GlpBio

Taltirelin acetate

目录号: GC37732纯度: >98.50%同义词: TA-0910 acetate
Taltirelin acetate (TA-0910 acetate) 是一种促甲状腺激素释放激素受体 (TRH-R) 超激动剂，IC50 值为 910 nM，刺激细胞溶质Ca2+ 浓度增加 (Ca2+ 释放) 的 EC50 值为 36 nM。
Taltirelin acetate
Cas No.: 1549593-23-8
规格价格库存数量操作
5mg¥675.00现货
1
10mg¥904.00现货
1
50mg¥2,880.00现货
1
100mg¥4,500.00现货
1
10mM (in 1mL DMSO)¥743.00现货
1
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文献被引

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产品描述 Description

Taltirelin acetate (TA-0910 acetate) is a superagonist at thyrotropin-releasing hormone receptor (TRH-R) with an IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ concentration (Ca2+ release)[1]. IC50: 910 nM (Thyrotropin-releasing hormone receptor)[1]

[1]. Thirunarayanan N, et al. Taltirelin is a superagonist at the human thyrotropin-releasing hormone receptor. Front Endocrinol (Lausanne). 2012 Oct 9;3:120.

产品文档 Product Documents

Purity:>98.50%

化学性质Chemical Properties

CAS 号
1549593-23-8
同义词
TA-0910 acetate
SMILES
O=C(N(CCC1)[C@@H]1C(N)=O)[C@@H](NC([C@@H](NC2=O)CC(N2C)=O)=O)CC3=CN=CN3.CC(O)=O
分子式
C19H27N7O7
分子量
465.46 g/mol
溶解性
DMSO: 125 mg/mL (268.55 mM)
保存条件
Store at -20°C
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
为了提高溶解度，请将管子加热至 37°C，然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案：配备蓝冰进行发货。所有其他可用尺寸：配备 RT，或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol