PAD
PAD(肽精氨酸脱氨酶)
PAD 相关产品(21)
- GC32303Streptonigrin (Bruneomycin)CAS: 3930-19-6
A phenylpyridylquinoline with diverse biological activities
- GC35706Cl-amidineCAS: 913723-61-2纯度: >98.00% / >97.00%
Cl-amidine is an irreversible pan-peptidylarginine deiminase (PAD) inhibitor with IC50 values of 5.9 ± 0.3 μM, 0.8 ± 0.3 μM, 6.2 ± 1.0 μM for PAD4, PAD1 and PAD3, respectively. Cl-amidine induces apoptosis.
- GC43789GSK199 (hydrochloride)CAS: 1549811-53-1纯度: >98.00%
GSK199 (hydrochloride)是一种具有口服活性和可逆性的选择性肽基精氨酸脱亚氨酶4(PAD4)抑制剂,在缺少钙离子情况下IC 50 值为200nM。
- GC45548Photoswitchable PAD Inhibitor (technical grade)CAS: 2226393-62-8纯度: >70.00%
A photoactivated PAD inhibitor
- GC48263YW3-56 (hydrochloride) (technical grade)CAS: 2309756-20-3纯度: >80.00%
A PAD2 and PAD4 inhibitor
- GC91565GSK199 analog (hydrochloride)CAS: 2048226-46-4纯度: >95.00%
GSK199 analog is an inhibitor of peptidyl arginine deiminase 4 (PAD4) and a derivative of the PAD4 inhibitor GSK199.
| 货号 | 产品名称 | CAS号 | 纯度 | 结构 |
|---|---|---|---|---|
| GC18925 | Cl-Amidine (hydrochloride) | 1373232-26-8 | >98.50% | |
A PAD inhibitor | ||||
| GC19184 | GSK484 hydrochloride | 1652591-81-5 | >98.00% | |
GSK484是一种选择性PAD4抑制剂,已被用作抗缺血化合物,对PAD4具有抑制活性。 | ||||
| GC31755 | BB-Cl-Amidine | 1802637-39-3 | - | |
BB-Cl-Amidine 是一种肽基精氨酸脱氨酶 (PAD) 抑制剂,常用于研究 PAD 功能。 | ||||
| GC32303 | Streptonigrin (Bruneomycin) | 3930-19-6 | - | |
A phenylpyridylquinoline with diverse biological activities | ||||
| GC33261 | YW3-56 | 1374311-17-7 | - | |
YW3-56是有效的肽酰精氨酸脱亚胺酶(PAD)抑制剂,其对PAD4的IC50值为1-5μM。 | ||||
| GC35480 | BB-Cl-Amidine hydrochloride | 2436747-41-8 | >99.00% | |
A PAD4 inhibitor | ||||
| GC35706 | Cl-amidine | 913723-61-2 | >98.00% / >97.00% | |
Cl-amidine is an irreversible pan-peptidylarginine deiminase (PAD) inhibitor with IC50 values of 5.9 ± 0.3 μM, 0.8 ± 0.3 μM, 6.2 ± 1.0 μM for PAD4, PAD1 and PAD3, respectively. Cl-amidine induces apoptosis. | ||||
| GC40098 | BB-Cl-Yne | 2219324-71-5 | >98.00% | |
A clickable PAD inhibitor | ||||
| GC42910 | BB-F-Yne | 2219331-30-1 | >98.00% | |
A clickable PAD inhibitor | ||||
| GC43202 | CAY10723 | 2095107-57-4 | >98.00% | |
A PAD2 inhibitor | ||||
| GC43651 | F-Amidine (trifluoroacetate salt) | 877617-46-4 | >95.00% | |
A PAD inhibitor | ||||
| GC43788 | GSK121 (trifluoroacetate salt) | 1652591-80-4 | >98.00% | |
A PAD4 inhibitor | ||||
| GC43789 | GSK199 (hydrochloride) | 1549811-53-1 | >98.00% | |
GSK199 (hydrochloride)是一种具有口服活性和可逆性的选择性肽基精氨酸脱亚氨酶4(PAD4)抑制剂,在缺少钙离子情况下IC 50 值为200nM。 | ||||
| GC45005 | TDFA (trifluoroacetate salt) | - | >98.00% | |
A PAD4 inhibitor | ||||
| GC45402 | CAY10729 (trifluoroacetate salt) (technical grade) | - | >70.00% | |
A PAD1 inhibitor | ||||
| GC45548 | Photoswitchable PAD Inhibitor (technical grade) | 2226393-62-8 | >70.00% | |
A photoactivated PAD inhibitor | ||||
| GC47050 | CAY10727 | 1671088-84-8 | >90.00% | |
A PAD3 inhibitor | ||||
| GC48263 | YW3-56 (hydrochloride) (technical grade) | 2309756-20-3 | >80.00% | |
A PAD2 and PAD4 inhibitor | ||||
| GC48495 | BMS-P5 | 1550371-22-6 | >99.50% | |
A PAD4 inhibitor | ||||
| GC90710 | CAY10723 (hydrochloride) | - | >95.00% | |
一种PAD2抑制剂 | ||||
| GC91565 | GSK199 analog (hydrochloride) | 2048226-46-4 | >95.00% | |
GSK199 analog is an inhibitor of peptidyl arginine deiminase 4 (PAD4) and a derivative of the PAD4 inhibitor GSK199. | ||||
