关于 "GABA Receptor" 的结果73+ 个结果
筛选:Membrane Transporter/Ion Channel×
- TPMPA (hydrate)
选择性 GABA\u003csub\u003eA\u003c/sub\u003e-ρ1 (ρ1 GABA\u003csub\u003eC\u003c/sub\u003e) 受体拮抗剂
- S-8510 phosphate (SB-737552 phosphate)CAS: 151466-23-8
S-8510 (phosphate) 是一种反向苯二氮卓 (BDZ) 受体激动剂,对 -GABA 和 +GABA 的 Kis 分别为 34.6 nM、36.2 nM。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC11284 | 6-(4-Methoxyphenyl)-3-pyridazinamine | 4776-87-8 | GABA Receptor | ||
A GABAA receptor antagonist | |||||
| GC16947 | CGP 52432 | 139667-74-6 | GABA Receptor | ||
A GABAB receptor antagonist | |||||
| GC11013 | U 93631 | 152273-12-6 | GABA Receptor | ||
A GABAA receptor ligand | |||||
| GC45044 | Thiomuscimol | 62020-54-6 | Neuroscience | ||
A GABAA receptor agonist | |||||
| GC34986 | (R)-Baclofen hydrochloride | 63701-55-3 | GABA Receptor | ||
A GABAB receptor agonist | |||||
| GC35669 | CGP 36742 | 123690-78-8 | GABA Receptor | ||
A GABAB receptor antagonist | |||||
| GC39126 | Thiocolchicoside | 602-41-5 | GABA Receptor | ||
A GABAA receptor antagonist | |||||
| GN10745 | (+)-Bicuculline | 485-49-4 | GABA Receptor | ||
(+)-荷包牡丹碱((+)-Bicuculline ))是一种竞争性GABAA受体拮抗剂,IC50为2μM。 | |||||
| GC10489 | CGP 54626 hydrochloride | 149184-21-4 | GABA Receptor | ||
A selective GABAB receptor antagonist | |||||
| GC11153 | CGP 35348 | 123690-79-9 | GABA Receptor | ||
A brain-accessible GABAB receptor antagonist | |||||
| GC48313 | γ-Lindane | 58-89-9 | Neuroscience | ||
An insecticide and GABAA receptor antagonist | |||||
| GC10772 | Flumazenil | 78755-81-4 | GABA Receptor | ||
A GABAA receptor antagonist and partial agonist | |||||
| GC10974 | AWD 131-138 | 188116-07-6 | GABA Receptor | ||
A partial agonist of the GABAA receptor | |||||
| GC11143 | NS 11394 | 951650-22-9 | GABA Receptor | ||
A subunit-selective positive allosteric modulator of the GABAA receptor | |||||
| GC31049 | RWJ-51204 | 205701-85-5 | GABA Receptor | ||
RWJ-51204是GABA(A)receptor的部分激动剂,Ki值为0.2-2nM。 | |||||
| GC69161 | Gidazepam | 129186-29-4 | GABA Receptor | ||
Gidazepam 是一种 GABA 受体通道 (GABA RCs) 激动剂。 | |||||
| GC12357 | Pentylenetetrazole | 54-95-5 | GABA Receptor | ||
Pentylenetetrazole是一种γ-氨基丁酸(GABA)A受体的非选择性拮抗剂。 | |||||
| GC14659 | Guvacine hydrochloride | 6027-91-4 | GABA Receptor | ||
An inhibitor of GABA uptake | |||||
| GC14477 | CI 966 hydrochloride | 110283-66-4 | GABA Receptor | ||
GABA transporter GAT-1 inhibitor | |||||
| GC60890 | Guvacine | 498-96-4 | GABA Receptor | ||
An inhibitor of GABA uptake | |||||
| GC16937 | Carbamoylcholine chloride | 51-83-2 | nAChR | ||
Cholinergic receptor agonist | |||||
| GC48191 | TPMPA (hydrate) | - | Behavioral Neuroscience | ||
选择性 GABA\u003csub\u003eA\u003c/sub\u003e-ρ1 (ρ1 GABA\u003csub\u003eC\u003c/sub\u003e) 受体拮抗剂 | |||||
| GC70546 | Fengabine | 80018-06-0 | GABA Receptor | ||
Fengabine是一种gaba能抗抑郁剂。 | |||||
| GC31121 | S-8510 phosphate (SB-737552 phosphate) | 151466-23-8 | GABA Receptor | ||
S-8510 (phosphate) 是一种反向苯二氮卓 (BDZ) 受体激动剂,对 -GABA 和 +GABA 的 Kis 分别为 34.6 nM、36.2 nM。 | |||||
