GlpBio

GPR35 agonist 3

目录号: GC70651纯度: >98.00%
GPR35 agonist 3是一种合成的GPR35激动剂，EC50值为1.4μM。
GPR35 agonist 3
Cas No.: 123021-85-2
规格价格库存数量操作
5 mg¥864.00现货
1
10 mg¥1,368.00现货
1
25 mg¥2,808.00现货
1
50 mg¥4,500.00现货
1
100 mg¥7,186.00现货
1
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产品描述 Description

GPR35 agonist 3 is a synthetic GPR35 agonist with an EC50value of 1.4 μM. GPR35 agonist 3 can be used for the research of various diseases, such as gastric cancer, type 2 diabetes, cardiovascular diseases, immune system and peripheral nervous system.

GPR35 agonist 3 shows GPR35 agonist potency with an EC50 value of 1.4 μM[1].
GPR35 agonist 3 has affinity and potency for GPR35 with values of 0.0508μM (Ki) and 0.349 μM (IC50)[1].

References:
[1]. Dominik Thimm, et al. 6-Bromo-8-(4-[(3)H]methoxybenzamido)-4-oxo-4H-chromene-2-carboxylic Acid: a powerful tool for studying orphan G protein-coupled receptor GPR35. J Med Chem

产品文档 Product Documents

Purity:>98.00%

化学性质Chemical Properties

CAS 号
123021-85-2
分子式
C12H9NO5S
分子量
279.27 g/mol
溶解性
DMSO : 125 mg/mL (447.60 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
保存条件
4°C, protect from light
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
为了提高溶解度，请将管子加热至 37°C，然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案：配备蓝冰进行发货。所有其他可用尺寸：配备 RT，或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol