EHMT2-IN-1 is a potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2. Used in the research of blood disorder or cancer[1]. EHMTI PEP|<100 nM (IC50)|EHMT2 PEP|<100 nM (IC50)|EHMT2 ICW|<100 nM (IC50)
EHMT2-IN-1 (Compound 108) potent EHMT inhibitor, with IC50s of all <100 nM for EHMT1 peptide, EHMT2 peptide and cellular EHMT2[1].
[1]. John Emmerson Campbell, et al. Amine-substituted heterocyclic compounds as ehmt2 inhibitors and methods of use thereof. WO2018118842A1