Isotope-Labeled Compounds(同位素标记化合物)
- 13C(77)
- 15N(12)
- Deuterium(630)
- Isotope-Labeled Amino Acids & Peptides(1)
- Isotope-Labeled Fatty Acids(2)
- Isotope-Labeled Synthetic Intermediates(5)
- Cat.No. 产品名称 Information
-
GC46258
(±)14(15)-DiHET-d11
(±)14,15-DiHETrE-d11
A neuropeptide with diverse biological activities
-
GC46257
(±)12(13)-EpOME-d4
(±)12,13-EODE-d4, Isoleukotoxin-d4, (±)Vernolic Acidd4
A neuropeptide with diverse biological activities
-
GC46256
(±)12(13)-DiHOME-d4
Isoleukotoxin diold4
A neuropeptide with diverse biological activities
-
GC46252
(±)11(12)-DiHET-d11
(±)11(12)-DHET-d11, (±)11,12-DiHETrE-d11
A neuropeptide with diverse biological activities
-
GC46251
(+)-Norpropoxyphene-d5 (maleate)
A neuropeptide with diverse biological activities
-
GC46246
(-)-Hyoscyamine-d3
L-Hyoscyamine-d3, (S)-Hyoscyamine-d3
A neuropeptide with diverse biological activities
-
GC61148
O-Desmethyl Midostaurin-d5
CGP62221-d5; O-Desmethyl PKC412-d5
O-DesmethylPKC412-d5(CGP62221-d5)是O-DesmethylPKC412的氘代物。O-DesmethylMidostaurin(CGP62221;O-DesmethylPKC412)是Midostaurin的活性代谢物,通过细胞色素P450肝酶代谢产生,可以作为Midostaurin在体内代谢的指标之一。
-
GC61064
Midostaurin-D5
PKC412-d5; CGP 41251-d5
Midostaurin-D5(PKC412-D5)是Midostaurin的氘代化合物。Midostaurin是一种多靶点蛋白激酶抑制剂,抑制PKCα/β/γ,Syk,Flk-1,Akt,PKA,c-Kit,c-Fgr,c-Src,FLT3,PDFRβ和VEGFR1/2的活性,IC50值为22-500nM。
-
GC60837
Fenpiverinium D3 bromide
FenpiveriniumD3bromide是Fenpiveriniumbromide的氘代物。Fenpiveriniumbromide具有抗胆碱能和抗痉挛作用。
-
GC60746
Debutyldronedarone D6 hydrochloride
D-盐酸丁二酮,SR35021 D6 hydrochloride
DebutyldronedaroneD6hydrochloride(SR35021D6hydrochloride)是Debutyldronedarone的氘代物。Debutyldronedarone是Dronedarone在人体中的主要循环活性代谢物(metabolite)。Debutyldronedarone的效力是Dronedarone的1/10到1/3。
-
GC60713
cis-Clopidogrel-MP Derivative 13CD3
Clopidogrel-MP-AM-13C,d3
cis-Clopidogrel-MPDerivative13CD3(Clopidogrel-MP-AM13CD3)是一种cis-Clopidogrel-MPDerivative氘代物。cis-Clopidogrel-MPDerivative(Clopidogrel-MP-AM)是Clopidogrel活性代谢产物的3'-甲氧基苯乙酮衍生物。Clopidogrel是一种具有口服活性血小板抑制剂,靶向P2Y12受体。
-
GC60573
Alkyne tyramide
Alk-Ph
Alkyne tyramide是一种可点击的抗坏血酸过氧化物酶2(APEX2)探针,具有水溶性和细胞壁渗透性,可显著提高完整酵母细胞中的APEX标记效率,还有助于识别APEX标记位点,从而可以明确分配线粒体蛋白的膜拓扑结构。
-
GC60420
(S)-Praziquantel D11
(S)-PraziquantelD11是(S)-Praziquantel的氘代物。(S)-Praziquantel是Praziquantel的有毒对映异构体,对蠕虫无效。
-
GC60400
(E)-10-Hydroxynortriptyline D3
E-10-OH-NT-d3
(E)-10-HydroxynortriptylineD3(E-10-OH-NTD3)是(E)-10-HydroxyNortriptyline的一种氘代化合物。(E)-10-HydroxyNortriptyline是Nortriptyline的代谢物。Nortriptyline是三环类抗抑郁药,是Amitriptyline的主要活性代谢物,用于缓解抑郁症状。
-
GC39722
Phenylacetylglutamine-D5
N-苯乙酰基-L-谷氨酰胺-D5,NSC 203800-d5; Phenylacetyl-L-glutamine-d5
Phenylacetylglutamine-D5 (NSC 203800-D5;Phenylacetyl-L-glutamine-D5) 是 Phenylacetylglutamine 的一种氘代化合物。Phenylacetylglutamine 是一种结肠微生物代谢物,源于氨基酸发酵。
-
GC39582
Methimazole D3
甲巯咪唑 D3
An internal standard for the quantification of methimazole
-
GC50190
Fenretinide - d4
4-HPR-d4, 4-Hydroxy(phenyl)retinamide-d4, Retinoic Acid p-hydroxyphenylamide-d4
An internal standard for the quantification of fenretinide
-
GC46232
Tiamulin-d10 (hydrochloride)
泰妙菌素盐酸盐-D10
An internal standard for the quantification of tiamulin
-
GC46191
Oclacitinib-13C-d3
A neuropeptide with diverse biological activities
-
GC46153
Hexacosanoic Acid methyl ester-d3
C26:0 methyl ester-d3, Ceric Acid methyl ester-d3, Cerotic Acid methyl ester-d3
A neuropeptide with diverse biological activities
-
GC46125
Dantrolene-d4
A neuropeptide with diverse biological activities
-
GC46120
Cisapride-d6
A neuropeptide with diverse biological activities
-
GC46084
Almorexant-13C-d3
ACT 078573-13C,d3
具有多种生物活性的神经肽
-
GC46051
1-Palmitoyl-d9-2-Arachidonoyl-3-Palmitoyl-sn-glycerol
1-Palmitin-d9-2-Arachidonin-3-Palmitin, TG(16:0-d9/20:4/16:0)
A neuropeptide with diverse biological activities
-
GC46048
17(S)-HDHA-d5
17(S)-Hydroxy docosahexaenoic acid-d5, 17(S)-HDoHE-d5
A neuropeptide with diverse biological activities
-
GC45922
(±)11(12)-EET-d11 methyl ester
(±)11,12-EpETrE-d11 methyl ester
A neuropeptide with diverse biological activities
-
GC45921
(±)8(9)-EET-d11 methyl ester
(±)8,9-EpETrE-d11 methyl ester
A neuropeptide with diverse biological activities
-
GC45920
(±)14(15)-EET-d11 methyl ester
(±)14,15-EpETrE-d11 methyl ester
A neuropeptide with diverse biological activities
-
GC45919
(±)5(6)-EET-d11 methyl ester
(±)5,6-EpETrE-d11 methyl ester
A neuropeptide with diverse biological activities
-
GC45902
Trametinib-13C-d3
GSK1120212-13C,d3; JTP-74057-13C,d3
A neuropeptide with diverse biological activities
-
GC45894
Daunorubicin-13C-d3
A neuropeptide with diverse biological activities
-
GC45892
Caspofungin-d4 (acetate)
A neuropeptide with diverse biological activities
-
GC45886
Levofloxacin-d8 (hydrochloride)
A neuropeptide with diverse biological activities
-
GC45882
(±)-Jasmonic Acid-d5
A neuropeptide with diverse biological activities
-
GC45879
Palonosetron-d3 (hydrochloride)
盐酸帕洛诺司琼 d3 (盐酸盐)
A neuropeptide with diverse biological activities
-
GC45829
Troglitazone-d4
CS-045-d4
Troglitazone-d4 是氘标记的曲格列酮。 Troglitazone 是一种 PPARγ 激动剂,对人和鼠 PPARγ 受体的 EC50 分别为 550 nM 和 780 nM。
-
GC45820
Balsalazide-d4
Balsalazide-d4 是氘标记的 Balsalazide。
-
GC45819
Indacaterol-d3
An internal standard for the quantification of indacaterol
-
GC45801
Hesperetin-13C-d3
A neuropeptide with diverse biological activities
-
GC45800
Cytarabine-13C3
Ara-C-13C3, 1-β-D-Arabinofuranosylcytosine-13C3
A neuropeptide with diverse biological activities
-
GC45797
Cloxacillin-13C4 (sodium salt)
A neuropeptide with diverse biological activities
-
GC45794
Linaclotide-d4
A neuropeptide with diverse biological activities
-
GC45788
Maraviroc-d6
马拉韦罗D6
An internal standard for the quantification of maraviroc
-
GC45787
Moxidectin-d3
CL-301423-d3
A neuropeptide with diverse biological activities
-
GC45786
Lomitapide-d8
AEGR-733-d8; BMS-201038-d8
A neuropeptide with diverse biological activities
-
GC45768
Pranlukast-d4
ONO-1078-d4
A neuropeptide with diverse biological activities
-
GC45766
Amprenavir-d4
安瑞那韦 d4
A neuropeptide with diverse biological activities
-
GC45764
Ciclopirox-d11 (sodium salt)
HOE 296b-d11
A neuropeptide with diverse biological activities
-
GC45762
Acitretin-d3
Ro 10-1670-d3
A neuropeptide with diverse biological activities
-
GC45754
Lenvatinib-d4
E7080-d4
Lenvatinib-d4 (E7080-d4) 是氘标记的 Lenvatinib。 Lenvatinib (E7080) 是一种口服的多靶点酪氨酸激酶抑制剂,可抑制 VEGFR1-3、FGFR1-4、PDGFR、KIT 和 RET,显示出有效的抗肿瘤活性。