关于 "Bromodomain" 的结果26+ 个结果
筛选:Bromodomain×
- BET bromodomain inhibitorCAS: 1380087-89-7
BET 溴结构域抑制剂是从专利 WO/2015/153871A2 化合物实施例 11 中提取的一种有效的 BET 抑制剂。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC16531 | Bromodomain Inhibitor, (+)-JQ1 | 1268524-70-4 | Ligand for Target Protein for PROTAC | ||
A selective inhibitor of BET bromodomains | |||||
| GC16299 | BET bromodomain inhibitor | 1380087-89-7 | Epigenetic Reader Domain | ||
BET 溴结构域抑制剂是从专利 WO/2015/153871A2 化合物实施例 11 中提取的一种有效的 BET 抑制剂。 | |||||
| GC10174 | SGC-CBP30 | 1613695-14-9 | Histone Acetyltransferases | ||
A potent inhibitor of CREBBP/EP300 bromodomains | |||||
| GC14199 | RVX-208 | 1044870-39-4 | HIV | ||
A selective BET bromodomain antagonist | |||||
| GC14699 | CPI-203 | 1446144-04-2 | Other Apoptosis | ||
A bioavailable inhibitor of BET bromodomains | |||||
| GC17482 | OF-1 | 919973-83-4 | Epigenetic Reader Domain | ||
A bromodomain probe for BRPF proteins | |||||
| GC15175 | BAZ2-ICR | 1665195-94-7 | Epigenetic Reader Domain | ||
A BAZ2A/B bromodomain inhibitor | |||||
| GC12440 | GSK 5959 | 901245-65-6 | Epigenetic Reader Domain | ||
An inhibitor of the BRPF1 bromodomain | |||||
| GC10727 | Ischemin sodium salt | - | Bromodomain | ||
CBP bromodomain inhibitor | |||||
| GC15789 | GSK2801 | 1619994-68-1 | Epigenetic Reader Domain | ||
A probe for BAZ2A/B bromodomains | |||||
| GC12588 | I-BRD9 | 1714146-59-4 | Epigenetic Reader Domain | ||
A BRD9 bromodomain inhibitor | |||||
| GC16817 | BI-9564 | 1883429-22-8 | Epigenetic Reader Domain | ||
A selective BRD9/7 bromodomain inhibitor | |||||
| GC16726 | BI-7273 | 1883429-21-7 | Epigenetic Reader Domain | ||
A potent BRD9 bromodomain inhibitor | |||||
| GC15152 | PF-CBP1 | 1962928-21-7 | Bromodomain | ||
An inhibitor of the CBP and p300 bromodomains | |||||
| GC10382 | CPI-637 | 1884712-47-3 | Histone Acetyltransferases | ||
An inhibitor of CBP/EP300 bromodomains | |||||
| GC13025 | GSK6853 | 1910124-24-1 | Epigenetic Reader Domain | ||
A selective chemical probe for the bromodomain of BRPF1 | |||||
| GC16763 | NI-57 | 1883548-89-7 | Epigenetic Reader Domain | ||
A BRPF bromodomain inhibitor | |||||
| GC14168 | UMB-32 | 1635437-39-6 | Bromodomain | ||
An inhibitor of BRD4, TAF1, and TAF1L bromodomains | |||||
| GC14361 | PFI 3 | 1819363-80-8 | Epigenetic Reader Domain | ||
Probe for bromodomains of SMARCA2/4 and PB1(bromodomain 5) | |||||
| GC15375 | PFI-1 (PF-6405761) | 1403764-72-6 | Autophagy | ||
A BET bromodomain inhibitor | |||||
| GC10402 | Bromosporine | 1619994-69-2 | Epigenetic Reader Domain | ||
A non-specific bromodomain inhibitor | |||||
| GC16611 | GW841819X | - | Bromodomain | ||
BET bromodomain inhibitor | |||||
| GC13822 | (-)-JQ1 | 1268524-71-5 | Epigenetic Reader Domain | ||
A selective inhibitor of BET bromodomains | |||||
| GC60182 | GSK046 | 2474876-09-8 | Bromodomain | ||
A BD2 bromodomain inhibitor | |||||
