Histamine Receptor
Histamine Receptor(组胺受体)
Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.
Histamine Receptor 相关产品(236)
- GC11046JNJ 5207852 dihydrochlorideCAS: 398473-34-2纯度: >98.00%
Selective, non-imidazole histamine H 3 R antagonist
- GC11121A 943931 dihydrochlorideCAS: 1227675-50-4
Antagonist of histamine H4 receptor,potent and selective
- GC11220Imetit dihydrobromideCAS: 32385-58-3纯度: >98.00% / >95.00%
A histamine H 3 and H 4 receptor agonist
- GC11695CinnarizineCAS: 298-57-7纯度: >99.50%
A calcium channel inhibitor and histamine H 4 receptor antagonist
- GC11809(R)-(-)-α-Methylhistamine dihydrobromideCAS: 868698-49-1纯度: >99.00% / >98.00%
(R)-(-)-α-Methylhistamine dihydrobromide 是一种有效的、选择性的、可穿透脑的 H3 组胺受体激动剂，Kd 为 50.3 nM。
- GC12030Epinastine HClCAS: 108929-04-0纯度: >99.00%
A histamine H 1 receptor antagonist and mast cell stabilizer
- GC12085ROS 234 dioxalateCAS: 184576-87-2
ROS 234 dioxalate 是一种有效的 H3 拮抗剂，对豚鼠回肠 H3 受体的 pKB 为 9.46，对大鼠大脑皮层 H3 受体的 pKi 为 8.90，在体外的 ED50 为 19.12 mg/kg (ip)大鼠大脑皮层。
- GC13266trans-Triprolidine hydrochlorideCAS: 550-70-9
trans-Triprolidine hydrochloride 是一种具有口服活性的组胺 H1 拮抗剂。
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC11046 | JNJ 5207852 dihydrochloride | 398473-34-2 | >98.00% | |
Selective, non-imidazole histamine H 3 R antagonist | ||||
| GC11121 | A 943931 dihydrochloride | 1227675-50-4 | - | |
Antagonist of histamine H4 receptor,potent and selective | ||||
| GC11220 | Imetit dihydrobromide | 32385-58-3 | >98.00% / >95.00% | |
A histamine H 3 and H 4 receptor agonist | ||||
| GC11291 | Mepyramine maleate | 59-33-6 | >99.50% | |
Mepyramine maleate主要用作H 1 拮抗剂，其亲和pK d 为9.4。 | ||||
| GC11330 | Tiotidine | 69014-14-8 | >98.50% | |
Tiotidine (ICI 125211) 是一种有效的选择性组胺 H2 受体拮抗剂（豚鼠右心房的 pA2=7.3-7.8）。 | ||||
| GC11695 | Cinnarizine | 298-57-7 | >99.50% | |
A calcium channel inhibitor and histamine H 4 receptor antagonist | ||||
| GC11809 | (R)-(-)-α-Methylhistamine dihydrobromide | 868698-49-1 | >99.00% / >98.00% | |
(R)-(-)-α-Methylhistamine dihydrobromide 是一种有效的、选择性的、可穿透脑的 H3 组胺受体激动剂，Kd 为 50.3 nM。 | ||||
| GC11883 | Dimaprit dihydrochloride | 23256-33-9 | - | |
A histamine H 2 receptor agonist | ||||
| GC12030 | Epinastine HCl | 108929-04-0 | >99.00% | |
A histamine H 1 receptor antagonist and mast cell stabilizer | ||||
| GC12085 | ROS 234 dioxalate | 184576-87-2 | - | |
ROS 234 dioxalate 是一种有效的 H3 拮抗剂，对豚鼠回肠 H3 受体的 pKB 为 9.46，对大鼠大脑皮层 H3 受体的 pKi 为 8.90，在体外的 ED50 为 19.12 mg/kg (ip)大鼠大脑皮层。 | ||||
| GC12238 | Oxomemazine | 3689-50-7 | - | |
Oxomemazine 是一种基于吩噻嗪的组胺 H1 受体阻滞剂，具有明显的抗毒蕈碱特性。 | ||||
| GC12265 | Iodophenpropit dihydrobromide | 145196-87-8 | - | |
A histamine H 3 receptor antagonist | ||||
| GC12293 | Perphenazine | 58-39-9 | >99.50% | |
A typical antipsychotic | ||||
| GC12371 | JNJ 10181457 dihydrochloride | 544707-19-9 | - | |
Histamine H3 receptor antagonist | ||||
| GC12472 | Amthamine dihydrobromide | 142457-00-9 | - | |
A histamine H 2 receptor agonist | ||||
| GC12737 | 4-Methylhistamine dihydrochloride | 36376-47-3 | >95.00% | |
A histamine H 4 receptor agonist | ||||
| GC12749 | Conessine | 546-06-5 | - | |
Conessine是一种甾体生物碱，作为强效、选择性的组胺H3受体拮抗剂（pK i =8.27）。 | ||||
| GC12892 | Doxepin (hydrochloride) | 1229-29-4 | >98.00% | |
A tricyclic antidepressant | ||||
| GC12966 | Immepip dihydrobromide | 164391-47-3 | >98.00% | |
Immepip dihydrobromide是一种强效且特异性的H3受体激动剂。 | ||||
| GC13024 | Metiamide | 34839-70-8 | - | |
Metiamide (SK&F 92058) 是一种组胺 H2 受体拮抗剂，由另一种 H2 拮抗剂布立马胺发展而来。 | ||||
| GC13266 | trans-Triprolidine hydrochloride | 550-70-9 | - | |
trans-Triprolidine hydrochloride 是一种具有口服活性的组胺 H1 拮抗剂。 | ||||
| GC13388 | Zolantidine dimaleate | 104076-39-3 | - | |
H2 receptor antagonist | ||||
| GC13465 | Chlorcyclizine (hydrochloride) | 14362-31-3 | >99.50% | |
A histamine H 1 antagonist | ||||
| GC13496 | Thioperamide | 106243-16-7 | - | |
A histamine H 3 receptor antagonist | ||||