SRT 1460

目录号: GC65019纯度: >98.00%同义词: 3,4,5-三甲氧基-N-(2-(3-(哌嗪-1-基甲基)咪唑并[2,1-B]噻唑-6-基)苯基)苯甲酰胺
SRT-1460 is a potent and selective activator of Sirtuin 1 (SIRT1) with EC1.5 of 2.9 μM. SRT-1460 reduces cell viability and growth of pancreatic cancer cells and induces apoptosis.

SRT 1460
Cas No.: 925432-73-1
规格价格库存数量操作
1mg¥293.00现货
1
5mg¥672.00现货
1
10mg¥1,005.00现货
1
25mg¥1,502.00现货
1
50mg¥2,244.00现货
1
100mg¥3,367.00现货
1
10mM (in 1mL DMSO)¥750.00现货
1

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产品描述 Description

SRT-1460 is a potent and selective activator of Sirtuin 1 (SIRT1) with EC1.5 of 2.9 μM. SRT-1460 reduces cell viability and growth of pancreatic cancer cells and induces apoptosis.

[1] Jill C Milne, et al. Nature. 2007 Nov 29;450(7170):712-6. [2] Claudia C S Chini, et al. Clin Cancer Res. 2016 May 15;22(10):2496-507.

实验参考方法 Experimental Reference Method

SIRT1

2.9μM(EC1.5)

产品文档 Product Documents

Purity:>98.00%

化学性质Chemical Properties

CAS 号
925432-73-1
同义词
3,4,5-三甲氧基-N-(2-(3-(哌嗪-1-基甲基)咪唑并[2,1-B]噻唑-6-基)苯基)苯甲酰胺
分子式
C26H29N5O4S
分子量
507.6 g/mol
溶解性
DMSO : 10 mg/mL (19.70 mM; Need ultrasonic)
保存条件
Store at -20°C
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。
储备液的保存方式和期限:-80°C 储存时,请在 6 个月内使用,-20°C 储存时,请在 1 个月内使用。
为了提高溶解度,请将管子加热至 37°C,然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案:配备蓝冰进行发货。所有其他可用尺寸:配备 RT,或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol