5-HT Receptor(5-羟色胺受体)
5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.
Products for 5-HT Receptor
- Cat.No. 产品名称 Information
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GC33344
WAY 163909
(8AR,11AR)-9H-4,5,6,7,8A,10,11,11A-八氢环戊并[4,5]吡咯并[3,2,1-JK][1,4]苯并二氮杂卓
WAY163909是有效的且有选择性的5-HT(2C)receptor激动剂,Ki值为10.5±1.1nM。 -
GC50213
WAY 181187 oxalate
SAX-187 oxalate
WAY-181187 (SAX-187) oxalate 是一种有效的选择性全 5-HT6 受体激动剂,Ki 为 2.2 nM,EC50 为 6.6 nM。 -
GC10108
WAY-100635
WAY 100635; WAY100635
A serotonin 5-HT1A antagonist -
GC15754
WAY-100635 Maleate
A serotonin 5-HT1A antagonist
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GC16270
WAY-100635 maleate salt
WAY 100635 maleate salt; WAY100635 maleate salt
A serotonin 5-HT1A antagonist -
GC45157
WAY-161503
WAY161503盐酸盐
A 5-HT2C receptor agonist -
GC31041
Wf-516
Wf-516是一种5-HTreuptake的抑制剂,同时为5-HT1A和5-HT2A受体拮抗剂,对人体5-HT1A和5-HT2A受体的Ki值分别为5nM和40nM,具有抗抑郁作用。
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GC14743
WY 45233 succinate
去甲文拉法辛(O-去甲文拉法辛)琥珀酸,O-Desmethylvenlafaxine succinate; Wy-45233 succinate
serotonin and noradrenalin reuptake inhibitor -
GC50027
Xaliproden hydrochloride
盐酸扎利罗登,SR57746A; SR57746 hydrochloride
A 5-HT1A receptor agonist -
GN10074
Xanthotoxol
花椒毒醇,8-Hydroxypsoralen
A coumarin with diverse biological activities -
GC19389
YL0919
YL0919
YL0919 (YL0919) 是一种具有双重活性的口服抗抑郁药,作为高度选择性的 5-HT 摄取阻滞剂和有效的 5-HT1Areceptor 激动剂 (Ki=0.19 nM)。 -
GC31503
YM348
YM348是一种口服有效的5-HT2C受体激动剂,对克隆的人类5-HT2C受体具有高亲和力,Ki为0.89nM。
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GC31203
Zatosetron maleate (LY 277359 maleate)
扎托司琼马来酸盐; LY 277359 maleate
Zatosetron maleate (LY 277359 maleate) 是一种有效的选择性 5HT3 受体拮抗剂。 -
GC10630
Zimelidine dihydrochloride
齐美利定二盐酸盐
5-HT re-uptake inhibitor
-
GC11020
Ziprasidone
齐拉西酮; CP-88059
齐拉西酮 (CP-88059) 是一种口服活性抗精神病药,是一种 5-HT 和多巴胺受体拮抗剂的组合。 -
GC61389
Ziprasidone amino acid
齐拉西酮开环物,氨基酸杂质,Ziprasidone Impurity C; Ziprasidone open ring impurity
Ziprasidoneaminoacid(ZiprasidoneImpurityC)是Ziprasidone的杂质。Ziprasidone是5-HT和多巴胺(dopaminereceptor)受体拮抗剂,具有抗精神病活性。 -
GC37969
Ziprasidone D8
齐拉西酮-D8,CP-88059 D8
An internal standard for the quantification of ziprasidone -
GC11521
Ziprasidone HCl
盐酸齐拉西酮; CP-88059 hydrochloride
An atypical antipsychotic -
GC13627
Ziprasidone hydrochloride monohydrate
盐酸齐拉西酮水合物; CP 88059 hydrochloride monohydrate
An atypical antipsychotic -
GC17808
Zolmitriptan
佐米曲普坦,BW-311C90; 311C90
An agonist of 5-HT1B and 5-HT1D receptors