关于 "Na+/K+ ATPase" 的结果8+ 个结果
筛选:Ras×
- K-Ras-IN-1CAS: 84783-01-7
K-Ras-IN-1 (MDK-3017) inhibits K-Ras by binding to K-Ras in a hydrophobic pocket that is occupied by Tyr-71 in the apo-Ras crystal structure.
Ras - PROTAC K-Ras Degrader-1CAS: 2378258-52-5
PROTAC K-Ras Degrader-1 是一种基于 PROTAC 技术的有效的 K-Ras 降解剂,在 SW1573 中对其降解率为 ≥70%。
Ras - 6H05 trifluoroacetate (K-Ras inhibitor)
6H05 is a selective, and allosteric inhibitor of oncogenic K-Ras(G12C).
Ras
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC33153 | K-Ras-IN-1 | 84783-01-7 | Ras | ||
K-Ras-IN-1 (MDK-3017) inhibits K-Ras by binding to K-Ras in a hydrophobic pocket that is occupied by Tyr-71 in the apo-Ras crystal structure. | |||||
| GC36399 | K-Ras G12C-IN-2 | 1629267-75-9 | Ras | ||
K-Ras G12C-IN-2 是一种不可逆的 K-Ras G12C 抑制剂。 | |||||
| GC36398 | K-Ras G12C-IN-1 | 1629265-17-3 | Ras | ||
K-Ras G12C-IN-1是突变型K-Ras G12C不可逆小分子抑制剂。 | |||||
| GC36400 | K-Ras G12C-IN-3 | 1629268-19-4 | Ras | ||
K-Ras G12C-IN-3是突变型K-Ras G12C不可逆小分子抑制剂。 | |||||
| GC12247 | K-Ras(G12C) inhibitor 12 | 1469337-95-8 | Other Apoptosis | ||
An allosteric inhibitor of oncogenic K-Ras(G12C) | |||||
| GC38942 | PROTAC K-Ras Degrader-1 | 2378258-52-5 | Ras | ||
PROTAC K-Ras Degrader-1 是一种基于 PROTAC 技术的有效的 K-Ras 降解剂,在 SW1573 中对其降解率为 ≥70%。 | |||||
| GC62622 | K-Ras G12C-IN-4 | 2376328-55-9 | Ras | ||
K-Ras G12C-IN-4,化合物 1,是 KRASG12C 的有效共价抑制剂。 | |||||
| GC34427 | 6H05 trifluoroacetate (K-Ras inhibitor) | - | Ras | ||
6H05 is a selective, and allosteric inhibitor of oncogenic K-Ras(G12C). | |||||
