Virus Protease
Virus Protease(病毒蛋白酶)
Virus Protease 相关产品(63)
- GC10603(-)-epicatechin gallateCAS: 1257-08-5纯度: >98.00%
(-)-epicatechin gallate是一种天然黄烷醇，属于茶多酚中的酯型儿茶素类化合物，(-)-epicatechin gallate通过抑制环加氧酶-1(COX-1)发挥抗炎作用（IC₅₀=7.5μM）。
- GC10889ArtesunateCAS: 88495-63-0纯度: >98.00%
青蒿琥酯（Artesunate）是一种抗疟疾化合物，是信号转导及转录激活蛋白3（STAT-3）和膜谷胱甘肽S-转移酶（EXP1）的抑制剂。
- GC11302HinokitiolCAS: 499-44-5纯度: >99.50% / >98.00%
Hinokitiol是一种在 Formosan cypress 中天然存在的tropolone类化合物，具有抗菌和抗癌特性。
- GC14745Plerixafor (AMD3100)CAS: 110078-46-1纯度: >98.00% / >99.00%
Plerixafor(AMD3100) 是 CXCR4 和 CXCL12 介导的趋化作用的小分子抑制剂，IC50 值分别为 44 nM 和 5.7 nM 。
- GC14885Foscarnet SodiumCAS: 63585-09-1纯度: >99.50%
Foscarnet sodium (Trisodium phosphonoformate) 是一种病毒 DNA 聚合酶活性抑制剂，可导致病毒复制的可逆抑制。
- GC15706Aspirin (Acetylsalicylic acid)CAS: 50-78-2纯度: >99.50%
A non-selective, irreversible COX inhibitor
- GC18131AminothiazoleCAS: 96-50-4纯度: >98.00%
氨基噻唑（2-氨基噻唑）是一种典型的杂环胺，是合成生物活性分子的前体，包括硫化剂、杀菌剂、杀菌剂、抗生素、染料和化学反应促进剂。
- GC30056Danthron (Dantron)CAS: 117-10-2纯度: >98.50%
Danthron (Chrysazin, Antrapurol) functions in regulating glucose and lipid metabolism by activating AMPK. Danthron is a natural product extracted from the traditional Chinese medicine rhubarb. Danthron used to be a laxativa and now is currently used as an antioxidant in synthetic lubricants, in the synthesis of experimental antitumor agents, as a fungicide and as an intermediate for making dyes.
- GC30763Benzenebutyric acid (4-Phenylbutyric acid)CAS: 1821-12-1纯度: >98.00% / >99.00%
4-Phenylbutyric acid (4-PBA, Benzenebutyric acid) is a histone deacetylase (HDAC) inhibitor and a key epigenetic inducer of anti-HCV hepatic hepcidin. 4-Phenylbutyric acid inhibits LPS-induced inflammation through regulating endoplasmic-reticulum (ER) stress and autophagy in acute lung injury models.
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC10395 | Dynasore | 304448-55-3 | >98.50% / >98.00% | |
Dynasore 作为 GTPase 抑制剂，可以快速、可逆地抑制发动蛋白活性，从而阻止内吞作用。 | ||||
| GC10603 | (-)-epicatechin gallate | 1257-08-5 | >98.00% | |
(-)-epicatechin gallate是一种天然黄烷醇，属于茶多酚中的酯型儿茶素类化合物，(-)-epicatechin gallate通过抑制环加氧酶-1(COX-1)发挥抗炎作用（IC₅₀=7.5μM）。 | ||||
| GC10889 | Artesunate | 88495-63-0 | >98.00% | |
青蒿琥酯（Artesunate）是一种抗疟疾化合物，是信号转导及转录激活蛋白3（STAT-3）和膜谷胱甘肽S-转移酶（EXP1）的抑制剂。 | ||||
| GC11302 | Hinokitiol | 499-44-5 | >99.50% / >98.00% | |
Hinokitiol是一种在 Formosan cypress 中天然存在的tropolone类化合物，具有抗菌和抗癌特性。 | ||||
| GC11877 | ESI-09 | 263707-16-0 | >98.50% | |
ESI-09是一种新型且具有细胞渗透性和特异性的cAMP直接激活交换蛋白（EPAC）抑制剂，对EPAC1和EPAC2的IC 50 值分别为3.2和1.4μM。 | ||||
| GC12943 | STING agonist-1 | 702662-50-8 | >99.50% | |
An indirect activator of STING signaling | ||||
| GC13089 | PIK-93 | 593960-11-3 | >99.00% | |
A PI4KIIIβ inhibitor | ||||
| GC13433 | AZ 960 | 905586-69-8 | >98.00% | |
A JAK2 inhibitor | ||||
| GC13596 | SRPIN340 | 218156-96-8 | >99.50% | |
A selective inhibitor of SRPK1 | ||||
| GC13793 | NH125 | 278603-08-0 | >98.00% | |
NH125是一种多靶标的活性物质，是多种组氨酸蛋白激酶家族成员的抑制剂，其中NH125可抑制真核延长因子2激酶（eEF-2K）活性，IC 50 =60nM。 | ||||
| GC14745 | Plerixafor (AMD3100) | 110078-46-1 | >98.00% / >99.00% | |
Plerixafor(AMD3100) 是 CXCR4 和 CXCL12 介导的趋化作用的小分子抑制剂，IC50 值分别为 44 nM 和 5.7 nM 。 | ||||
| GC14885 | Foscarnet Sodium | 63585-09-1 | >99.50% | |
Foscarnet sodium (Trisodium phosphonoformate) 是一种病毒 DNA 聚合酶活性抑制剂，可导致病毒复制的可逆抑制。 | ||||
| GC15116 | Probucol | 23288-49-5 | >99.50% | |
An antioxidant and hypocholesterolemic compound | ||||
| GC15706 | Aspirin (Acetylsalicylic acid) | 50-78-2 | >99.50% | |
A non-selective, irreversible COX inhibitor | ||||
| GC16086 | Phenytoin | 57-41-0 | >99.50% | |
An anticonvulsant agent | ||||
| GC16386 | Tubacin | 537049-40-4 | >95.00% | |
Tubacin (tubulin acetylation inducer)是一种选择性抑制组蛋白去乙酰化酶6 (HDAC6)，诱导α-微管蛋白乙酰化的小分子，IC50为0.004µM。 | ||||
| GC16553 | N-Desmethylclozapine | 6104-71-8 | >99.50% | |
An active metabolite of clozapine | ||||
| GC17949 | Plerixafor 8HCl (AMD3100 8HCl) | 155148-31-5 | >99.00% | |
An antagonist of CXCR4 | ||||
| GC18131 | Aminothiazole | 96-50-4 | >98.00% | |
氨基噻唑（2-氨基噻唑）是一种典型的杂环胺，是合成生物活性分子的前体，包括硫化剂、杀菌剂、杀菌剂、抗生素、染料和化学反应促进剂。 | ||||
| GC18485 | Retro-2 | 1429192-00-6 | >98.00% | |
Retro-2是一种强效埃博拉病毒（EBOV）感染抑制剂，EC 50 值为12.2μM。 | ||||
| GC19082 | Brequinar | 96187-53-0 | >99.50% / >98.00% | |
布喹那（Brequinar）是一种特异性的二氢乳清酸脱氢酶DHODH抑制剂，在体外IC50值约为20nM。 | ||||
| GC30056 | Danthron (Dantron) | 117-10-2 | >98.50% | |
Danthron (Chrysazin, Antrapurol) functions in regulating glucose and lipid metabolism by activating AMPK. Danthron is a natural product extracted from the traditional Chinese medicine rhubarb. Danthron used to be a laxativa and now is currently used as an antioxidant in synthetic lubricants, in the synthesis of experimental antitumor agents, as a fungicide and as an intermediate for making dyes. | ||||
| GC30763 | Benzenebutyric acid (4-Phenylbutyric acid) | 1821-12-1 | >98.00% / >99.00% | |
4-Phenylbutyric acid (4-PBA, Benzenebutyric acid) is a histone deacetylase (HDAC) inhibitor and a key epigenetic inducer of anti-HCV hepatic hepcidin. 4-Phenylbutyric acid inhibits LPS-induced inflammation through regulating endoplasmic-reticulum (ER) stress and autophagy in acute lung injury models. | ||||
| GC30785 | 4E2RCat | 432499-63-3 | >98.00% | |
4E2RCat是eIF4E-eIF4G相互作用的抑制剂，IC50值为13.5μM。 | ||||