Cancer Biology(癌症生物学)
- Cancer Biology Peptides(33)
- Ras-like GTPases(11)
- Leukemia(1)
- Others(60)
- Tumor Microenvironment(43)
- Cell Migration & Metastasis(42)
- Cell Death(6)
- Cat.No. 产品名称 Information
-
GC49285
Adenosine 5’-methylenediphosphate (hydrate)
Adenosine 5'-(α,β-methylene)diphosphate, AMP-CP, APCP, 5'-APCP
An inhibitor of ecto-5’-nucleotidase -
GP10113
Adrenomedullin (1-12), human
H2N-Tyr-Arg-Gln-Ser-Met-Asn-Asn-Phe-Gln-Gly-Leu-Arg-OH
An N-terminal fragment of adrenomedullin
-
GC42740
Adrenomedullin (1-52) (human) (trifluoroacetate salt)
Adrenomedullin (1-52)-NH2
Adrenomedullin (1-52) is a peptide with diverse biological activities. -
GP10109
Adrenorphin
H2N-Tyr-Gly-Gly-Phe-Met-Arg-Arg-Val-amide
Adrenorphin 是一种阿片样物质八肽,作为 μ-阿片样物质受体的有效激动剂,Ki 为 12 nM。
-
GC11189
AI-10-49
AI-10-49 是一种蛋白质-蛋白质相互作用抑制剂,选择性结合 CBFβ-SMMHC 并破坏其与 RUNX1 的结合,FRET IC50 为 0.26 uM。
-
GC46825
Alachlor
甲草胺
An herbicide -
GC26242
Alexa Fluor 594 labeled Concanavalin A
刀豆蛋白A来源于洋刀豆(刀豆),Alexa Fluor 594标记;Alexa Fluor 594标记的刀豆凝集素A;Alexa Fluor594标记的刀豆球蛋白A;Ale lexa Flu or 594标记的伴刀豆球蛋白A;
刀豆蛋白A (Concanavalin ACon A) ,来源于Canavalia ensiformis洋豆 (刀豆),是一种凝集素蛋白 (Mw 104kDa) 。
-
GC92051
Alkyne-Cyclo(RGDyK) (trifluoroacetate salt)
Alkyne-c(RGDyK)
Alkyne-Cyclo(RGDyK) (trifluoroacetate salt)是αVβ3整合素环肽配体环(RGDyK)的可点击形式。 -
GC18482
all-trans-5,6-epoxy Retinoic Acid
5,6-epoxy-atRA, 5,6-epoxy RA
An agonist of RAR isoforms -
GC91986
Allolithocholic Acid-d4
3α-hydroxy-5α-Cholanoic Acid-d4; allo-LCA-d4
Allolithocholic Acid-d4旨在用作GC或LC-MS定量异石胆酸的内标。 -
GC74502
Alnuctamab
EM901; CC-93269
Alnuctamab(EM901)是一种不对称的2臂人源化IgG T细胞接合剂(TCE)。 -
GC49046
Altemicidin
(-)-Altemicidin
A monoterpene alkaloid with acaricidal and anticancer activities -
GC63535
ALV2
ALV2 是一种有效和选择性的 Helios 降解剂。ALV2 可以结合 CRBN,IC50 为 0.57 μM。Helios 是一种锌指转录因子,可以在炎症性肿瘤微环境中维持稳定的 Treg 细胞表型。
-
GC46835
Alyssin
5-Methylsulfinylpentyl isothiocyanate, 5-Methylsulfinylpentyl ITC
An isothiocyanate with diverse biological activities -
GP10057
Amyloid β-Peptide (10-20) (human)
Tyr-Glu-Val-His-His-Gln-Lys-Leu-Val-Phe-Phe
Amyloid β-Peptide (10-20) (human) 是 Amyloid-β 的片段;肽,可用于神经系统疾病的研究。
-
GC46853
Anagyrine
安纳基林,(-)-Anagyrine; Monolupine; Rhombinine
An alkaloid with anthelmintic and anticancer activities -
GC46854
Anastrozole-d12
ZD1033-d12
An internal standard for the quantification of anastrozole -
GC49419
Aniline-d5
苯胺-2,3,4,5,6-d5
An internal standard for the quantification of aniline -
GC63618
Antrafenine
安曲非宁; Stakane
Antrafenine (Stakane) 是一种非麻醉性缓解疼痛试剂,在药理学和毒理学研究中表现出长时间的作用和良好的耐受性。 -
GC49799
Apatinib-d8
An internal standard for the quantification of apatinib
-
GC40674
APHA Compound 8
组蛋白去乙酰化酶
A class I and II HDAC inhibitor -
GC60592
APS6-45
APS6-45(Compound 10) is an orally active tumor-calibrated inhibitor (TCI) that inhibits RAS/MAPK signaling and exhibits antitumor activity.
-
GC42854
ARN14988
A potent inhibitor of acid ceramidase
-
GC91634
ARN25062
ARN25062 is a derivative of ARN22089, an inhibitor of the protein-protein interaction between Cdc42 and p21-activated kinase (PAK).
-
GC49103
Aromadendrene
(+)-香橙烯
A sesquiterpene with diverse biological activities -
GC46089
Asperfuran
(-)-Asperfuran
A fungal metabolite -
GC42861
Aspochalasin M
A fungal metabolite
-
GC46090
Aspulvinone O
A fungal metabolite
-
GC46091
Aszonapyrone A
A meroditerpene fungal metabolite with diverse biological activities
-
GC42870
Atrazine Mercapturate
阿特拉津代谢物
A metabolite of atrazine -
GC48511
Avrainvillamide
(+)-Avrainvillamide; CJ-17,665
A fungal metabolite -
GC63301
AWL-II-38.3
AWL-II-38.3 is a potent Ephrin type-A receptor 3 (EphA3) kinase inhibitor.
-
GC63551
AZD-CO-Ph-PEG4-Ph-CO-AZD
AZD-CO-PH-四聚乙二醇-PH-CO-AZD
AZD-CO-Ph-PEG4-Ph-CO-AZD 是一种可用于抗体-siRNA 结合合成的 bis-β-lactam 连接子。 -
GC45938
Bacopaside X
假马齿苋皂苷VII,Bacopaside VII
A triterpenoid saponin -
GC91050
Bactobolin A (hydrochloride)
BN-183B
一种具有抗生素和抗癌活性的微生物代谢产物。
-
GC50603
BAY 293 Negative Control
Negative control for BAY 293
-
GC74427
Belrestotug
贝瑞苏塔单抗; EOS-448; EOS884448; GSK4428859A
Belrestotug (EOS-448)是一种抗tigit (VSIG9, VSTM3)人免疫球蛋白G1 kappa (hIgG1 kappa)的拮抗抗体。 -
GC49403
Benzarone
苯扎隆,Fragivix
An active metabolite of benzbromarone -
GC41532
Benzisoxazole Hsp90 Inhibitor
BHI
Hsp90 chaperone inhibitor -
GC63665
Benzylacyclouridine
BAU; 5-Benzylacyclouridine
Benzylacyclouridine (BAU) 是一种有效且特异性的尿苷磷酸化酶抑制剂,尿苷磷酸化酶是尿苷分解代谢中的第一种酶。Benzylacyclouridine 可以调节 5-氟尿嘧啶 (5-FU) 及其衍生物的细胞毒副作用。 -
GC42925
Berteroin
5-Methylthiopentyl isothiocyanate
A natural sulforaphane analog -
GC48458
Betulinic glycine amide
A derivative of betulinic acid
-
GC60075
BI99179
BI99179 是一种有效的选择性 I 型脂肪酸合成酶 (FAS) 抑制剂,IC50 为 79 nM。在大鼠中口服 BI 99179 表现出显着的外周和中央暴露。
-
GC46925
Bicalutamide-d4
比卡鲁胺 d4
An internal standard for the quantification of bicalutamide -
GC91030
Biotin-Cholesterol
Biotin-Provitamin D
一种生物素化的胆固醇
-
GC52392
Biotin-H10 (trifluoroacetate salt)
Biotin-GGGSGMKMQVRIYLV-OH, Biotin-Gly-Gly-Gly-Ser-Gly-Met-Lys-Met-Gln-Val-Arg-Ile-Tyr-Leu-Val-OH
A biotinylated form of H10 -
GC48713
Biotinyl hexylamine
A synthetic intermediate
-
GC42941
Bis(methylthio)gliotoxin
二(甲硫基)焦霉毒素,Bisdethiobis(methylthio)gliotoxin; FR 49175; Dimethylgliotoxin
A fungal metabolite with diverse biological activities -
GC48463
Bisubstrate Inhibitor 78
An inhibitor of NNMT
-
GC74481
Bivatuzumab
比伐珠单抗; BIWA 4; Anti-CD44 Recombinant Antibody
Bivatuzumab(抗CD44重组抗体;BIWA 4)是一种针对CD44v6的人源化单克隆抗体。