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5-HT Receptor(5-羟色胺受体)

5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.

Products for  5-HT Receptor

  1. Cat.No. 产品名称 Information
  2. GC33344 WAY 163909

    (8AR,11AR)-9H-4,5,6,7,8A,10,11,11A-八氢环戊并[4,5]吡咯并[3,2,1-JK][1,4]苯并二氮杂卓

    WAY163909是有效的且有选择性的5-HT(2C)receptor激动剂,Ki值为10.5±1.1nM。
  3. GC50213 WAY 181187 oxalate

    SAX-187 oxalate

    WAY-181187 (SAX-187) oxalate 是一种有效的选择性全 5-HT6 受体激动剂,Ki 为 2.2 nM,EC50 为 6.6 nM。
  4. GC10108 WAY-100635

    WAY 100635; WAY100635

    A serotonin 5-HT1A antagonist
  5. GC15754 WAY-100635 Maleate A serotonin 5-HT1A antagonist
  6. GC16270 WAY-100635 maleate salt

    WAY 100635 maleate salt; WAY100635 maleate salt

    A serotonin 5-HT1A antagonist
  7. GC45157 WAY-161503

    WAY161503盐酸盐

    A 5-HT2C receptor agonist
  8. GC31041 Wf-516 Wf-516是一种5-HTreuptake的抑制剂,同时为5-HT1A和5-HT2A受体拮抗剂,对人体5-HT1A和5-HT2A受体的Ki值分别为5nM和40nM,具有抗抑郁作用。
  9. GC14743 WY 45233 succinate

    去甲文拉法辛(O-去甲文拉法辛)琥珀酸,O-Desmethylvenlafaxine succinate; Wy-45233 succinate

    serotonin and noradrenalin reuptake inhibitor
  10. GC50027 Xaliproden hydrochloride

    盐酸扎利罗登,SR57746A; SR57746 hydrochloride

    A 5-HT1A receptor agonist
  11. GN10074 Xanthotoxol

    花椒毒醇,8-Hydroxypsoralen

    A coumarin with diverse biological activities
  12. GC19389 YL0919

    YL0919

    YL0919 (YL0919) 是一种具有双重活性的口服抗抑郁药,作为高度选择性的 5-HT 摄取阻滞剂和有效的 5-HT1Areceptor 激动剂 (Ki=0.19 nM)。
  13. GC31503 YM348 YM348是一种口服有效的5-HT2C受体激动剂,对克隆的人类5-HT2C受体具有高亲和力,Ki为0.89nM。
  14. GC31203 Zatosetron maleate (LY 277359 maleate)

    扎托司琼马来酸盐; LY 277359 maleate

    Zatosetron maleate (LY 277359 maleate) 是一种有效的选择性 5HT3 受体拮抗剂。
  15. GC10630 Zimelidine dihydrochloride

    齐美利定二盐酸盐

    5-HT re-uptake inhibitor

  16. GC11020 Ziprasidone

    齐拉西酮; CP-88059

    齐拉西酮 (CP-88059) 是一种口服活性抗精神病药,是一种 5-HT 和多巴胺受体拮抗剂的组合。
  17. GC61389 Ziprasidone amino acid

    齐拉西酮开环物,氨基酸杂质,Ziprasidone Impurity C; Ziprasidone open ring impurity

    Ziprasidoneaminoacid(ZiprasidoneImpurityC)是Ziprasidone的杂质。Ziprasidone是5-HT和多巴胺(dopaminereceptor)受体拮抗剂,具有抗精神病活性。
  18. GC37969 Ziprasidone D8

    齐拉西酮-D8,CP-88059 D8

    An internal standard for the quantification of ziprasidone
  19. GC11521 Ziprasidone HCl

    盐酸齐拉西酮; CP-88059 hydrochloride

    An atypical antipsychotic
  20. GC13627 Ziprasidone hydrochloride monohydrate

    盐酸齐拉西酮水合物; CP 88059 hydrochloride monohydrate

    An atypical antipsychotic
  21. GC17808 Zolmitriptan

    佐米曲普坦,BW-311C90; 311C90

    An agonist of 5-HT1B and 5-HT1D receptors

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