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Cancer Biology(癌症生物学)

  1. Cat.No. 产品名称 Information
  2. GC19775 M2N12 M2N12 是一种有效且高度选择性的细胞分裂周期 25C 蛋白磷酸酶 (Cdc25C) 抑制剂,IC50 值为 0.09 μM。 M2N12 对 Cdc25A 和 Cdc25B 也有很好的活性,IC50 值分别为 0.53 μM 和 1.39 μM。 M2N12具有抗肿瘤活性,可用于癌症研究。
  3. GC41185 MAGL Inhibitor Compound 23 An inhibitor of MAGL
  4. GC46031 Malabaricone B

    NSC 287967, NSC 630196

    A diarylnonanoid with diverse biological activities
  5. GC44118 Malvidin (chloride)

    氯化锦葵色素,Syringidin

    A plant pigment with antioxidant properties
  6. GC44126 Manzamine A

    Keramamine A

    A β-carboline alkaloid
  7. GP10140 MAP kinase fragment [Multiple species]

    H2N-Lys-Tyr-Ile-His-Ser-Ala-Asn-Val-Leu-OH

    Lys-Tyr-Ile-His-Ser-Ala-Asn-Val-Leu

  8. GC74475 Mapatumumab

    马帕木单抗; HGS-ETR1; Anti-Human TNFRSF10A Recombinant Antibody

    Mapatumumab (HGS-ETR1)是一种完全人IgG1激动性单克隆抗体,靶向肿瘤坏死因子相关凋亡诱导配体受体1 (TRAIL-R1)。
  9. GC47606 Mca-PLGL-Dap(Dnp)-AR-NH2 (trifluoroacetate salt)

    Mca-Pro-Leu-Gly-Leu-Dap(Dnp)-Ala-Arg-NH2, 7-Methoxycoumarin-4-acetyl-P-L-G-L-β-(2,4-dinitrophenylamino)A-R amide

    A neuropeptide with diverse biological activities
  10. GC91980 MCI-INI-3 MCI-INI-3是醛脱氢酶1A3(ALDH1A3;Ki=0.55μM)的抑制剂。
  11. GC44168 Metanephrine

    间甲肾上腺素

    An inactive metabolite of epinephrine

  12. GC49423 Metanephrine-d3 (hydrochloride)

    DL-Metanephrine-d3

    An internal standard for the quantification of metanephrine
  13. GC49879 Metformin hydroxy analog 2

    二甲双胍杂质3

    An oxidation product of metformin
  14. GC48805 Methapyrilene (hydrochloride)

    盐酸美沙吡林,Thenylpyramine hydrochloride

    An H1 receptor antagonist and non-genotoxic carcinogen
  15. GC47649 Methotrexate (hydrate)

    二水合氨甲嘌呤

    A folic acid and aminopterin derivative
  16. GC47650 Methotrexate-d3

    甲氨蝶呤 d3

    An internal standard for the quantification of methotrexate
  17. GC49241 Methyl Diethyldithiocarbamate

    S-甲基N,N二乙基二硫代氨基甲酸

    An active metabolite of disulfiram
  18. GC47674 Mifepristone-d3

    RU486-d3; RU 38486-d3

    A neuropeptide with diverse biological activities
  19. GC74577 Minretumomab

    明瑞莫单抗; CC-49

    Minretumomab(CC-49)是一种针对TAG-72(肿瘤相关糖蛋白72)的小鼠单克隆抗体。
  20. GC50686 Miro1 Reducer Promotes proteasomal degradation of Miro1 (mitochondrial Rho GTPase 1)
  21. GC16331 Misonidazole

    米索硝唑,NSC 261037,Ro 7-0582,SR 1354

    A nitroimidazole that targets hypoxic cells
  22. GC12876 ML-097

    CID-2160985

    A pan activator of Ras-related GTPases
  23. GC13315 ML-098

    CID-7345532

    A selective Rab7 activator
  24. GC16765 ML-099

    CID-888706

    A pan activator of Ras-related GTPases
  25. GC18616 MMP-8 Inhibitor I

    Matrix Metalloproteinase-8 Inhibitor I

    A selective inhibitor of MMP-8
  26. GC74487 Modotuximab

    扎妥昔单抗; DS 1024; Sym 004

    Modotuximab (Anti-Human EGFR Recombinant Antibody)是一种靶向人EGFR蛋白的igg1 - κ型嵌合抗体。
  27. GC61843 Mofezolac

