关于 "Histone Acetyltransferases" 的结果12 个结果
筛选:Autophagy×
- Panobinostat (LBH589)CAS: 404950-80-7
Panobinostat (LBH589)是一种强效,且具有口服活性和抗肿瘤活性的广谱组蛋白去乙酰化酶(HDAC)抑制剂,IC 50 值为5nM。
- Entinostat (MS-275,SNDX-275)CAS: 209783-80-2
Entinostat (MS-275,SNDX-275)是一种强效的、可口服的组蛋白去乙酰化酶(HDACs)抑制剂,对HDAC1和HDAC3的IC₅₀分别为0.368μM和0.501μM,但对HDAC8的抑制作用相对较弱。
Autophagy
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC12171 | BIX 01294 | 935693-62-2 | Autophagy | ||
An inhibitor of G9a histone methyltransferase | |||||
| GC15610 | UNC0638 | 1255580-76-7 | Autophagy | ||
A G9a and GLP histone methyltransferase inhibitor | |||||
| GC15857 | Sodium butyrate | 156-54-7 | Autophagy | ||
A short-chain fatty acid and HDAC inhibitor | |||||
| GC15002 | Sodium Phenylbutyrate | 1716-12-7 | Autophagy | ||
Sodium Phenylbutyrate是一种组蛋白去乙酰化酶(HDAC)抑制剂。 | |||||
| GC15315 | Scriptaid | 287383-59-9 | Autophagy | ||
HDAC inhibitor | |||||
| GC10322 | Tubastatin A HCl | 1310693-92-5 | Autophagy | ||
A potent HDAC6 inhibitor | |||||
| GC17390 | Vorinostat (SAHA, MK0683) | 149647-78-9 | HIV | ||
An HDAC inhibitor | |||||
| GC12257 | Panobinostat (LBH589) | 404950-80-7 | HIV | ||
Panobinostat (LBH589)是一种强效,且具有口服活性和抗肿瘤活性的广谱组蛋白去乙酰化酶(HDAC)抑制剂,IC50值为5nM。 | |||||
| GC14998 | Rocilinostat (ACY-1215) | 1316214-52-4 | Other Apoptosis | ||
A selective inhibitor of HDAC6 | |||||
| GC11625 | Entinostat (MS-275,SNDX-275) | 209783-80-2 | Autophagy | ||
Entinostat (MS-275,SNDX-275)是一种强效的、可口服的组蛋白去乙酰化酶(HDACs)抑制剂,对HDAC1和HDAC3的IC₅₀分别为0.368μM和0.501μM,但对HDAC8的抑制作用相对较弱。 | |||||
| GC13055 | Mocetinostat (MGCD0103, MG0103) | 726169-73-9 | Autophagy | ||
An orally available HDAC inhibitor | |||||
| GC14590 | AR-42 (OSU-HDAC42) | 935881-37-1 | Other Apoptosis | ||
HDAC inhibitor,novel and potent | |||||
