关于 "Caspase" 的结果23 个结果
- Cell-permeable Caspase-1 Inhibitor ICAS: 201608-12-0
Acetyl-AAVALLPAVLLALLAP-YVAD aldehyde, reversible inhibitor of caspase 1 (ICE).
- Caspase-3/7 Inhibitor IICAS: 775289-20-8
Potent inhibitor for caspase-3. Ac-DNLD-CHO inhibited caspase-3 (Ki app = 0.68 nM) more selectively than caspase-7, -8, and -9 (Ki app = 55.7, >200, and > 200 nM, respectively).
- Procaspase-3/6 activator 1CAS: 1100353-03-4
Procaspase-3/6 activator 1 (compound 1541) 是一种高度特异性和有效的 procaspases-3 和 -6 的激活剂,具有 EC50 值分别为 2.4 ± 0.2 和 2.8 ± 0.3 μM。Procaspase-3/6 activator 1 不会激活 procaspases-1 或 -7。
- Cell-permeable Caspase-3 Inhibitor ICAS: 201608-15-3
Acetyl-AAVALLPAVLLALLAP-DEVD-aldehyde, highly specific, potent and reversible cell-permeable inhibitor of CPP32 (Ki<1nM).
- Boc-D-FMKCAS: 634911-80-1
Boc-D-FMK is a cell-permeable broad-spectrum caspase inhibitor that fully inhibits the pro-apoptotic effect of tumor necrosis factor-α (TNFα) with the half maximal inhibition concentration IC50 value of 39 μM .
- Z-WEHD-FMKCAS: 210345-00-9
Z-WEHD-FMK 是一种有效的、细胞渗透性和不可逆的 caspase-1/5 抑制剂。 Z-WEHD-FMK 还表现出对组织蛋白酶 B 活性的强大抑制作用 (IC50=6 μM)。 Z-WEHD-FMK 可用于研究细胞凋亡的证据。
| 货号 | 产品名称 | CAS号 | 靶点 / 通路 | 引用 | 结构 |
|---|---|---|---|---|---|
| GC10787 | Caspase-8 Inhibitor Z-IETD-FMK | - | - | ||
Novel and selective caspase-8 inhibitor | |||||
| GA21257 | Cell-permeable Caspase-1 Inhibitor I | 201608-12-0 | - | ||
Acetyl-AAVALLPAVLLALLAP-YVAD aldehyde, reversible inhibitor of caspase 1 (ICE). | |||||
| GA21250 | Caspase-3/7 Inhibitor II | 775289-20-8 | - | ||
Potent inhibitor for caspase-3. Ac-DNLD-CHO inhibited caspase-3 (Ki app = 0.68 nM) more selectively than caspase-7, -8, and -9 (Ki app = 55.7, >200, and > 200 nM, respectively). | |||||
| GC43146 | Caspase-9 Inhibitor III (trifluoroacetate salt) | - | MMP | ||
A caspase-9 inhibitor | |||||
| GC74748 | Procaspase-3/6 activator 1 | 1100353-03-4 | - | ||
Procaspase-3/6 activator 1 (compound 1541) 是一种高度特异性和有效的 procaspases-3 和 -6 的激活剂,具有 EC50 值分别为 2.4 ± 0.2 和 2.8 ± 0.3 μM。Procaspase-3/6 activator 1 不会激活 procaspases-1 或 -7。 | |||||
| GC75214 | Caspase-3-IN-1 | 872254-32-5 | - | ||
Caspase-3-IN-1 (compound 11b) 是一种有效的 Caspase-3 抑制剂,其 IC50 值为 14.5 nM。 | |||||
| GA21258 | Cell-permeable Caspase-3 Inhibitor I | 201608-15-3 | - | ||
Acetyl-AAVALLPAVLLALLAP-DEVD-aldehyde, highly specific, potent and reversible cell-permeable inhibitor of CPP32 (Ki<1nM). | |||||
| GC18137 | Ivachtin | 745046-84-8 | Caspase | ||
A reversible caspase-3 inhibitor | |||||
| GC12407 | Z-IETD-FMK | 210344-98-2 | Caspase | ||
Z-IETD-FMK(Z-IE(OMe)TD(OMe)-FMK)是一种选择性和细胞可渗透的 caspase-8抑制剂。 | |||||
| GC17602 | Ac-DEVD-AFC | 201608-14-2 | Peptides | ||
A fluorogenic caspase subsrate | |||||
| GC10951 | Ac-DEVD-CMK | 285570-60-7 | Caspase | ||
An inhibitor of caspase-3 | |||||
| GC13326 | Ac-YVAD-AFC | 219137-85-6 | Fluorescence | ||
A caspase-1 and -4 substrate | |||||
| GC11993 | PAC-1 | 315183-21-2 | Other Apoptosis | ||
PAC-1是一种具有口服活性的小分子procaspase-3激活剂,可诱导癌细胞凋亡,EC50为2.08μM。 | |||||
| GC16774 | Boc-D-FMK | 634911-80-1 | Other Apoptosis | ||
Boc-D-FMK is a cell-permeable broad-spectrum caspase inhibitor that fully inhibits the pro-apoptotic effect of tumor necrosis factor-α (TNFα) with the half maximal inhibition concentration IC50 value of 39 μM . | |||||
| GC12287 | Z-DEVD-FMK | 210344-95-9 | Caspase | ||
Z-DEVD-FMK是一种特异性的不可逆的半胱氨酸-天冬氨酸蛋白酶3(caspase-3)抑制剂,IC50为18μM。 | |||||
| GC11218 | Z-VDVAD-FMK | 210344-92-6 | Caspase | ||
Z-VDVAD-FMK是一种不可逆的、具有细胞渗透性的caspase-2特异性抑制剂。 | |||||
| GC13413 | Z-VEID-FMK | 210344-96-0 | Caspase | ||
Caspase-6抑制剂 | |||||
| GC12190 | Z-WEHD-FMK | 210345-00-9 | Peptides | ||
Z-WEHD-FMK 是一种有效的、细胞渗透性和不可逆的 caspase-1/5 抑制剂。 Z-WEHD-FMK 还表现出对组织蛋白酶 B 活性的强大抑制作用 (IC50=6 μM)。 Z-WEHD-FMK 可用于研究细胞凋亡的证据。 | |||||
| GC45193 | Z-YVAD-CMK (trifluoroacetate salt) | - | Caspase | ||
An inhibitor of caspase-1 and caspase-3 | |||||
| GC40556 | Ac-LETD-AFC | 210345-02-1 | Proteolysis | ||
A caspase-8 fluorogenic substrate | |||||
| GC15479 | Ac-IETD-pNA | 219138-21-3 | Peptides | ||
A caspase-8 chromogenic substrate | |||||
| GC13859 | Z-DEVD-AFC | 1135416-11-3 | Neuroscience | ||
A caspase-3 fluorogenic substrate | |||||
| GC13400 | Ac-VDVAD-AFC | 210344-94-8 | Proteolysis | ||
A fluorogenic substrate for caspase-2 | |||||