    莫苯唑酸

    A COX-1 inhibitor
  28. GC46176 Multiflorenol A triterpene
  29. GC41325 Mycophenolic Acid β-D-Glucuronide

    霉酸Β-D-葡萄糖醛酸,MPAG,Mycophenolic Acid Glucosiduronate

    A metabolite of mycophenolic acid
  30. GP10114 Myelopeptide-2 (MP-2)

    H2N-Leu-Val-Val-Tyr-Pro-Trp-OH

    用于恢复人T淋巴细胞的肽

  31. GC47809 Nε-(1-Carboxymethyl)-L-lysine-d3

    CML-d3

    A neuropeptide with diverse biological activities
  32. GC63657 N,N,N′,N′-Tetracyclohexyl-3-oxapentanediamide

    Calcium ionophore II

    A calcium ionophore
  33. GC49256 N-acetyl Lenalidomide

    N-乙酰来那度胺

    A metabolite of lenalidomide
  34. GC18506 N-Arachidonoyl Dopamine

    NADA

    An arachidonoyl amino acid and CB1 receptor agonist
  35. GC47748 N-Arachidonoyl Dopamine-d8

    NADAd8

    An internal standard for the quantification of N-arachidonoyl dopamine
  36. GC48335 N-glycolyl-Ganglioside GM3 Mixture (ammonium salt)

    GM3-Neugc, NeuGc-GM3, NGcGM3, N-glycolyl-GM3, N-glycolyl-Monosialoganglioside GM3, N-Glycolylneuraminyllactosylceramide

    A mixture of N-glycolyl-ganglioside GM3
  37. GC49350 N-Nitroso Sarcosine

    N-亚硝基肌氨酸

    A carcinogen
  38. GC49354 N-Nitroso Sarcosine-d3

    N-亚硝基肌氨酸-D3

    An internal standard for the quantification of nitroso sarcosine
  39. GC47786 N-Nitroso-N-methyl-4-Aminobutyric Acid

    氯沙坦基因毒杂质

    A tobacco-specific nitrosamine carcinogen
  40. GC49859 N-Nitroso-N-methylaniline

    N-甲基-N-亚硝基苯胺

    An N-nitrosamine
  41. GC49731 N-Nitrosodimethylamine-d6

    氘代N-亚硝基二甲胺D6

    An internal standard for the quantification of N-nitrosodimethylamine
  42. GC49814 N-Nitrosomethylisopropylamine

    N-甲基-N-亚硝基-2-丙胺

    An N-nitrosamine
  43. GC63625 N-Palmitoyl-L-glutamine N-Palmitoyl-L-glutamine是一种由棕榈酸与L-谷氨酰胺结合而成的生物活性脂酰胺,具有调节细胞功能和信号通路的潜力。
  44. GC52162 N1-Acetylputrescine

    N-乙酰基-1,4-丁二胺

    A metabolite of putrescine
  45. GC44285 N1-Acetylspermine (hydrochloride)

    N1-乙酰精胺三盐酸盐

    An acetyl derivative of spermine
  46. GC63633 N7-Methyl-guanosine-5’-triphosphate-5’-adenosine

    N7-甲基鸟苷-5'-三磷酸-5'-腺苷,m7GpppA

    N7-Methyl-guanosine-5’-triphosphate-5’-adenosine (m7GpppA) 是一种二核苷酸帽类似物,可用于体外 RNA 转录。
  47. GC48584 Naftopidil-d5

    KT-611-d5; BM-15275-d5

    An internal standard for the quantification of naftopidil
  48. GC40081 Nargenicin

    阿根诺卡菌素,Antibiotic 47444

    A macrolide antibiotic
  49. GC70621 NBD-Pen NBD-Pen是一种荧光探针。
  50. GC45926 Nelfinavir-d3 An internal standard for the quantification of nelfinavir
  51. GC18750 NEO2734

    EP31670

    NEO2734 (EP31670) 是一种口服有效的双重 p300/CBP 和 BET 溴结构域选择性抑制剂,对 p300/CBP 和 BET 溴结构域的 IC50 值均 <30 nM。 NEO2734 在 SPOP 突变型和野生型前列腺癌中具有活性。

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