Thyroid hormone Receptor
Thyroid hormone Receptor(甲状腺激素受体)
Thyroid hormone receptor is a nuclear hormone receptor that activates or represses transcriptioin. It has effects on heart rate, lipid and lipoprotein metabolism.
Thyroid hormone Receptor 相关产品(65)
- GC10413Thyroid Hormone Receptor Antagonist (1-850)CAS: 251310-57-3
Blocks T3 binding to the thyroid hormone receptor
- GC11268L-ThyroxineCAS: 51-48-9纯度: >98.00%
L-Thyroxine是一种合成甲状腺激素，可模拟甲状腺分泌的天然甲状腺素，对调节新陈代谢、促进生长发育等起着关键作用。L-Thyroxine常用于治疗甲状腺功能减退症及其他甲状腺相关疾病。
- GC12409Liothyronine SodiumCAS: 55-06-1纯度: >99.00%
Liothyronine sodium 是一种强效的甲状腺激素受体TRα和TRβ激动剂，其 Ki 值为 2.33nM。
- GC17983TaltirelinCAS: 103300-74-9纯度: >99.00%
Taltirelin (TA0910) 是促甲状腺素释放激素受体 (TRH-R) 的超级激动剂，IC50 为 910 nM，EC50 为 36 nM，可刺激细胞溶质 Ca2+ 浓度（Ca2+ 释放）的增加。
- GC186963,5-Diiodothyropropionic AcidCAS: 1158-10-7纯度: >98.00%
An inotropic thyroid hormone analogue of L-thyroxine
- GC26431Pentacosafluorotridecanoic AcidCAS: 72629-94-8纯度: >97.00%
Perfluorotridecanoic Acid (Perfluorinated Compound (PFC)) is a perfluorinated alkyl acid (PFAA) and a possible organic pollutant.
- GC31328Thyroxine sulfate (T4 Sulfate)CAS: 77074-49-8纯度: >99.50%
硫酸甲状腺素 (T4 Sulfate) 是一种甲状腺激素代谢物。
- GC31402TR antagonist 1CAS: 500794-88-7纯度: >98.50%
TRantagonist1是高亲和力的甲状腺激素受体(thyroidhormonereceptor(TR))拮抗剂，对TRα和TRβ的IC50值分别为36和22nM。
- GC33845Protirelin Acetate (TRF Acetate)CAS: 120876-23-5纯度: >98.00%
Protirelin (Thyroliberin, Lopremone, Synthetic TRH, Thyrotropin-releasing hormone, Rifathyroin) is a tripeptide that stimulates the release of thyrotropin and prolactin.
- GC36465LiothyronineCAS: 6893-02-3纯度: >98.00%
An thyroid hormone which binds to TRβ1, and activates its activity
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GA20967 | Boc-D-His-OH | 50654-94-9 | - | |
An amino acid building block | ||||
| GA23395 | pTH (1-34) (rat) | 98614-76-7 | >95.00% | |
pTH (1-34)（大鼠）是一种甲状旁腺激素。 | ||||
| GC10384 | 3,3',5'-Triiodo-L-thyronine | 5817-39-0 | - | |
A thyroid hormone variant | ||||
| GC10413 | Thyroid Hormone Receptor Antagonist (1-850) | 251310-57-3 | - | |
Blocks T3 binding to the thyroid hormone receptor | ||||
| GC11268 | L-Thyroxine | 51-48-9 | >98.00% | |
L-Thyroxine是一种合成甲状腺激素，可模拟甲状腺分泌的天然甲状腺素，对调节新陈代谢、促进生长发育等起着关键作用。L-Thyroxine常用于治疗甲状腺功能减退症及其他甲状腺相关疾病。 | ||||
| GC12409 | Liothyronine Sodium | 55-06-1 | >99.00% | |
Liothyronine sodium 是一种强效的甲状腺激素受体TRα和TRβ激动剂，其 Ki 值为 2.33nM。 | ||||
| GC12903 | Sobetirome | 211110-63-3 | >98.00% | |
Sobetirome是一种甲状腺激素受体β（TRβ）选择性激动剂，对TRβ-1的EC 50 为0.16μM。 | ||||
| GC15001 | Tiratricol | 51-24-1 | >99.50% / >98.00% | |
A thyroid hormone receptor agonist | ||||
| GC17983 | Taltirelin | 103300-74-9 | >99.00% | |
Taltirelin (TA0910) 是促甲状腺素释放激素受体 (TRH-R) 的超级激动剂，IC50 为 910 nM，EC50 为 36 nM，可刺激细胞溶质 Ca2+ 浓度（Ca2+ 释放）的增加。 | ||||
| GC18205 | 3,5-Diiodothyroacetic Acid | 1155-40-4 | >98.00% | |
A thyroid hormone derivative | ||||
| GC18243 | MGL-3196 | 920509-32-6 | >99.50% / >99.00% | |
MGL-3196是一种高选择性的口服甲状腺激素受体β（THRβ）激动剂，EC 50 为0.21μM。 | ||||
| GC18696 | 3,5-Diiodothyropropionic Acid | 1158-10-7 | >98.00% | |
An inotropic thyroid hormone analogue of L-thyroxine | ||||
| GC26431 | Pentacosafluorotridecanoic Acid | 72629-94-8 | >97.00% | |
Perfluorotridecanoic Acid (Perfluorinated Compound (PFC)) is a perfluorinated alkyl acid (PFAA) and a possible organic pollutant. | ||||
| GC30588 | Protirelin (Synthetic thyrotropin-releasing factor) | 24305-27-9 | - | |
A tropic hormone | ||||
| GC31328 | Thyroxine sulfate (T4 Sulfate) | 77074-49-8 | >99.50% | |
硫酸甲状腺素 (T4 Sulfate) 是一种甲状腺激素代谢物。 | ||||
| GC31402 | TR antagonist 1 | 500794-88-7 | >98.50% | |
TRantagonist1是高亲和力的甲状腺激素受体(thyroidhormonereceptor(TR))拮抗剂，对TRα和TRβ的IC50值分别为36和22nM。 | ||||
| GC31616 | KAT681 (T0681) | 373641-87-3 | - | |
KAT681 (T0681) 是一种肝脏选择性的拟甲状腺素。 | ||||
| GC32415 | PCO371 | 1613373-33-3 | >95.00% | |
PCO371是一种具有口服活性的小分子PTHR1完全激动剂，PCO371结合在PTH1R与Gs蛋白的胞内界面上。 | ||||
| GC33764 | Eprotirome (KB2115) | 355129-15-6 | >99.50% | |
A thyroid hormone mimetic | ||||
| GC33845 | Protirelin Acetate (TRF Acetate) | 120876-23-5 | >98.00% | |
Protirelin (Thyroliberin, Lopremone, Synthetic TRH, Thyrotropin-releasing hormone, Rifathyroin) is a tripeptide that stimulates the release of thyrotropin and prolactin. | ||||
| GC34822 | T3-ATA S-isomer | 2438721-48-1 | - | |
T3-ATAS-isomer是T3-ATA的S-异构体，是甲状腺激素的活性形式。 | ||||
| GC34824 | T4-ATA S-isomer | 2448470-97-9 | >99.50% | |
T4-ATAS-isomer是T4-ATA的S-异构体，是甲状腺激素的活性形式。 | ||||
| GC36465 | Liothyronine | 6893-02-3 | >98.00% | |
An thyroid hormone which binds to TRβ1, and activates its activity | ||||
| GC36487 | L-Thyroxine sodium salt pentahydrate | 6106-07-6 | >98.00% | |
A synthetic form of thyroxine | ||||