关于 "Dopamine Receptor" 的结果39+ 个结果

Foslevodopa 是多巴胺受体 (dopamine receptor) 的激动剂。

(–)-Apomorphine (hydrochloride) is an analytical reference standard categorized as a dopamine receptor agonist.

D3 dopamine receptor agonist; less active enantiomer of 7-OH-DPAT, in comparison with (R)-(+)-7-OH-DPAT

Selective D3 dopamine receptor agonist. Its more active enantiomer is trans-(+)-PD-128907 and less active enantiomer is (-)-PD 128907

Aripiprazole monohydrate is a third-generation antipsychotic with a dopamine receptor-binding profile distinct from other second-generation antipsychotics, used in schizophrenia.

Formally derived from the C-terminal dipeptide of oxytocin., cyclo(Leu-Gly) is active in memory processes. The diketopiperazine blocks the narcotic-induced dopamine receptor supersensitivity.

Tiapride is a drug that selectively blocks D2 and D3 dopamine receptors in the brain and is used to treat a variety of neurological and psychiatric disorders.

Potent and selective dopamine receptor agonist; derivative of Rotigotine (N-0437); * N-0734, N-0434 ((±)-PPHT) and N-0437 are potent and selective DA agonists that lack significant α 2 activity

Naxagolide ((+)-PHNO; Dopazinol) 是一种有效的多巴胺 D2 (dopamine D2) (Dopamine Receptor) 激动剂。Naxagolide 具有用于帕金森病 (PD) 研究的潜力。

Promazine (Romtiazin, Sinophenin) is an antagonist at types 1, 2, and 4 dopamine receptors, 5-HT receptor types 2A and 2C, muscarinic receptors 1 through 5, alpha(1)-receptors, and histamine H1-receptors with antipsychotic effects.

Selective dopamine D4 antagonist; Displayed high affinity (Ki = 10 nM) and selectivity for the D4 receptor expressed in clonal cell lines, lacking measurable affinity for other dopamine receptors, and noradrenalin, serotonin and histamine receptor families (Ki > 2000 nM)

Quetiapine D4 hemifumarate 是 Quetiapine hemifumarate 的氘代物。Quetiapine 是一种 5-HT 受体激动剂，也是一种多巴胺受体 (dopamine receptor) 拮抗剂。具有抗抑郁和抗焦虑作用。

(+)-AJ 76 hydrochloride是一种对突触前受体具有优先作用的多巴胺受体（dopamine receptors, DRs）拮抗剂（hD3、hD4、hD2S、hD2L和rD2受体的pKi值分别为6.95、6.67、6.37、6.21和6.07）。

Pimozide-d4-1 氘代标记的 Pimozide。Pimozide 是 dopamine receptor 的拮抗剂，对 dopamine D2，D3 和 D1 受体的 Ki 值分别为 1.4 nM，2.5 nM 和 588 nM，同时对 α1-adrenoceptor 也有较高亲和性，Ki 值为 39 nM；Pimozide 也是 STAT3 和 STAT5 的抑制剂。

OPC 4392 hydrochloride 是突触前多巴胺受体 (dopamine receptor) 的激动剂和突触后 D2 受体的拮抗剂。OPC 4392 可逆转 Reserpine -诱导的多巴胺积累，抑制 Apomorphine -诱导的小鼠模型中的刻板行为和攀爬行为。