关于 "Nuclear Receptors" 的结果106+ 个结果

An antagonist of σ 1 receptors

5-HT1B/1D receptors agonist, potent and selective

Negative allosteric modulator of mGlu7 receptors; brain penetrant

Anisodamine (6-Hydroxyhyoscyamine) is a naturally occurring atropine derivative and exhibits anti-inflammatory activity. It also inhibits α1-adrenergic receptors and muscarinic acetylcholine receptors (mAChRs).

A neuropeptide and agonist of NPFF1 and NPFF2 receptors

A potent agonist of D 2 receptors

An allosteric agonist of M 1 receptors

Dual antagonist of TP and EP 4 receptors

A nonpeptide antagonist of vasopressin V 1 receptors

An inverse agonist of 5-HT 2C receptors

A partial agonist of GPR109A/HCA 2 receptors

A selective agonist for the EP 2 receptors

A β-adrenergic receptor antagonist

(-)-Norepinephrine (Arterenol, Levarterenol, L-Noradrenaline) is a natural neurotransmitter and hormone. It is an agonist of adrenergic receptors with Ki values of 330, 56, and 740 nM for α1, α2, and β1 adrenoceptors, respectively.

Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an agonist of the 5-HT1 and 5-HT4 receptors and as an antagonist of the 5-HT2 receptors

A positive allosteric modulator of adenosine A 3 receptors

A positive allosteric modulator of muscarinic M 5 receptors

Selective positive allosteric modulator of M4 receptors; active in vivo; antipsychotic

A positive allosteric modulator of adenosine A 1 receptors

An amide of oleic acid and agonist of CB 1 receptors

An agonist at AT 1 and AT 2 receptors

An agonist of S1P 1 and S1P 5 receptors

An agonist at AT 1 and AT 2 receptors

A neuropeptide agonist of NMU 1 and NMU 2 receptors