GlpBio

Timapiprant sodium

目录号: GC37795纯度: >99.50%同义词: OC000459 sodium
Timapiprant sodium (OC000459 sodium), a potent, selective, and orally active D prostanoid receptor 2 (DP2, also known as CRTH2) antagonist, potently displaces [3H]PGD2 from human recombinant DP2, rat recombinant DP2, and human native DP2 with Ki values of 13, 3 and 4 nM, respectively.
Timapiprant sodium
Cas No.: 950688-14-9
规格价格库存数量操作
5mg¥540.00现货
1
10mg¥864.00现货
1
50mg¥2,880.00现货
1
100mg询价现货
1
200mg询价现货
1
10mM (in 1mL DMSO)¥594.00现货
1
Free Sample (0.1-0.5 mg)询价现货
1
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文献被引

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产品描述 Description

Timapiprant sodium (OC000459 sodium), a potent, selective, and orally active D prostanoid receptor 2 (DP2, also known as CRTH2) antagonist, potently displaces [3H]PGD2 from human recombinant DP2, rat recombinant DP2, and human native DP2 with Ki values of 13, 3 and 4 nM, respectively.

[1] Singh D, et al. Eur Respir J. 2013 Jan;41(1):46-52.

产品文档 Product Documents

Purity:>99.50%

化学性质Chemical Properties

CAS 号
950688-14-9
同义词
OC000459 sodium
SMILES
OC(CN1C2=CC=C(F)C=C2C(CC3=NC4=C(C=CC=C4)C=C3)=C1C)=O.[Na+]
分子式
C21H17FN2NaO2+
分子量
371.36 g/mol
溶解性
DMSO: 100 mg/mL (270.01 mM)
保存条件
Store at -20°C
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
为了提高溶解度，请将管子加热至 37°C，然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案：配备蓝冰进行发货。所有其他可用尺寸：配备 RT，或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol