GlpBio

Prolyl Endopeptidase Inhibitor 1

目录号: GC38838纯度: >98%同义词: Boc-Pro-prolinal; (Boc)-Prolyl-prolinal; BPP
COASDSData Sheet
Prolyl Endopeptidase Inhibitor 1 (Boc-Pro-prolinal) 是一种有效的脯氨酸内肽酶 (PEP; PE) 抑制剂，Ki 值为 15 nM。Prolyl endopeptidase-IN-1 具有抗遗忘作用。
Prolyl Endopeptidase Inhibitor 1
Cas No.: 86925-97-5
规格价格库存数量操作
1mg¥1,170.00现货
1
5mg¥2,610.00现货
1
10mg¥4,140.00现货
1
10mM (in 1mL DMSO)¥3,814.00现货
1
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产品描述 Description

Prolyl Endopeptidase Inhibitor 1 (Boc-Pro-prolinal) is a potent prolyl endopeptidase (PEP; PE) inhibitor, with a Ki value of 15 nM. Prolyl Endopeptidase Inhibitor 1 has anti-amnesic effect[1].

Prolyl Endopeptidase Inhibitor 1 (Boc-Pro-prolinal) strongly inhibits the mammalian prolyl endopeptidase with a Ki value of nM order, while the Ki value for the microbial enzyme is only of microM order (Ki=3.2 μM for Flavobacterium)[1].

[1]. Yoshimoto T, et al. Specific inhibitors for prolyl endopeptidase and their anti-amnesic effect. J Pharmacobiodyn. 1987 Dec;10(12):730-5. [2]. Yoshimoto T, et al. Comparison of inhibitory effects of prolinal-containing peptide derivatives on prolyl endopeptidases from bovine brain and Flavobacterium. J Biochem. 1985 Oct;98(4):975-9.

产品文档 Product Documents

Purity:>98%
COASDSData Sheet

化学性质Chemical Properties

CAS 号
86925-97-5
同义词
Boc-Pro-prolinal; (Boc)-Prolyl-prolinal; BPP
SMILES
O=C(N1[C@H](C(N2[C@H](C=O)CCC2)=O)CCC1)OC(C)(C)C
分子式
C15H24N2O4
分子量
296.36 g/mol
溶解性
DMSO : 100 mg/mL (337.43 mM; Need ultrasonic)
保存条件
Store at -20°C
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
为了提高溶解度，请将管子加热至 37°C，然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案：配备蓝冰进行发货。所有其他可用尺寸：配备 RT，或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol