关于 "Histone Acetyltransferases" 的结果6 个结果
- Benzenebutyric acid (4-Phenylbutyric acid)CAS: 1821-12-1
4-Phenylbutyric acid (4-PBA, Benzenebutyric acid) is a histone deacetylase (HDAC) inhibitor and a key epigenetic inducer of anti-HCV hepatic hepcidin. 4-Phenylbutyric acid inhibits LPS-induced inflammation through regulating endoplasmic-reticulum (ER) stress and autophagy in acute lung injury models.
- TubacinCAS: 537049-40-4
Tubacin (tubulin acetylation inducer)是一种选择性抑制组蛋白去乙酰化酶6 (HDAC6),诱导α-微管蛋白乙酰化的小分子,IC50为0.004µM。
- Panobinostat (LBH589)CAS: 404950-80-7
Panobinostat (LBH589)是一种强效,且具有口服活性和抗肿瘤活性的广谱组蛋白去乙酰化酶(HDAC)抑制剂,IC 50 值为5nM。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC17284 | Anacardic acid | 16611-84-0 | Epigenetic Reader Domain | ||
A histone acetyltransferase inhibitor | |||||
| GC30763 | Benzenebutyric acid (4-Phenylbutyric acid) | 1821-12-1 | Virus Protease | ||
4-Phenylbutyric acid (4-PBA, Benzenebutyric acid) is a histone deacetylase (HDAC) inhibitor and a key epigenetic inducer of anti-HCV hepatic hepcidin. 4-Phenylbutyric acid inhibits LPS-induced inflammation through regulating endoplasmic-reticulum (ER) stress and autophagy in acute lung injury models. | |||||
| GC17390 | Vorinostat (SAHA, MK0683) | 149647-78-9 | HIV | ||
An HDAC inhibitor | |||||
| GC16386 | Tubacin | 537049-40-4 | Virus Protease | ||
Tubacin (tubulin acetylation inducer)是一种选择性抑制组蛋白去乙酰化酶6 (HDAC6),诱导α-微管蛋白乙酰化的小分子,IC50为0.004µM。 | |||||
| GC12257 | Panobinostat (LBH589) | 404950-80-7 | HIV | ||
Panobinostat (LBH589)是一种强效,且具有口服活性和抗肿瘤活性的广谱组蛋白去乙酰化酶(HDAC)抑制剂,IC50值为5nM。 | |||||
| GC32066 | RRx-001 | 925206-65-1 | Parasite | ||
RRx-001 是一种源自航空航天的抗癌剂,具有产生活性氮物质 (RNS) 的化学作用,可导致表观遗传改变,例如癌细胞中的 DNA 甲基化和组蛋白乙酰化。 | |||||
