GlpBio

(Rac)-CP-601927 hydrochloride

目录号: GC63511纯度: >98%
COASDSData Sheet
(Rac)-CP-601927 hydrochloride 是 CP-601927 的外消旋物。CP-601927 是一种 nAChR 激动剂，对 α4β2 和 α3β4 nAChR 的 Ki 值分别为 1.2 nM 和 102 nM。
(Rac)-CP-601927 hydrochloride
Cas No.: 230615-01-7
规格价格库存数量操作
5 mg¥3,420.00现货
1
10 mg¥5,400.00现货
1
25 mg¥10,350.00现货
1
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产品描述 Description

(Rac)-CP-601927 hydrochloride is the racemate of CP-601927. CP-601927 is a nAChR agonist with Ki values 1.2 nM and 102 nM for α4β2 and α3β4 nAChR, respectively[1].

CP-601927 induces significant antidepressant-like effects in mice. CP-601927 could decrease cholinergic signaling as a result of its reduced efficacy or via desensitization of α4β2* nAChRs[1].

[1]. Yann S Mineur, et al. α4β2 nicotinic acetylcholine receptor partial agonists with low intrinsic efficacy have antidepressant-like properties. Behav Pharmacol. 2011 Aug;22(4):291-9.

产品文档 Product Documents

Purity:>98%
COASDSData Sheet

化学性质Chemical Properties

CAS 号
230615-01-7
分子式
C12H13ClF3N
分子量
263.69 g/mol
溶解性
DMSO : 100 mg/mL (379.23 mM; Need ultrasonic); H<sub>2</sub>O : 100 mg/mL (379.23 mM; Need ultrasonic)
保存条件
4&#176;C, away from moisture
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
为了提高溶解度，请将管子加热至 37°C，然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案：配备蓝冰进行发货。所有其他可用尺寸：配备 RT，或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol