Hippo Signaling

Hippo Signaling(Hippo信号通路)

Hippo signaling is a conserved pathway for organ size control by modulating cell proliferation, apoptosis and tissue-specific stem cell regeneration. It is associated with carcinogenesis.

Hippo Signaling 相关产品(6)

  • GC14482 structure
    GC14482Verteporfin
    CAS: 129497-78-5
    纯度: >98.00%

    维替泊芬是一种有效的 PD-L1 表达抑制剂,用于治疗年龄相关性黄斑变性、鲜红斑痣和癌症。

  • GC11245 structure
    GC11245XMU-MP-1
    CAS: 2061980-01-4
    纯度: >99.00%

    XMU-MP-1是可逆的、选择性的MST1/2激酶的抑制剂,对MST1和MST2的IC 50 分别为71.1±12.9 nM和38.1±6.9 nM。

  • GC32914 structure
    GC32914EMT inhibitor-1
    CAS: 1638526-21-2
    纯度: >99.00%

    EMTinhibitor-1是Hippo,TGF-β和Wnt信号通路的抑制剂,并拥有抗肿瘤活性。

  • GC61410 structure
    GC61410I3MT-3
    CAS: 459420-09-8
    纯度: >98.00%

    I3MT-3 (HMPSNE, compound 3) is a potent, selective, and cell-membrane permeable inhibitor of 3-mercaptopyruvate sulfurtransferase (3MST) with IC50 of 2.7 μM. I3MT-3 targets a persulfurated cysteine residue located in the active site of 3MST.

  • GC69261 structure
    GC69261IHMT-MST1-58
    CAS: 2414484-25-4
    纯度: >99.00%

    IHMT-MST1-58 是一种有效的、选择性的 STE20-like protein 1 kinase (MST1) 抑制剂,具有口服活性,IC50 值为 23 nM。IHMT-MST1-58 可用于 1 型或 2 型糖尿病的研究。

  • GC73860 structure
    GC73860JA310
    CAS: 3022928-90-8
    纯度: >99.50%

    JA310是一种高选择性MST3激酶抑制剂。