Pamicogrel (KBT3022)

目录号: GC32640纯度: >99.00%同义词: 帕米格雷; KBT3022
A COX inhibitor and an antiplatelet agent

Pamicogrel (KBT3022)
Cas No.: 101001-34-7
规格价格库存数量操作
5mg¥495.00现货
1
10mg¥792.00现货
1
25mg¥1,575.00现货
1
50mg¥2,520.00现货
1
100mg¥4,005.00现货
1
10mM (in 1mL DMSO)¥489.00现货
1

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产品描述 Description

Pamicogrel is a COX inhibitor and an antiplatelet agent.1,2,3 It inhibits platelet aggregation induced by arachidonic acid or collagen in washed isolated rabbit platelets (IC50s = 1.5 and 0.43 ?M, respectively).2 Pamicogrel (1 mg/kg) reduces thrombus weight in a guinea pig model of arteriovenous shunt thrombosis.3

1.Light, P.Pamicogrel (Kanebo)IDrugs2(9)938-942(1999) 2.Yokota, K., Yamamoto, N., Morimoto, Y., et al.Effect of KBT-3022, a new diphenylthiazole derivative, on platelet functionsJ. Pharm. Pharmacol.47(9)768-774(1995) 3.Yokota, K., Yamashita, A., and Oda, M.Anti-thrombotic activity of KBT-3022 in experimental models of thrombosisJpn. J. Pharmacol.68(2)201-206(1995)

产品文档 Product Documents

Purity:>99.00%

化学性质Chemical Properties

CAS 号
101001-34-7
同义词
帕米格雷; KBT3022
SMILES
O=C(OCC)CN1C(C2=NC(C3=CC=C(OC)C=C3)=C(C4=CC=C(OC)C=C4)S2)=CC=C1
分子式
C25H24N2O4S
分子量
448.53 g/mol
溶解性
DMSO: 83.33 mg/mL (185.78 mM)
保存条件
Store at -20°C
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。
储备液的保存方式和期限:-80°C 储存时,请在 6 个月内使用,-20°C 储存时,请在 1 个月内使用。
为了提高溶解度,请将管子加热至 37°C,然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案:配备蓝冰进行发货。所有其他可用尺寸:配备 RT,或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol