关于 "LPA Receptor" 的结果95+ 个结果
筛选:GPCR/G protein×
- 1-oleoyl-2-hydroxy-sn-glycero-3-phosphate (sodium salt)CAS: 325465-93-8
1-油酰基溶血磷脂酸（1-油酰基-sn-甘油-3-磷酸）钠作为一种有效的生物活性磷脂，是LPA受体激活剂[2]。
- Ki16198CAS: 355025-13-7
Ki16198 是一种有效且具有口服活性的 LPA 受体拮抗剂，即 Ki16425 的甲酯。 Ki16198 抑制 LPA1 和 LPA3 诱导的磷酸肌醇产生，Ki 值分别为 0.34 μM 和 0.93 μM。 Ki16198 对体内胰腺癌的肿瘤发生和转移有效。
- Batefenterol (GSK961081)CAS: 743461-65-6
A muscarinic receptor antagonist and β 2 -adrenergic receptor agonist
- AlloxazineCAS: 490-59-5
Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC14812 | GW 627368 | 439288-66-1 | Prostaglandin Receptor | ||
A potent EP4 receptor antagonist | |||||
| GC14173 | L-161,982 | 147776-06-5 | Prostaglandin Receptor | ||
A potent, selective EP4 receptor antagonist | |||||
| GC18112 | LP 44 | 824958-12-5 | 5-HT Receptor | ||
A selective 5-HT7 receptor agonist | |||||
| GC11784 | LCZ696 | 936623-90-4 | Other Apoptosis | ||
A dual angiotensin II receptor antagonist and neprilysin inhibitor | |||||
| GC16496 | Ticlopidine | 55142-85-3 | Adenosine Receptor | ||
A P2Y12 receptor antagonist with antiplatelet activity | |||||
| GC10051 | MDL 100907 | 139290-65-6 | 5-HT Receptor | ||
Selective antagonist of the serotonin receptor 5-HT2A | |||||
| GC15140 | 1-oleoyl-2-hydroxy-sn-glycero-3-phosphate (sodium salt) | 325465-93-8 | LPA Receptor | ||
1-油酰基溶血磷脂酸（1-油酰基-sn-甘油-3-磷酸）钠作为一种有效的生物活性磷脂，是LPA受体激活剂[2]。 | |||||
| GC15062 | Ki16198 | 355025-13-7 | LPA Receptor | ||
Ki16198 是一种有效且具有口服活性的 LPA 受体拮抗剂，即 Ki16425 的甲酯。 Ki16198 抑制 LPA1 和 LPA3 诱导的磷酸肌醇产生，Ki 值分别为 0.34 μM 和 0.93 μM。 Ki16198 对体内胰腺癌的肿瘤发生和转移有效。 | |||||
| GC10147 | AM630 | 164178-33-0 | Cannabinoid Receptor | ||
AM630是一种强效且选择性的CB2受体反向激动剂。 | |||||
| GC10310 | SB 206553 hydrochloride | 1197334-04-5 | 5-HT Receptor | ||
A 5-HT2C and 5-HT2B receptor antagonist | |||||
| GC31690 | Batefenterol (GSK961081) | 743461-65-6 | mAChR | ||
A muscarinic receptor antagonist and β2-adrenergic receptor agonist | |||||
| GC16470 | Methysergide maleate | 129-49-7 | 5-HT Receptor | ||
A 5-HT1 receptor agonist and 5-HT2 receptor antagonist | |||||
| GC25051 | Alloxazine | 490-59-5 | Adenosine Receptor | ||
Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor. | |||||
| GC17089 | MRS 2690 | 15039-58-4 | P2Y Receptor | ||
P2Y14 receptor agonist | |||||
| GC15635 | PSB 1114 | 1657025-60-9 | P2Y Receptor | ||
P2Y2 receptor agonist | |||||
| GC16422 | Somatostatin 1-28 | 74315-46-1 | Somatostatin Receptor | ||
Somatostatin receptor agonist | |||||
| GC10271 | [Ac-Tyr1,D-Phe2]GRF 1-29, amide (human) | 93965-89-0 | VIP Receptors | ||
VIP receptor antagonist | |||||
| GC15163 | [D-Phe12]-Bombesin | 108437-87-2 | Bombesin Receptors | ||
Bombesin receptor antagonist | |||||
| GC14119 | BIM 23052 | 133073-82-2 | Somatostatin Receptor | ||
sst5 receptor agonist | |||||
| GC10777 | Cortistatin-8 | 485803-62-1 | Ghrelin Receptors | ||
ghrelin receptor antagonist | |||||
| GC17156 | [D-Phe12,Leu14]-Bombesin | 108437-88-3 | Bombesin Receptors | ||
Bombesin receptor antagonist | |||||
| GC14959 | 2-[1-(4-Piperonyl)piperazinyl]benzothiazole | 155106-73-3 | 5-HT Receptor | ||
5-HT4 receptor | |||||
| GC11188 | GR 135531 | 190277-13-5 | Melatonin Receptors | ||
MT3 receptor agonist | |||||