关于 "Nuclear Receptors" 的结果14+ 个结果
筛选:5-HT Receptor×
- 5-HT2A receptor agonist-3CAS: 1391499-52-7
5-HT2A receptor agonist-3Ki=2.5nM、对5-HT2A的选择性是结构相似的5-HT2C受体的124倍。
5-HT Receptor - Donitriptan hydrochlorideCAS: 170911-68-9
5-HT1B/1D receptors agonist, potent and selective
5-HT Receptor - Cinitapride Hydrogen TartrateCAS: 1207859-16-2
Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an agonist of the 5-HT1 and 5-HT4 receptors and as an antagonist of the 5-HT2 receptors
5-HT Receptor - Frovatriptan succinate hydrateCAS: 158930-17-7
An agonist of 5-HT 1B and 5-HT 1D receptors
5-HT Receptor - SB 200646 hydrochlorideCAS: 143797-62-0
A dual antagonist of 5-HT 2C and 5-HT 2B receptors
5-HT Receptor
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC71279 | 5-HT2A receptor agonist-3 | 1391499-52-7 | 5-HT Receptor | ||
5-HT2A receptor agonist-3Ki=2.5nM、对5-HT2A的选择性是结构相似的5-HT2C受体的124倍。 | |||||
| GC16891 | Quetiapine Fumarate | 111974-72-2 | 5-HT Receptor | ||
An antagonist of diverse neurological receptors | |||||
| GC13265 | Donitriptan hydrochloride | 170911-68-9 | 5-HT Receptor | ||
5-HT1B/1D receptors agonist, potent and selective | |||||
| GC14491 | B-HT 920 | 36085-73-1 | Dopamine Receptor | ||
A potent agonist of D2 receptors | |||||
| GC10535 | S 32212 hydrochloride | 847871-78-7 | 5-HT Receptor | ||
An inverse agonist of 5-HT2C receptors | |||||
| GC25253 | Cinitapride Hydrogen Tartrate | 1207859-16-2 | 5-HT Receptor | ||
Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an agonist of the 5-HT1 and 5-HT4 receptors and as an antagonist of the 5-HT2 receptors | |||||
| GC13133 | Ipsapirone | 95847-70-4 | 5-HT Receptor | ||
A partial agonist of serotonin 5-HT1A receptors | |||||
| GC17053 | Eletriptan HBr | 177834-92-3 | 5-HT Receptor | ||
An agonist of 5-HT1B and 5-HT1D receptors | |||||
| GC17808 | Zolmitriptan | 139264-17-8 | 5-HT Receptor | ||
An agonist of 5-HT1B and 5-HT1D receptors | |||||
| GC15153 | Almotriptan Malate | 181183-52-8 | 5-HT Receptor | ||
An agonist of 5-HT1B and 5-HT1D receptors | |||||
| GC14558 | Dihydroergotamine mesylate | 6190-39-2 | 5-HT Receptor | ||
An agonist of 5-HT1B and 5-HT1D receptors | |||||
| GC30206 | Roluperidone (CYR-101) | 359625-79-9 | Sigma Receptor | ||
A dual antagonist of 5-HT2A and σ2 receptors | |||||
| GC38781 | Frovatriptan succinate hydrate | 158930-17-7 | 5-HT Receptor | ||
An agonist of 5-HT1B and 5-HT1D receptors | |||||
| GC14052 | SB 200646 hydrochloride | 143797-62-0 | 5-HT Receptor | ||
A dual antagonist of 5-HT2C and 5-HT2B receptors | |||||
