和β2受体的IC 50 值分别为40nM、408nM和648nM。
- GC12463(S)-(-)-AtenololCAS: 93379-54-5纯度: >99.50%
(S)-(-)-Atenolol是一种强效的β-肾上腺素能受体阻滞剂。(S)-(-)-Atenolol是Atenolol的S(-)对映体，Atenolol的R(+)对映体几乎不具有β受体阻滞剂活性。
- GC12778Clenbuterol (hydrochloride)CAS: 21898-19-1纯度: >99.00%
Clenbuterol (hydrochloride)是一种β 2 -肾上腺素受体激动剂，EC 50 为31.9nM。Clenbuterol (hydrochloride)可有效抑制脂多糖（LPS）诱导的TNF-α和IL-1β释放。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC11077 | Imiloxan hydrochloride | 81167-22-8 | >98.00% | |
α2-adrenoceptor antagonist | ||||
| GC11130 | Indacaterol Maleate | 753498-25-8 | >98.00% | |
A long-acting β 2 -adrenergic receptor agonist | ||||
| GC11174 | ZD 2079 | 178600-17-4 | - | |
ZD 2079 (ZD2079 hydrochloride) 是一种有效的 β3-adrenoceptor 激动剂，对去氧肾上腺素预收缩的大鼠肠系膜动脉的 pD2 为 3.72。 | ||||
| GC11239 | Midodrine (hydrochloride) | 43218-56-0 | >99.00% | |
A prodrug form of desglymidodrine | ||||
| GC11373 | Scopine HCl | 85700-55-6 | >98.00% | |
A metabolite of scopolamine | ||||
| GC11385 | G-Protein antagonist peptide | 143675-79-0 | - | |
G-蛋白拮抗肽是抑制G蛋白与其受体结合的P物质相关肽。 | ||||
| GC11479 | Xylometazoline HCl | 1218-35-5 | >99.50% | |
An α-adrenergic receptor agonist | ||||
| GC11824 | Asenapine | 65576-45-6 | >98.50% | |
An atypical antipsychotic | ||||
| GC11913 | ST 91 | 4749-61-5 | - | |
α2-adrenoceptor agonist | ||||
| GC11937 | (R)-(+)-m-Nitrobiphenyline oxalate | 945618-97-3 | - | |
α2C-AR (adrenoceptor) agonist | ||||
| GC11952 | (R)-(+)-Atenolol | 56715-13-0 | >99.00% | |
An enantiomer of (±)-atenolol | ||||
| GC12023 | Celiprolol (hydrochloride) | 57470-78-7 | >98.00% | |
A β 1 adrenergic receptor antagonist | ||||
| GC12042 | DSP-4 | 40616-75-9 | >98.00% | |
A noradrenergic neurotoxin | ||||
| GC12073 | Xylazine | 7361-61-7 | >98.00% | |
Xylazine（赛拉嗪；BAY 1470）是一种有效的α2-肾上腺素受体的强激动剂，在兽医学中广泛用作镇静剂，还能诱导肌肉松弛。 | ||||
| GC12144 | (R)-(-)-Niguldipine hydrochloride | - | - | |
L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist | ||||
| GC12206 | HEAT hydrochloride | 30007-39-7 | - | |
HEAT (BE2254) hydrochloride 是一种选择性 alpha 1 adrenergic receptor 拮抗剂。 | ||||
| GC12227 | SR 59230A hydrochloride | 1135278-41-9 | >99.50% / >98.00% | |
SR 59230A hydrochloride是一种高效、选择性的β3-肾上腺素受体拮抗剂，对β3、β1和β2受体的IC 50 值分别为40nM、408nM和648nM。 | ||||
| GC12243 | HOKU-81 | 58020-43-2 | - | |
HOKU-81 (4-Hydroxytulobuterol) 是 Tulobuterol 的代谢物之一。 | ||||
| GC12293 | Perphenazine | 58-39-9 | >99.50% | |
A typical antipsychotic | ||||
| GC12463 | (S)-(-)-Atenolol | 93379-54-5 | >99.50% | |
(S)-(-)-Atenolol是一种强效的β-肾上腺素能受体阻滞剂。(S)-(-)-Atenolol是Atenolol的S(-)对映体，Atenolol的R(+)对映体几乎不具有β受体阻滞剂活性。 | ||||
| GC12626 | Cimaterol | 54239-37-1 | >98.00% | |
A β-adrenergic agonist | ||||
| GC12761 | ICI 89406 | 53671-71-9 | - | |
ICI 89406 是一种选择性 β1 肾上腺素能受体拮抗剂，适合用正电子发射器标记，用于 PET。 | ||||
| GC12778 | Clenbuterol (hydrochloride) | 21898-19-1 | >99.00% | |
Clenbuterol (hydrochloride)是一种β 2 -肾上腺素受体激动剂，EC 50 为31.9nM。Clenbuterol (hydrochloride)可有效抑制脂多糖（LPS）诱导的TNF-α和IL-1β释放。 | ||||
| GC12823 | (R,S)-Atenolol | 29122-68-7 | >99.50% | |
A β 1 -AR antagonist | ||||