AN3199

目录号: GC31728纯度: >99.50%
AN3199是一种PDE4抑制剂,IC50为94.5nM。

AN3199
Cas No.: 1187187-10-5
规格价格库存数量操作
5mg¥675.00现货
1
10mg¥1,080.00现货
1
25mg¥2,160.00现货
1
50mg¥3,456.00现货
1
100mg¥5,184.00现货
1
10mM (in 1mL DMSO)¥743.00现货
1

文献被引

本产品暂无引用记录;以下为 GlpBio 产品在 Nature / Cell / Science 等顶刊的客户引用样例
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产品描述 Description

AN3199 is a PDE4 inhibitor with IC50 of 94.5 nM.IC50 value: 94.5 nM [1]Target: PDE4The detailed information please refer to Compound 11 in the reference.

[1]. Zhang YK, et al. Design and synthesis of boron-containing PDE4 inhibitors using soft-drug strategy for potential dermatologic anti-inflammatory application. Bioorg Med Chem Lett. 2010 Apr 1;20(7):2270-4. [2]. Akama Tsutomu, et al. Preparation of boron-containing small molecules as anti-inflammatory agents. From PCT Int. Appl. (2009), WO 2009111676 A2 20090911.

产品文档 Product Documents

Purity:>99.50%

化学性质Chemical Properties

CAS 号
1187187-10-5
SMILES
O=C(C1=CC=C(OC2=CC=C(B(O)OC3)C3=C2)N=C1)OCCCC
分子式
C17H18BNO5
分子量
327.14 g/mol
溶解性
DMSO : 100 mg/mL (305.68 mM)
保存条件
Store at -20°C
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。
储备液的保存方式和期限:-80°C 储存时,请在 6 个月内使用,-20°C 储存时,请在 1 个月内使用。
为了提高溶解度,请将管子加热至 37°C,然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案:配备蓝冰进行发货。所有其他可用尺寸:配备 RT,或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol