CLP-3094

目录号: GC62209纯度: >99.00%同义词: 2-[2-(4-氯-苯氧基)-乙基硫基]-1H-苯并咪唑
CLP-3094, a potent inhibitor targeting the binding function 3 (BF3) site of androgen receptor (AR), inhibits AR transcriptional activity with IC50 of 4 μM, also is a selective, potent GPR142 antagonist.

CLP-3094
Cas No.: 312749-73-8
规格价格库存数量操作
5 mg¥1,170.00现货
1
10 mg¥2,070.00现货
1
10mM (in 1mL DMSO)¥1,287.00现货
1

文献被引

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产品描述 Description

CLP-3094, a potent inhibitor targeting the binding function 3 (BF3) site of androgen receptor (AR), inhibits AR transcriptional activity with IC50 of 4 μM, also is a selective, potent GPR142 antagonist.

[1] Munuganti RS, et al. J Med Chem. 2013 Feb 14;56(3):1136-48.

产品文档 Product Documents

Purity:>99.00%

化学性质Chemical Properties

CAS 号
312749-73-8
同义词
2-[2-(4-氯-苯氧基)-乙基硫基]-1H-苯并咪唑
分子式
C15H13ClN2OS
分子量
304.79 g/mol
溶解性
DMSO : 100 mg/mL (328.09 mM; Need ultrasonic)
保存条件
Store at -20°C
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。
储备液的保存方式和期限:-80°C 储存时,请在 6 个月内使用,-20°C 储存时,请在 1 个月内使用。
为了提高溶解度,请将管子加热至 37°C,然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案:配备蓝冰进行发货。所有其他可用尺寸:配备 RT,或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol