关于 "ALK" 的结果7+ 个结果
筛选:Apoptosis×
- (E)-2-Hexadecenal AlkyneCAS: 1778692-99-1
A click chemistry probe for a sphingolipid degradation product
- SIAIS164018 hydrochloride
SIAIS164018 hydrochloride是一种基于protac的ALK和EGFR降解剂,ALK和ALK G1202R的IC50值分别为2.5 nM和6.6 nM。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC73642 | ALK-IN-26 | 2447607-85-2 | ALK | ||
ALK-IN-26是ALK抑制剂,对ALK酪氨酸激酶的IC50值为7.0 μM。 | |||||
| GC41701 | (E)-2-Hexadecenal Alkyne | 1778692-99-1 | Cytoskeleton & Motor Proteins | ||
A click chemistry probe for a sphingolipid degradation product | |||||
| GC35288 | Alkannin | 517-88-4 | Other Apoptosis | ||
A naphthoquinone with diverse biological activities | |||||
| GC64013 | ZX-29 | 2254805-62-2 | Autophagy | ||
ZX-29 is a potent and selective ALK inhibitor with an IC50s of 2.1, 1.3 and 3.9 nM for ALK, ALK L1196M and ALK G1202R mutations, respectively. | |||||
| GC16694 | TAE684 (NVP-TAE684) | 761439-42-3 | Other Apoptosis | ||
A selective ALK inhibitor | |||||
| GC73129 | SIAIS164018 hydrochloride | - | ALK | ||
SIAIS164018 hydrochloride是一种基于protac的ALK和EGFR降解剂,ALK和ALK G1202R的IC50值分别为2.5 nM和6.6 nM。 | |||||
| GC91040 | AP-1 | - | Ubiquitination/ Proteasome | ||
一种促进ALK降解的PROTAC | |||||
