关于 "Topoisomerase" 的结果7 个结果
筛选:Autophagy×
- Etoposide phosphateCAS: 117091-64-2
Etoposidephosphate(BMY-40481)是一种有效的抗癌(anti-cancer)化疗试剂和一种选择性拓扑异构酶II(topoisomeraseII)抑制剂,可以防止DNA链的重新连接。Etoposidephosphate是依托泊苷的磷酸酯前药,被认为与Etoposide活性相当。Etoposidephosphate诱导细胞周期阻滞、凋亡(apoptosis)和自噬(autophagy)。
Autophagy
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC15617 | Etoposide | 33419-42-0 | Other Apoptosis | ||
Etoposide(VP-16)是一种非特异性拓扑异构酶II(Topoisomerase II)抑制剂,IC50值为59.2 μM。 | |||||
| GC12326 | Amsacrine | 51264-14-3 | Autophagy | ||
A topoisomerase II poison | |||||
| GC11747 | Amsacrine hydrochloride | 54301-15-4 | Autophagy | ||
A topoisomerase II poison | |||||
| GC11048 | Irinotecan HCl Trihydrate | 136572-09-3 | Autophagy | ||
A potent inhibitor of DNA topoisomerase I | |||||
| GN10449 | SN-38 (NK012) | 86639-52-3 | Autophagy | ||
A potent inhibitor of DNA topoisomerase I | |||||
| GC36329 | Irinotecan hydrochloride | 100286-90-6 | Autophagy | ||
A potent inhibitor of DNA topoisomerase I | |||||
| GC60826 | Etoposide phosphate | 117091-64-2 | Autophagy | ||
Etoposidephosphate(BMY-40481)是一种有效的抗癌(anti-cancer)化疗试剂和一种选择性拓扑异构酶II(topoisomeraseII)抑制剂,可以防止DNA链的重新连接。Etoposidephosphate是依托泊苷的磷酸酯前药,被认为与Etoposide活性相当。Etoposidephosphate诱导细胞周期阻滞、凋亡(apoptosis)和自噬(autophagy)。 | |||||
