关于 "ALK" 的结果20+ 个结果
- ALK inhibitor 1CAS: 761436-81-1
ALK inhibitor 1 (compound 17) is a potent pyrimidin ALK inhibitor which can inhibit testis-specific serine/threonine kinase (TSSK2; IC50=31 nM) and focal adhesion kinase (FAK; IC50=2 nM).
- ALK kinase inhibitor-1CAS: 1462949-64-9
ALK kinase inhibitor-1 是一种间变性淋巴瘤激酶 ALK 抑制剂,详细信息请参考专利文献 US20130261106A1 中的化合物 I-202。
- EML4-ALK kinase inhibitor 1CAS: 1373409-08-5
EML4-ALK kinase inhibitor 1 是有效的、具有口服活性的类棘皮细胞微管相关蛋白4-间变性淋巴瘤激酶 (EML4-ALK) 的抑制剂,其 IC50 值为 1 nM。
- WRVYEKC(dnp)ALK tetraTFA
WRVYEKC(dnp)ALK tetraTFA含有色氨酸,可以通过氨基肽酶活性从二硝基酚DNP猝灭剂中释放出来。
- Kratom Alkaloids Mixture
A mixture containing alkaloids found in M. speciosa (Kratom) in a solution of 0.1 N ammonia in methanol intended for HPLC or LC-MS applications
- Thalidomide 4'-oxyacetamide-alkylC1-PEG3-alkylC3-amineCAS: 2564466-93-7
Functionalized cereblon ligand for PROTAC® research and development; incorporates an E3 ligase ligand plus an alkylC1-PEG3-alkylC3 linker with terminal amine ready for conjugation to a target protein ligand
- Alkyne tyramideCAS: 1694495-59-4
Alkyne tyramide是一种可点击的抗坏血酸过氧化物酶2(APEX2)探针,具有水溶性和细胞壁渗透性,可显著提高完整酵母细胞中的APEX标记效率,还有助于识别APEX标记位点,从而可以明确分配线粒体蛋白的膜拓扑结构。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC35287 | ALK inhibitor 1 | 761436-81-1 | ALK | ||
ALK inhibitor 1 (compound 17) is a potent pyrimidin ALK inhibitor which can inhibit testis-specific serine/threonine kinase (TSSK2; IC50=31 nM) and focal adhesion kinase (FAK; IC50=2 nM). | |||||
| GC17376 | ALK inhibitor 2 | 761438-38-4 | ALK | ||
An inhibitor of TSSK2 | |||||
| GC35290 | ALK-IN-6 | 2055821-33-3 | ALK | ||
ALK-IN-6 (compound 11) 是口服有效的,间变性淋巴瘤激酶 (ALK) 的抑制剂,其对野生型 ALK、ALK F1196M 和ALK F1174L 的 IC50 值分别为 71 nM、18.72 nM 和36.81 nM。 | |||||
| GP22702 | ALK/P80 Human | - | Other | ||
ALK/P80 Protein Human Recombinant | |||||
| GC35289 | ALK-IN-5 | 2351929-66-1 | ALK | ||
ALK-IN-5 是一种高效选择性的,可渗透大脑屏障的 (ALK) 激酶抑制剂,IC50 值为 2.9 nM。 | |||||
| GC73642 | ALK-IN-26 | 2447607-85-2 | ALK | ||
ALK-IN-26是ALK抑制剂,对ALK酪氨酸激酶的IC50值为7.0 μM。 | |||||
| GC73883 | ALK-IN-28 | 1108743-80-1 | ALK | ||
ALK-IN-28(化合物22)是间变性淋巴瘤激酶(ALK)的抑制剂。 | |||||
| GC63387 | ALK kinase inhibitor-1 | 1462949-64-9 | ALK | ||
ALK kinase inhibitor-1 是一种间变性淋巴瘤激酶 ALK 抑制剂,详细信息请参考专利文献 US20130261106A1 中的化合物 I-202。 | |||||
| GC35979 | EML4-ALK kinase inhibitor 1 | 1373409-08-5 | - | ||
EML4-ALK kinase inhibitor 1 是有效的、具有口服活性的类棘皮细胞微管相关蛋白4-间变性淋巴瘤激酶 (EML4-ALK) 的抑制剂,其 IC50 值为 1 nM。 | |||||
| GC72228 | WRVYEKC(dnp)ALK tetraTFA | - | Enzyme Substrates | ||
WRVYEKC(dnp)ALK tetraTFA含有色氨酸,可以通过氨基肽酶活性从二硝基酚DNP猝灭剂中释放出来。 | |||||
| GB59089 | Lignin alkalie | 8068-05-1 | - | ||
| GC52319 | Kratom Alkaloids Mixture | - | Analytical Standards | ||
A mixture containing alkaloids found in M. speciosa (Kratom) in a solution of 0.1 N ammonia in methanol intended for HPLC or LC-MS applications | |||||
| GC19584 | Alkaline Phosphatase | 9001-78-9 | Peptides | ||
10-50units/mg protein(37℃,pH 9.8) | |||||
| GP21429 | Alkaline Phosphatase Bovine | - | Phosphatase | ||
Alkaline Phosphatase Bovine Intestinal | |||||
| GC20061 | ClAP (Alkaline Phosphatase, Calf intestinal) | 9001-78-9 | - | ||
4000u/mg protein,小牛肠,硫酸铵悬液 | |||||
| GC27476 | Aluminum oxide, 99%, alkaline 100-200mesh | 1344-28-1 | - | ||
| GC20227 | Alkaline proteinase(BR,200U/mg) | 9014-01-1 | - | ||
| GC50709 | Thalidomide 4'-oxyacetamide-alkylC1-PEG3-alkylC3-amine | 2564466-93-7 | PROTAC | ||
Functionalized cereblon ligand for PROTAC® research and development; incorporates an E3 ligase ligand plus an alkylC1-PEG3-alkylC3 linker with terminal amine ready for conjugation to a target protein ligand | |||||
| GC60573 | Alkyne tyramide | 1694495-59-4 | Isotope-Labeled Compounds | ||
Alkyne tyramide是一种可点击的抗坏血酸过氧化物酶2(APEX2)探针,具有水溶性和细胞壁渗透性,可显著提高完整酵母细胞中的APEX标记效率,还有助于识别APEX标记位点,从而可以明确分配线粒体蛋白的膜拓扑结构。 | |||||
| GC91056 | MTDB-Alkyne | 2923694-73-7 | COVID-19 | ||
一个可点击的RNA伪结合物绑定剂 | |||||
