GlpBio

关于 "Hypertension" 的结果10 个结果

货号产品名称CAS 号靶点化学结构
GC33770Anti-hypertensive sulfonanilide 1129280-22-4OthersGC33770 structure
Anti-hypertensivesulfonanilide1是有效抗高血压剂,来自专利EP0338793A2,化合物XVIIIa,b*,实例1。
GC14977Minoxidil38304-91-5Potassium ChannelGC14977 structure
An anti-hypertensive vasodilator
GC34912Levamlodipine besylate150566-71-5Calcium ChannelGC34912 structure
Levamlodipine Besylate is a powerful dihydropyridine calcium channel blocker, possessing vasodilation properties and used in the treatment of hypertension and angina.
GC25140Bisoprolol66722-44-9Adrenergic ReceptorGC25140 structure
Bisoprolol is a cardioselective β1-adrenergic blocking agent used for secondary prevention of myocardial infarction (MI), heart failure, angina pectoris and mild to moderate hypertension.
GC32508Nanofin (2,6-Lupetidine)504-03-0OthersGC32508 structure
Nanofin (2,6-Dimethylpiperidine, Lupetidine, Naniopinum) is a ganglion blocker alkaloid having nicotinic acetylcholine receptor antagonist action. It has antihypertensive effect used for mild to moderate hypertension.
GC25663Nebivolol118457-14-0Adrenergic ReceptorGC25663 structure
Nebivolol (Bystolic,R 065824) is a β1 receptor blocker with nitric oxide-potentiating vasodilatory effect used in treatment of hypertension and also for left ventricular failure.
GC36046Fimasartan247257-48-3Angiotensin ReceptorOther ApoptosisGC36046 structure
Fimasartan (Kanarb) is a non-peptide angiotensin II receptor antagonist (ARB) with noncompetitive, insurmountable binding with the AT1 receptor. It is used for the treatment of hypertension and heart failure.
GA22715H-Lys-Tyr-OH35978-98-4GA22715 structure
Both single-dose administration and repetitive oral application of the dipeptide KY significantly decreased blood pressure in spontaneously hypertensive rats.
GB40384Terguride37686-84-3GB40384 structure

Terguride (37686-84-3) is a semi-synthetic ergoline derivative which acts as a partial dopamine D2 agonist and 5HT2B/2C receptor antagonist. Displays antiparkinsonian effects in MPTP-treated cynomolgus monkeys. Partial agonist at recruitment of β-arrestin2 to the D2 receptor. Terguride ameliorates monocrotaline-induced pulmonary hypertension in rats.

GA22011H-Ala-Leu-Pro-Met-His-Ile-Arg-OH132160-04-4GA22011 structure
The lactokinin ALPMHIR is an angiotensin-converting enzyme (ACE) inhibitory peptide, which corresponds to a sequence released by tryptic digestion from the milk protein β-lactoglobulin. It might be useful in the treatment of hypertension although its ACE inhibitory activity is about a 100 times lower than that of the antihypertensive drug captopril.