Transcription Factors
Transcription Factors(转录因子)
Transcription Factors 相关产品(111)
- GC13941Cyclosporin ACAS: 59865-13-3纯度: >98.00% / >97.00% / >99.00%
Cyclosporin A是一种免疫抑制剂,其主要的三个靶点是亲环蛋白、钙调神经磷酸酶和转运蛋白,其抑制亲环蛋白A和钙调神经磷酸酶活性的IC 50 分别为360nM和5nM。
- GC14266CCG 203971CAS: 1443437-74-8纯度: >99.00%
An inhibitor of the Rho/MKL1/SRF transcriptional pathway
- GC14832N-3-oxo-octanoyl-L-Homoserine lactoneCAS: 147795-39-9纯度: >97.00%
N-3-Oxo-octanoyl-L-homoserine lactone是一种属于N-酰基高丝氨酸内酯(AHL)家族的群体感应信号分子,常用于研究细菌通讯和生物膜形成。
- GC16227Anhydrotetracycline (hydrochloride)CAS: 13803-65-1纯度: >98.00%
Anhydrotetracycline (hydrochloride)是一种四环素生物合成前体,是竞争性四环素破坏酶广谱抑制剂。Anhydrotetracycline (hydrochloride)是真核细胞中四环素阻遏蛋白(TetR)和反向四环素阻遏蛋白(revTetR)转录抑制因子的调节因子。
- GC18773(Rac)-BenpyrineCAS: 1333714-43-4纯度: >99.00%
An inhibitor of the TNF-α-TNFR1 protein-protein interaction
- GC18796Herbicidin ACAS: 55353-31-6纯度: >98.00%
An adenine nucleoside antibiotic with herbicidal activity
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC16165 | T-5224 | 530141-72-1 | >98.00% | |
T-5224 是一种非肽类小分子 AP-1 抑制剂,特异性抑制 AP-1 与启动子区 AP-1 结合位点的结合,最初开发为抗炎药用于治疗类风湿性关节炎 (RA) 抑制炎症细胞因子和 MMPs 而没有任何副作用。 | ||||
| GC10151 | OAC1 | 300586-90-7 | >99.00% / >98.00% | |
An Oct4-activating compound | ||||
| GC10233 | BRD 7552 | 1137359-47-7 | >98.00% | |
An inducer of PDX1 expression | ||||
| GC10724 | OAC3 | 182564-41-6 | - | |
An Oct4-activating compound | ||||
| GC11197 | KL 001 | 309928-48-1 | >97.00% | |
A cryptochrome protein stabilizer | ||||
| GC11307 | ML-264 | 1550008-55-3 | >99.50% | |
A selective KLF5 inhibitor | ||||
| GC12499 | O4I1 | 175135-47-4 | - | |
An inducer of Oct3/4 | ||||
| GC12727 | Ro 5-3335 | 30195-30-3 | >99.50% | |
Ro 5-3335 是一种苯二氮卓类药物,可作为核心结合因子 (CBF) 白血病的抑制剂。 Ro 5-3335 是一种 RUNX1-CBFβ 相互作用抑制剂,可抑制 RUNX1/CBFB 依赖性反式激活。 | ||||
| GC13231 | BI 6015 | 93987-29-2 | >95.00% | |
An HNF4α antagonist | ||||
| GC13941 | Cyclosporin A | 59865-13-3 | >98.00% / >97.00% / >99.00% | |
Cyclosporin A是一种免疫抑制剂,其主要的三个靶点是亲环蛋白、钙调神经磷酸酶和转运蛋白,其抑制亲环蛋白A和钙调神经磷酸酶活性的IC 50 分别为360nM和5nM。 | ||||
| GC14266 | CCG 203971 | 1443437-74-8 | >99.00% | |
An inhibitor of the Rho/MKL1/SRF transcriptional pathway | ||||
| GC14685 | CID 5951923 | 749872-43-3 | - | |
A KLF5 inhibitor | ||||
| GC14832 | N-3-oxo-octanoyl-L-Homoserine lactone | 147795-39-9 | >97.00% | |
N-3-Oxo-octanoyl-L-homoserine lactone是一种属于N-酰基高丝氨酸内酯(AHL)家族的群体感应信号分子,常用于研究细菌通讯和生物膜形成。 | ||||
| GC15474 | CBFβ Inhibitor | 493028-20-9 | - | |
Binds CBFβ and disrupts CBF function | ||||
| GC16227 | Anhydrotetracycline (hydrochloride) | 13803-65-1 | >98.00% | |
Anhydrotetracycline (hydrochloride)是一种四环素生物合成前体,是竞争性四环素破坏酶广谱抑制剂。Anhydrotetracycline (hydrochloride)是真核细胞中四环素阻遏蛋白(TetR)和反向四环素阻遏蛋白(revTetR)转录抑制因子的调节因子。 | ||||
| GC17327 | OAC2 | 6019-39-2 | >99.50% | |
An Oct4-activating compound | ||||
| GC17839 | Stauprimide | 154589-96-5 | - | |
Primes stem cells for differentiation | ||||
| GC18169 | FX1 | 1426138-42-2 | >98.00% | |
A BCL6 inhibitor | ||||
| GC18194 | 4-Epidoxycycline | 6543-77-7 | - | |
A metabolite of doxycycline | ||||
| GC18392 | Cellocidin | 543-21-5 | - | |
An antibiotic | ||||
| GC18624 | Roslin-2 | 29574-21-8 | - | |
A reactivator of p53 | ||||
| GC18652 | FQI 1 | 599151-35-6 | - | |
An inhibitor of Late SV40 Factor | ||||
| GC18773 | (Rac)-Benpyrine | 1333714-43-4 | >99.00% | |
An inhibitor of the TNF-α-TNFR1 protein-protein interaction | ||||
| GC18796 | Herbicidin A | 55353-31-6 | >98.00% | |
An adenine nucleoside antibiotic with herbicidal activity | ||||
