Cathepsin Inhibitor 2

目录号: GC33892纯度: >98%
CathepsinInhibitor2是一种有效的CathepsinS抑制剂,Ki值<20nM。详细信息请参考专利文献WO2009123623A1中的段落0229。

Cathepsin Inhibitor 2
Cas No.: 1017931-53-1
规格价格库存数量操作
1mg¥3,834.00现货
1

文献被引

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产品描述 Description

Cathepsin Inhibitor 2 is a potent Cathepsin S inhibitor extracted from patent WO2009123623A1, has a Ki of <20 nM.

Cathepsin Inhibitor 2 (Please refer to paragraph 0229 for detailed information) potently inhibits Cathepsin S, Cathepsin F, Cathepsin L, and Cathepsin B with Kis of <20 nM, 21-500 nM, 21-500 nM, and 21-500 nM, respectively[1].

[1]. LINK, John, O, et al. DI-FLUORO CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS. WO2009123623A1.

产品文档 Product Documents

化学性质Chemical Properties

CAS 号
1017931-53-1
SMILES
FC(F)(F)[C@H](C1=CC=C(F)C=C1)N[C@@H](CC(F)(F)CCC)C(NC2(CC2)C#N)=O
分子式
C19H21F6N3O
分子量
421.38 g/mol
溶解性
DMSO : 100 mg/mL (237.32 mM; Need ultrasonic)
保存条件
Store at -20&#176;C
General tips
请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。
储备液的保存方式和期限:-80°C 储存时,请在 6 个月内使用,-20°C 储存时,请在 1 个月内使用。
为了提高溶解度,请将管子加热至 37°C,然后在超声波浴中震荡一段时间。
Shipping Condition
评估样品解决方案:配备蓝冰进行发货。所有其他可用尺寸:配备 RT,或根据请求配备蓝冰。

计算工具摩尔浓度 / 稀释 / 分子量 / 单位换算 / 体内配方 / 溶解度

g/mol